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3-{1-[1-(1,4-dithiepan-6-yl)piperidin-4-yl]-1H-pyrazol-5-yl}-1-(2-methylphenyl)urea
[(3,5-dimethoxyphenyl)methyl]({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)methylamine
3,6-dimethyl-N-{[1-(propan-2-yl)piperidin-3-yl]methyl}-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide
(1S,5R)-6-benzyl-3-[3-(1H-1,2,4-triazol-1-yl)propanoyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
3-(5-{[4-(5-methylfuran-2-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}thiophen-3-yl)prop-2-yn-1-ol
3-{5-[2,2-dimethyl-1-(thiophen-2-yl)cyclopropanecarbonyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
2-ethyl-5-(4-{5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl}piperazine-1-carbonyl)pyrimidine
4-{2-[(4-benzyl-5-{1-[(2-methylphenyl)methyl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}morpholine
5-{[4-(3-propylmorpholine-4-carbonyl)-1,3-oxazol-2-yl]methoxy}isoquinoline
4-methyl-5-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyrimidine
3-methyl-1-[(3-methylphenyl)methyl]-4-[2-(pyridin-3-yl)acetyl]piperazin-2-one
(3S,4S)-1-[3-(3-fluorophenyl)benzoyl]-4-methylpiperidine-3,4-diol
(3S,4R)-1-{[2-(furan-2-yl)phenyl]methyl}-4-(4-methoxyphenyl)-N,N-dimethylpyrrolidin-3-amine
2-ethyl-8-[2-(2,2,3,3-tetrafluoropropoxy)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
N-(furan-2-ylmethyl)-N,1-dimethyl-5-({[4-(trifluoromethyl)phenyl]methyl}amino)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-(butan-2-yl)-4-ethanesulfonamido-N-(pyridin-3-ylmethyl)benzamide
6-(butane-1-sulfonyl)-N-methyl-4-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-2-amine
1-(diethylamino)-3-(2-methoxy-4-{[methyl(pyridin-2-ylmethyl)amino]methyl}phenoxy)propan-2-ol
1-(5-cyclopropyl-1,3-oxazole-4-carbonyl)-3-(4-methylphenoxymethyl)piperidine
3-{2-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}-1-[4-(4-methyl-4H-1,2,4-triazol-3-yl)phenyl]urea
4-{[4-fluoro-3-(trifluoromethyl)phenyl]methyl}-1,3λ6,4-oxathiazinane-3,3-dione
3-[4-(1H-imidazol-2-yl)piperidine-1-carbonyl]-5-methoxybenzoic acid
6-chloro-2-[4-(pyrimidin-2-yloxy)phenyl]-1H-1,3-benzodiazole
2-ethoxy-5-{2-[(oxolan-2-ylmethyl)amino]pyrimidin-4-yl}benzoic acid
2-methyl-3-({4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}methyl)quinoxaline
N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}-3-(pyridin-3-yl)propanamide
5-methyl-3-{[5-(3-methylphenyl)-4-phenyl-1H-imidazol-1-yl]methyl}-1,2-oxazole
5-{6-amino-1H-pyrrolo[2,3-b]pyridin-4-yl}-N-butylfuran-2-carboxamide
(3aS,6aS)-5-(5-methoxy-2,4-dimethylbenzenesulfonyl)-1-methyl-octahydropyrrolo[3,4-b]pyrrole
2-(dimethylamino)-2-(4-fluorophenyl)-N-(2-hydroxyethyl)-N-propylacetamide
2,6-di-tert-butyl-4-[3-(2-hydroxypropan-2-yl)pyrrolidine-1-carbonyl]phenol
2-[4-(1-cyano-1-methylethyl)phenyl]-2-{methyl[(3-methylpyridin-2-yl)methyl]amino}acetic acid
2-[2-(1-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-3-yl)-1H-imidazol-1-yl]acetamide
N-[1-(1H-1,3-benzodiazol-2-yl)ethyl]-3-(2-fluorophenyl)-1H-pyrazole-5-carboxamide
4-{1-[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]piperidin-3-yl}pyrimidine
4-ethyl-1-methyl-3-{1-[6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
1-(4-chloro-2-fluorobenzoyl)-4-(3-methylpyridin-4-yl)-1,4-diazepane
3-(cyclopropylmethyl)-1-(pyridin-4-yl)piperidine-3-carboxylic acid
3-[5-(6-methyl-2-phenylpyrimidin-4-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanoic acid
4-{[(1H-imidazol-2-ylmethyl)(methyl)amino]methyl}-1H-pyrazole-3-carboxylic acid
N-benzyl-2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)-N-(2,2,2-trifluoroethyl)acetamide
3-[5-(2,5-dimethylfuran-3-yl)-1,3,4-oxadiazol-2-yl]-N-(1-phenylethyl)propanamide
4-(3-fluoropyridin-2-yl)-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-[(1-{[2-methyl-4-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-3-yl)methyl]acetamide
N-{2-oxo-2-[3-oxo-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-9-yl]ethyl}acetamide
3-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)-1-(furan-2-ylmethyl)piperidine
1-[(1R,2R,6S,7S)-4-azatricyclo[5.2.1.02,6]decan-4-yl]-3-(2H-1,3-benzodioxol-5-yl)propan-1-one
5-[(2-{4-[(dimethylamino)methyl]phenyl}piperidin-1-yl)methyl]-N,N-dimethyl-1,3-thiazol-2-amine
1-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-4-(2-fluorophenoxy)piperidine-4-carboxylic acid
2-[ethyl(methyl)amino]-1-[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidin-1-yl]ethan-1-one