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1-[(3S,4R)-3,4-dihydroxy-4-methylpiperidin-1-yl]-2-(2-methyl-1H-1,3-benzodiazol-5-yl)ethan-1-one
N-[2-(azepan-1-yl)ethyl]-N-methyl-2-oxo-1-phenylpyrrolidine-3-carboxamide
N-cyclohexyl-3-[(1-methyl-2-oxo-1,2-dihydroquinolin-4-yl)formamido]propanamide
4,6-dimethyl-2-{2-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}pyridine-3-carbonitrile
6-(3-chlorophenyl)-N-ethyl-N-methyl-8-oxo-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
2-(furan-3-yl)-2-[methyl(1,3-thiazol-2-ylmethyl)amino]acetic acid
8-(5-ethyl-1,3-oxazole-4-carbonyl)-3-(2-ethylbutyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
5-{[2,5-dimethoxy-4-(methylsulfanyl)phenyl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
3-benzyl-5-(3,4-dihydro-2H-1-benzopyran-3-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
7-(morpholin-4-ylmethyl)-4-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-(1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}piperidin-4-yl)-1-(4-phenylpiperazin-1-yl)propan-1-one
methyl[(1S)-2-methyl-1-[3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazol-5-yl]propyl]amine
1'-(1H-1,2,3-benzotriazole-5-carbonyl)-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
(2R)-2-amino-N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N,4-dimethylpentanamide
1-{2-oxo-2-[2-(1,3-thiazol-2-yl)piperidin-1-yl]ethyl}-1,2,3,4-tetrahydroquinolin-2-one
N-{4-[2-(5-amino-3-methyl-1H-pyrazol-1-yl)acetamido]-2-methoxyphenyl}-2,2-dimethylpropanamide
2-(4-ethylpiperazin-1-yl)-N-[1-(2-fluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]acetamide
1-[3-(1H-imidazol-1-ylmethyl)piperidin-1-yl]-4-(thiophen-2-yl)butan-1-one
3-fluoro-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-N-(pyridin-4-ylmethyl)pyridine-4-carboxamide
2,6-dimethyl-N-[1-(morpholin-4-ylmethyl)cyclopentyl]pyridine-4-carboxamide
N-methyl-N-[2-(2-methylphenyl)-1-{1-[(2E)-3-(thiophen-2-yl)prop-2-enoyl]piperidin-4-yl}ethyl]cyclobutanecarboxamide
8-(6-methylquinazolin-4-yl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
4-[2-(2,3-dichloro-4-methylphenyl)-1H-imidazol-1-yl]piperidine
2-{[4-ethyl-4-(hydroxymethyl)piperidin-1-yl]sulfonyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
2-(5-methyl-1H-pyrazol-1-yl)-1-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
N-[(7S,8aS)-2-methyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-[2-(propan-2-yl)-1H-1,3-benzodiazol-1-yl]acetamide
3-({[7-fluoro-2-oxo-1-(2-phenylethyl)-1,2-dihydroquinolin-3-yl]methyl}amino)-1λ6-thiolane-1,1-dione
5-{3-[5-(1H-imidazol-2-yl)-4-phenyl-1H-imidazol-1-yl]propyl}-1H-1,2,3,4-tetrazole
(4aS,7aR)-1-(2,4-dimethylbenzoyl)-4-(2-methoxyacetyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
8-(3-methoxypropanoyl)-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
1-(1-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}pyrrolidin-3-yl)-3,5-dimethyl-1H-pyrazole
2-(1-{[5-methyl-2-(3-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}piperidin-3-yl)-1,3-benzoxazole
N-methyl-3-(2-methylpropyl)-N-[1-(4-methylpyridin-2-yl)propan-2-yl]-1,2-oxazole-5-carboxamide
(benzylsulfamoyl)(methyl){[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}amine
3-{2-[(oxolan-2-ylmethyl)(thiophen-3-ylmethyl)amino]ethyl}-2,3-dihydro-1,3-benzoxazol-2-one
6-[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]pyridin-2-amine
(1S,5R)-6-(cyclopropylmethyl)-3-(2,3-difluoro-4-methoxybenzoyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-(4-methylpyridine-3-carbonyl)pyrrolidine-3-carboxylic acid
1-[(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(pyridin-2-yl)propan-1-one
3-(3-methoxyphenyl)-N-methyl-N-(quinolin-2-ylmethyl)-1H-pyrazole-5-carboxamide
6-[1-(4-chlorophenyl)-3-cyclopropyl-1H-1,2,4-triazol-5-yl]-2,2-dimethyl-3,4-dihydro-2H-pyran-4-one
ethyl 3-(2-methoxyethyl)-1-{[2-(4-methoxyphenyl)pyrimidin-5-yl]methyl}piperidine-3-carboxylate
N-[(4-sulfamoylphenyl)methyl]imidazo[1,2-a]pyrimidine-2-carboxamide
(4aS,8aR)-1-(3-aminopropyl)-6-[6-(trifluoromethyl)pyridin-2-yl]-decahydro-1,6-naphthyridin-2-one
(4aS,8aS)-2-{[2-(cyclopentyloxy)phenyl]methyl}-decahydro-2,7-naphthyridin-4a-ol
4-(4-{8-benzyl-2,8-diazaspiro[5.5]undecane-2-carbonyl}-5-cyclopropyl-1H-pyrazol-1-yl)-3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaene
2-{4-[2-(2-methylphenyl)pyrrolidine-1-carbonyl]piperidin-1-yl}acetamide
2-methoxy-4-(3,4,5-trimethoxyphenyl)pyridine-3-carbonitrile
N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-3-(2-fluorophenyl)-1H-pyrazole-5-carboxamide
N-[(2-methoxyphenyl)methyl]-N-{[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}cyclopropanamine