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(furan-2-ylmethyl)(1H-imidazol-4-ylmethyl)[2-(morpholin-4-yl)ethyl]amine
5-(2-methyl-4-oxo-4,5,6,7-tetrahydro-1-benzofuran-3-carbonyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
2-{1-[(2-chloro-4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[3-(2-methyl-1H-imidazol-1-yl)propyl]acetamide
1-(cyclobutylmethyl)-4-[(2,3,4-trimethoxyphenyl)methyl]piperazine
ethyl 2-{1-[3-(morpholin-4-yl)benzoyl]piperidin-2-yl}acetate
3-[(2,6-dioxopiperidin-1-yl)methyl]-N-methyl-1,2,4-oxadiazole-5-carboxamide
N-{[4-amino-6-(dimethylamino)-1,3,5-triazin-2-yl]methyl}-2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)acetamide
1-ethyl-N-{[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]methyl}-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
1-{3-[(3,4-dimethylphenyl)amino]piperidin-1-yl}-4-(4-fluorophenyl)butane-1,4-dione
4-cyclopentyl-N-[1-(pyrazin-2-yl)propan-2-yl]pyrimidin-2-amine
3-[2-(3-methoxyphenyl)piperidine-1-carbonyl]-2-(methylsulfanyl)pyridine
{3-[(1-methyl-1H-imidazol-5-yl)methyl]-9-(oxan-4-yl)-3,9-diazaspiro[5.5]undecan-1-yl}methanol
1-[2-(1-{2-[4-(dimethylamino)phenyl]acetyl}piperidin-2-yl)ethyl]pyrrolidin-2-one
5-(2-methoxyphenoxymethyl)-N-[(3-methylphenyl)methyl]-1H-pyrazole-3-carboxamide
2-hydroxy-N-[2-(3-phenylpropoxy)phenyl]acetamide
(3aS,6aS)-2-cyclobutanecarbonyl-5-[(2-methyl-1,3-thiazol-4-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-{3-[(dimethylsulfamoyl)amino]phenyl}-3-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}urea
1-{5,7-dimethylpyrazolo[1,5-a]pyrimidine-3-carbonyl}-4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine
4-{6-amino-1H-pyrrolo[2,3-b]pyridin-4-yl}-3-fluorobenzene-1-sulfonamide
6-methyl-3-[1-(2-methylpyridin-4-yl)-3-phenyl-1H-1,2,4-triazol-5-yl]-1,2-dihydropyridin-2-one
N-{1-[1-(2,5-dimethylfuran-3-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}-3-fluorobenzamide
N-[2-(N-methylmethanesulfonamido)ethyl]-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
N-methyl-2-phenyl-N-[(trimethyl-1H-pyrazol-4-yl)methyl]imidazo[1,2-a]pyridine-6-carboxamide
N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]-2-[3-oxo-1-(pyridin-3-ylmethyl)piperazin-2-yl]acetamide
5-{[3-(1-benzyl-1H-imidazol-2-yl)piperidin-1-yl]methyl}-1,2,4-oxadiazole-3-carboxamide
1-[(4-methyl-1H-imidazol-5-yl)methyl]-3-(1-methyl-1H-imidazole-2-carbonyl)piperidine
3-[1-(2,1,3-benzoxadiazol-4-ylmethyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)propanamide
N-(3-hydroxyphenyl)-4-[3-(2-methylpiperidin-1-yl)azetidin-1-yl]-4-oxobutanamide
3-butanamido-4-methyl-N-[1-(pyridin-4-yl)propan-2-yl]benzamide
2,6-difluoro-3-methoxy-N-methyl-N-(1H-pyrazol-3-ylmethyl)benzamide
2-{3-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]piperidin-1-yl}-2-oxo-N-(propan-2-yl)acetamide
(1R)-2-{3-[3-(2,5-dimethylpyrimidin-4-yl)phenyl]-1H-pyrazol-1-yl}-1-phenylethan-1-ol
N-{1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl}-4-(propan-2-yl)-1,2,3-thiadiazole-5-carboxamide
1-({[2-(2-chlorophenyl)-2-(dimethylamino)ethyl]carbamoyl}methyl)piperidine-4-carboxamide
ethyl 3-(2-phenoxyethyl)-1-[1-(pyridin-2-ylmethyl)piperidin-4-yl]piperidine-3-carboxylate
3-(2-methoxyphenyl)-5-(trimethyl-1H-pyrazol-4-yl)-1,2,4-oxadiazole
1-(3-{[4-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)-2-(3-methoxyphenoxy)ethan-1-one
2-(4-{[(3S,4S)-3-(dimethylamino)-4-hydroxypyrrolidin-1-yl]methyl}phenoxy)acetic acid
(4aS,8aR)-1-[2-(methylamino)ethyl]-6-(9H-purin-6-yl)-decahydro-1,6-naphthyridin-2-one
3,4-dimethyl-N-(5-oxo-1-phenylpyrrolidin-3-yl)benzene-1-sulfonamide
1-{3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl}-2-(methylsulfanyl)ethan-1-one
4-(4-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidine-1-carbonyl)benzonitrile
N-({2-methoxy-5-oxo-6-[2-(pyridin-2-yl)ethyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)benzamide
N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-2-(dimethylamino)-N-methyl-2-(4-methylphenyl)acetamide
N-(1-phenyl-1H-pyrazol-5-yl)-2-[3-(thiophen-3-yl)-1H-pyrazol-1-yl]acetamide
[(1-cyclopentylpiperidin-4-yl)methyl][(2,4-difluorophenyl)methyl](oxolan-2-ylmethyl)amine
4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]-1-(2-phenylpropyl)piperidine
1-(cyclohexylmethyl)-3-hydroxy-3-(pyrrolidin-1-ylmethyl)piperidin-2-one
1-[(3S,7S)-3-(hydroxymethyl)-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-trien-5-yl]-2-(pyridin-3-yl)ethan-1-one
N-ethyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1-(propan-2-yl)piperidine-4-carboxamide