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N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-5-ethylpyrimidin-2-amine
4-[(6-methylpyridin-3-yl)oxy]-1-(thiophen-3-ylmethyl)piperidine-4-carboxylic acid
N,4-diethyl-N-[2-hydroxy-2-(3-hydroxyphenyl)ethyl]-2-methyl-1,3-thiazole-5-carboxamide
8-[(1-methyl-1H-imidazol-2-yl)methyl]-3-{2-[4-(propan-2-yl)piperazin-1-yl]ethyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-{1-oxa-8-azaspiro[4.5]decan-3-yl}-7-oxo-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
N-methyl-2-(3-methyl-1,2-oxazol-5-yl)-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}acetamide
1-(furan-3-ylmethyl)-4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine
5-{[benzyl(methyl)amino]methyl}-N-[2-(pyrrolidin-1-yl)ethyl]-1,2-oxazole-3-carboxamide
N-methyl-N-[(5-methylfuran-2-yl)methyl]-4-(4H-1,2,4-triazol-4-yl)benzamide
N-(3-hydroxy-3-methylbutyl)-N-methyl-2-[3-oxo-1-(2-phenylethyl)piperazin-2-yl]acetamide
1-(3-{octahydro-1H-pyrido[1,2-a]piperazine-2-sulfonyl}benzoyl)pyrrolidine
(2S,4S)-N-ethyl-4-[2-(3-hydroxyphenyl)acetamido]-1-(1H-imidazol-2-ylmethyl)pyrrolidine-2-carboxamide
1-(4-methoxyphenyl)-N-methyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]cyclopropane-1-carboxamide
5-{[4-(azepane-1-carbonyl)-1,3-oxazol-2-yl]methoxy}isoquinoline
4-{2-[4-(1H-1,2,3,4-tetrazol-1-yl)phenoxy]acetyl}-1,4-diazepan-2-one
N-(1,4-dioxan-2-ylmethyl)-3-(4-methoxyphenyl)-N-methyl-5-(1H-1,2,3,4-tetrazol-1-yl)benzamide
{[2-(3-chlorophenyl)-8-methylquinolin-3-yl]methyl}(methyl)(pyrimidin-4-ylmethyl)amine
3-[(3R,4R)-3-(hydroxymethyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidine-1-carbonyl]-4-methylbenzene-1-sulfonamide
4-(3-propyl-1H-pyrazole-4-carbonyl)-2-(trifluoromethyl)morpholine
N-[3-(propan-2-yloxy)propyl]-5-[(quinolin-6-yloxy)methyl]-1,2-oxazole-3-carboxamide
(3S,4R)-1-{[6-(dimethylamino)pyridin-3-yl]methyl}-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
2-ethyl-8-(3-fluoropyridin-4-yl)-2,8-diazaspiro[4.5]decan-3-one
5-(3-chloro-4-methoxyphenyl)pyrimidin-2-amine
2-[4-(2H-1,3-benzodioxol-5-yl)-3-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl]-N-[2-(pyridin-3-yl)ethyl]acetamide
2-ethyl-N-[3-(4-methylphenyl)phenyl]-3-oxopiperazine-1-carboxamide
1-{4-[(2,3-dihydroxypropyl)amino]-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
N-(1H-indol-4-ylmethyl)-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
N-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}-1-(pyrimidin-2-yl)piperidin-3-amine
2-methyl-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-6-(propan-2-yl)pyrimidin-4-amine
N,N-dimethyl-2-phenyl-2-[(5-propyl-1,3,4-oxadiazol-2-yl)amino]acetamide
3-[6-(4-methylpiperazine-1-carbonyl)pyrazin-2-yl]quinoline
ethyl 1-(1-methyl-2-oxo-1,2-dihydroquinolin-4-yl)-5-[({spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-5-ylmethyl}amino)methyl]-1H-pyrazole-4-carboxylate
1-[2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
N-{2-[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]ethyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carboxamide
N-[2-(2-hydroxyethoxy)ethyl]-2-methyl-1-benzofuran-5-carboxamide
1-[(2-fluorophenyl)methyl]-N-[2-(2-hydroxyethoxy)ethyl]-6-oxopiperidine-3-carboxamide
1-(4-{[methyl(quinolin-4-ylmethyl)amino]methyl}phenoxy)-3-(piperidin-1-yl)propan-2-ol
(2S,4R)-4-amino-N-methyl-1-[(3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)sulfonyl]pyrrolidine-2-carboxamide
N-cyclopropyl-2-methyl-N-[(3-methylthiophen-2-yl)methyl]-6-(piperidin-4-yl)pyrimidin-4-amine
[(3R,4S)-4-(morpholin-4-ylmethyl)-1-(quinolin-2-ylmethyl)pyrrolidin-3-yl]methanol
N-(adamantan-1-yl)-3-{[4-(aminomethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidine-1-carboxamide
1-(2-methoxyethyl)-8-(oxan-4-yl)-3-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-(2-methoxypyridin-3-yl)-1,3-benzothiazol-2-amine
5-[3-(4-ethyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-4-methyl-2-(pyridin-3-yl)pyrimidine
3-{[1-(2-methyl-6-propylpyrimidin-4-yl)piperidin-4-yl]amino}-1λ6-thiolane-1,1-dione
3,4,7-trimethyl-N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-1H-indole-2-carboxamide
1-methyl-N-(3-methyl-1,1-dioxo-1λ6-thiolan-3-yl)-1H-imidazole-2-carboxamide
5-(methoxymethyl)-N-methyl-N-[(1-methylpiperidin-2-yl)methyl]-1,3,4-oxadiazole-2-carboxamide
N-[2-(3-methoxyphenyl)ethyl]-2-{1-[(2-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
N-(1,2-oxazol-3-ylmethyl)-5-oxo-1-[4-(propan-2-yl)phenyl]pyrrolidine-3-carboxamide