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2-[5-(azepan-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methylacetamide
1-benzyl-4-({[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}amino)pyrrolidin-2-one
1-(2-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethyl]amino}pyrimidin-4-yl)pyrrolidin-3-ol
{2-[3-(4-fluorophenoxymethyl)piperidin-1-yl]quinolin-3-yl}methanol
N-[(2-fluorophenyl)methyl]-N-(2-hydroxyethyl)-1,2-oxazole-3-carboxamide
N-(1-methylpiperidin-4-yl)-N-(pyridin-4-ylmethyl)-3-(thiophen-3-yl)propanamide
methyl 4-{3-[(4-methylpiperazin-1-yl)methyl]-1,2,4-oxadiazol-5-yl}benzoate
3-(3-fluorophenyl)-N-[(4-methylphenyl)(pyridin-4-yl)methyl]-1H-pyrazole-4-carboxamide
3-[1-(1-benzofuran-2-ylmethyl)piperidin-4-yl]-N-[(1-ethylpyrrolidin-2-yl)methyl]propanamide
(3E)-5,5-dimethyl-2-[methyl({[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl})amino]hex-3-enoic acid
(3R,4R)-1-(3-chloro-4-methoxybenzoyl)-3-cyclobutyl-4-methylpyrrolidin-3-ol
4-[4-(2-chloro-4-fluorobenzoyl)-5-methyl-2-oxopiperazin-1-yl]benzonitrile
methyl 5-[(4-hydroxybutan-2-yl)amino]-3-(2-methylbutanamido)-1-(oxolan-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-[(4-chlorophenyl)methyl]-8-[2-(oxolan-3-yl)ethyl]-2,8-diazaspiro[4.5]decan-3-one
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-2-(6-methyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-4-yl)acetamide
1-(2-methylpropyl)-4-[4-(thiophen-3-yl)-1H-imidazol-2-yl]pyrrolidin-2-one
1-{1-[(2-fluoro-5-methoxyphenyl)methyl]piperidin-3-yl}-4-(2-methoxyphenyl)piperazine
[(2S)-1-[(3-chlorothiophen-2-yl)methyl]pyrrolidin-2-yl]methanol
4-phenyl-3-(piperidin-3-yl)-1-(1,3-thiazol-2-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[(5-methyl-1H-1,3-benzodiazol-2-yl)methyl]-2-[1-(3-methylbutyl)-3-oxopiperazin-2-yl]acetamide
9-(cyclopropylmethyl)-N,N,1-trimethyl-10-oxo-1,4,9-triazaspiro[5.6]dodecane-4-sulfonamide
(4aS,8aR)-1-[3-(1H-imidazol-1-yl)propyl]-6-(1-methyl-1H-pyrrole-2-carbonyl)-decahydro-1,6-naphthyridin-2-one
2-(dimethylamino)-2-(2-methylphenyl)-1-[4-(1H-pyrrole-2-carbonyl)piperazin-1-yl]ethan-1-one
N-{[6-chloro-4-(pyrrolidin-1-yl)quinazolin-2-yl]methyl}-2,3-dihydro-1,4-benzodioxine-6-sulfonamide
2-{1-butyl-5-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-3-yl}acetamide
1-[3-(3-methoxyphenyl)benzoyl]azepan-4-amine
2-(2,3-dihydro-1H-inden-1-yl)-N-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}acetamide
1-[(3S,4R)-3-(dimethylamino)-4-(4-methylphenyl)pyrrolidin-1-yl]-2-(2-methyl-1H-1,3-benzodiazol-5-yl)ethan-1-one
[1-({[2-(ethoxymethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]amino}methyl)cyclobutyl]methanol
1-(oxan-4-yl)-N-{[3-(pyrimidin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidine-3-carboxamide
(3R,5S)-5-[4-(3-methylpyridin-2-yl)piperazine-1-carbonyl]pyrrolidin-3-ol
2-{4-[1-(2-methoxyacetyl)piperidine-3-carbonyl]piperazin-1-yl}benzonitrile
2-(2-hydroxyethyl)-8-[5-(propan-2-yl)pyrimidin-4-yl]-2,8-diazaspiro[5.5]undecan-3-one
ethyl 3-{[3-(4-phenylbenzoyl)piperidine-1-carbonyl]amino}propanoate
2-(naphthalen-1-ylmethyl)-4-(1,3-thiazol-2-ylmethyl)morpholine
3-cyclobutyl-4-(quinolin-2-yl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
1-(cyclohexylmethyl)-3-{1,4-dioxa-8-azaspiro[4.5]decan-8-ylmethyl}-3-hydroxypiperidin-2-one
N-[1-(5-{[2-(4-fluorophenoxy)ethyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)ethyl]thiophene-2-sulfonamide
N-[1-(3-methyl-1,2,4-oxadiazol-5-yl)ethyl]-2-(pyridin-4-yl)quinoline-4-carboxamide
3-ethyl-6-[4-(morpholin-4-yl)piperidine-1-carbonyl]-3H-imidazo[4,5-b]pyridin-2-amine
1-[(1-{[2-(2,4-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-3-yl)methyl]pyrrolidin-2-one
3-amino-N-{[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methylbenzamide
1-{octahydropyrrolo[1,2-a]piperazin-2-yl}-2-(phenylsulfanyl)ethan-1-one
5-(oxan-4-ylmethyl)-7-oxo-4H,7H-pyrazolo[1,5-a]pyrimidine-3-carbonitrile
2-(2-{3,9-diazaspiro[5.5]undecan-3-ylmethyl}phenoxy)acetic acid
N-(4,7-dimethyl-2-oxo-2H-chromen-6-yl)-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
{1-[6-amino-2-(morpholin-4-yl)pyrimidin-4-yl]-3-(prop-2-en-1-yl)piperidin-3-yl}methanol
7-chloro-2-{[2-(pyridin-2-yl)piperidin-1-yl]methyl}-4H-pyrido[1,2-a]pyrimidin-4-one
2-(2-{1-[2-(pyrrolidin-1-yl)benzoyl]piperidin-3-yl}-1H-imidazol-1-yl)acetamide
1-{2-[2-(3,4-dichlorophenyl)morpholin-4-yl]-2-oxoethyl}-3,3-dimethylurea