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4-acetyl-N-{1-[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}benzene-1-sulfonamide
14-(2-propoxyphenyl)-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
(2S,4R)-N-cycloheptyl-1-[(5-methoxy-2-methyl-3-phenyl-1-benzofuran-6-yl)methyl]-4-(1H-1,2,3,4-tetrazol-1-yl)pyrrolidine-2-carboxamide
1-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-[(5-methyl-1,3,4-oxadiazol-2-yl)sulfanyl]ethan-1-one
2-{3-methyl-4-[4-(2-methylpropyl)phenyl]-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-1-yl}acetic acid
(3R,9aR)-8-(3-chlorobenzoyl)-3-(hydroxymethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
(2R,3R,6R)-5-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-[1-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)-2-methylpropyl]-2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
4-[(4-methyl-1H-imidazol-5-yl)methyl]-N-(2-phenoxyethyl)morpholine-2-carboxamide
4-(5-{1-[2-(propan-2-yl)-1H-imidazol-1-yl]ethyl}-1,2,4-oxadiazol-3-yl)pyridine
3-{2-[1-(2H-1,3-benzodioxol-5-ylmethyl)-1H-1,2,4-triazol-5-yl]ethyl}pyridine
methyl (2S)-1-(4-{[2-(cyclohex-1-en-1-yl)ethyl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carbonyl)pyrrolidine-2-carboxylate
(4aS,8aS)-2-{[2-fluoro-4-(trifluoromethyl)phenyl]methyl}-decahydro-2,7-naphthyridin-4a-ol
1-[3-hydroxy-3-(pyrrolidin-1-ylmethyl)piperidin-1-yl]-2-(pyridin-4-ylsulfanyl)ethan-1-one
1-benzyl-4-[2-(1H-pyrazol-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-1H-pyrazole
(1S,5R)-3-cyclobutanecarbonyl-6-[(4-methylthiophen-2-yl)sulfonyl]-3,6-diazabicyclo[3.2.2]nonane
2-cyclopropyl-8-[(1-methyl-1H-indol-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}-N-[4-(1H-pyrazol-1-yl)butan-2-yl]benzamide
2-chloro-4-{[3-(2-hydroxyethyl)-4-[(6-methylpyridin-2-yl)methyl]piperazin-1-yl]methyl}-6-methoxyphenol
methyl 2-(ethylsulfamoyl)-6-{1-[3-(trifluoromethyl)phenyl]propan-2-yl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N,N-dimethyl-6-[(1R,6S)-9-methyl-3,9-diazabicyclo[4.2.1]nonan-3-yl]pyridine-3-carboxamide
N-(4-fluorophenyl)-1-(5-methyl-1,2-oxazole-3-carbonyl)piperidin-3-amine
4-(2-{[(7-methoxynaphthalen-2-yl)oxy]methyl}-1,3-oxazole-4-carbonyl)-1λ6-thiomorpholine-1,1-dione
methyl (1S,3S,3aR,6aS)-1-(hydroxymethyl)-5-methyl-4,6-dioxo-3-[4-(1H-pyrazol-1-yl)phenyl]-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-3-propyl-1H-pyrazole-4-carboxamide
1-[(1R,3S)-1-hydroxy-3-(2-hydroxyethoxy)-7-azaspiro[3.5]nonan-7-yl]-2-methoxyethan-1-one
1-{2-[1-(2-hydroxybutyl)-3-(thiophen-2-ylmethyl)-1H-1,2,4-triazol-5-yl]ethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
5-cyclopropyl-1-methyl-4-{[3-(naphthalen-1-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-1H-pyrazole
N-(1-{1-[2-(3-methylphenyl)acetyl]piperidin-4-yl}-1H-pyrazol-5-yl)cyclopropanecarboxamide
2-cyclopropyl-N-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-4-hydroxy-N-methylpyrimidine-5-carboxamide
[2-(1-{[4-fluoro-3-(trifluoromethyl)phenyl]methyl}piperidin-2-yl)ethyl]dimethylamine
8-[4-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
N,6-dimethyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
1-(2,3-dihydro-1H-isoindol-2-yl)-2-(morpholin-4-yl)-2-(pyridin-3-yl)ethan-1-one
1-[(1S,5R)-3-benzoyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(pyridin-3-yl)propan-1-one
3-{3-[5-(2-methyl-1H-imidazol-4-yl)-4-phenyl-1H-imidazol-1-yl]propoxy}pyridine
5-(2-fluorophenoxymethyl)-N-(3-hydroxypropyl)-N-methyl-1H-pyrazole-3-carboxamide
2-cyclopropanecarbonyl-7-[(4-propoxyphenyl)methyl]-2,7-diazaspiro[4.5]decane
(3aS,6aS)-2-cyclobutanecarbonyl-5-(6-ethyl-5-fluoropyrimidin-4-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-(2-methoxyethyl)-3-methyl-N-{[2-(2-methylphenyl)-7-(methylsulfanyl)quinolin-3-yl]methyl}thiophene-2-carboxamide
1-(3-chlorophenyl)-4-[1-(difluoromethyl)-1H-pyrazole-5-carbonyl]piperazin-2-one
9-[2-(1H-imidazol-1-yl)ethyl]-2-(3-methoxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
1-(4-methoxyphenyl)-4-(2-methyl-5-oxo-1,4-diazepan-1-yl)butane-1,4-dione
7-chloro-N-ethyl-3,5-dimethyl-N-(oxan-4-ylmethyl)-1-benzofuran-2-carboxamide
3-tert-butyl-1-methyl-4-[2-(propan-2-yl)-1,3-oxazol-4-yl]-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-[6,6-dimethyl-1-(2-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-oxo-2,3-dihydro-1H-imidazole-4-carboxamide
1,4,6-trimethyl-2-oxo-N-{1-[4-(1H-1,2,4-triazol-1-yl)phenyl]ethyl}-1,2-dihydropyridine-3-carboxamide
methyl({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl){[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}amine
3-(4-fluorophenyl)-4-(3,4,7-trimethyl-1H-indole-2-carbonyl)piperazin-2-one
2-[(2,6-dichlorophenyl)methyl]-4-hydroxy-N-(oxan-4-ylmethyl)pyrimidine-5-carboxamide