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4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(2-methyl-1H-pyrrole-3-carbonyl)piperidine
2-(2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]acetamide
(9aS)-2-[(5-ethylfuran-2-yl)methyl]-octahydro-1H-pyrrolo[1,2-a][1,4]diazepine
N-[2-(2-fluorophenyl)-1-{1-[(2-hydroxy-3-methoxyphenyl)methyl]piperidin-4-yl}ethyl]-N-methylthiophene-2-carboxamide
(1S,6R)-9-(1-benzylpiperidin-4-yl)-3,9-diazabicyclo[4.2.1]nonan-4-one
1-{2-[2-(cyclohexylmethyl)morpholin-4-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
(3R,4S)-4-{4-[1-(4,6-dimethylpyrimidin-2-yl)piperidin-4-yl]-1,4-diazepan-1-yl}oxolan-3-ol
N-[(1-phenylcyclopentyl)methyl]pyridazine-4-carboxamide
2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]-1-[3-(1H-imidazol-2-yl)piperidin-1-yl]ethan-1-one
1-methanesulfonyl-3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine
1-[2-({[4-(trifluoromethyl)pyrimidin-2-yl]amino}methyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl]ethan-1-one
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-2-(dimethyl-1,3-thiazol-5-yl)acetamide
({3-methoxy-2-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)({[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl})amine
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-2-(2,4-dimethyl-6-oxo-1,6-dihydropyrimidin-5-yl)-N-methylacetamide
8-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-[2-(4-methoxyphenyl)ethyl]-3-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[2-(dimethylamino)ethyl]-5-(pyridin-4-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
2-hydroxy-N-{[(3S,4S)-3-hydroxypiperidin-4-yl]methyl}-5-(1H-pyrrol-1-yl)benzamide
methyl 4-[4-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)piperazin-1-yl]benzoate
1-[(2,3-difluorophenyl)methyl]-4-{1-[(3-methyl-1H-pyrazol-5-yl)methyl]pyrrolidin-3-yl}piperidine
(2S,6S)-1-{[2-(2,3-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-methyl-2,6-bis(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine
2-(2-oxo-1,2,5,6,7,8-hexahydroquinoline-3-carbonyl)-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
5-(3-acetyl-2-fluorophenyl)-N-butylfuran-2-carboxamide
methyl 9-(cyclopentyloxy)-7-oxo-3-[3-(1H-1,2,4-triazol-1-yl)propanoyl]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
(1-{[(1H-1,3-benzodiazol-2-ylmethyl)(methyl)amino]methyl}cyclopentyl)methanol
4-[(2-methylprop-2-en-1-yl)oxy]-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]benzamide
N-({5-[4-(methylamino)pyrimidin-2-yl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)methanesulfonamide
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-2-methyloxane-2-carboxamide
N-[2-(4-methyl-1H-imidazol-2-yl)ethyl]-2-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
N-(1,3-benzothiazol-2-ylmethyl)-1-ethyl-3-(morpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-{3-[3-(hydroxymethyl)-3-(prop-2-en-1-yl)piperidin-1-yl]-3-oxopropyl}piperidin-2-one
8-[6-(dimethylamino)pyrazin-2-yl]-2-(2-methylpropyl)-2,8-diazaspiro[4.5]decan-3-one
N-{1-azabicyclo[2.2.2]octan-3-yl}-1-cyclopropyl-1H-pyrrole-2-carboxamide
N,N-dimethyl-4-{4-[(pyridin-2-ylmethyl)amino]piperidin-1-yl}-5,6,7,8-tetrahydroquinazolin-2-amine
5-ethyl-N-methyl-N-[(trimethyl-1H-pyrazol-4-yl)methyl]pyrimidin-2-amine
(4-{dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)methanol
2-methyl-4-{3-[3-(morpholine-4-carbonyl)piperidine-1-carbonyl]phenyl}butan-2-ol
(3R,4R)-1-[(3-chlorophenyl)methyl]-4-(4-hydroxypiperidin-1-yl)piperidin-3-ol
6-methyl-2-phenyl-N-[1-(pyridin-2-ylmethyl)piperidin-3-yl]pyrimidin-4-amine
9-(5-chloronaphthalene-1-carbonyl)-2-methyl-2,9-diazaspiro[5.5]undecan-3-one
4-[(5-{[(5-chlorothiophen-2-yl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidine
9-[4-(dimethylamino)pyrimidin-2-yl]-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
(1S,5R)-3-[5-(1H-imidazol-1-ylmethyl)furan-2-carbonyl]-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
3-[2-(1-cyclopentylpiperidin-2-yl)ethyl]-8-methoxy-3,4-dihydroquinazolin-4-one
1-(5-ethyl-1,3-oxazole-4-carbonyl)-3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidine
2-phenyl-1-{1-[2-(4H-1,2,4-triazol-4-yl)pyridine-4-carbonyl]piperidin-4-yl}ethan-1-ol
5-chloro-N-[5-oxo-1-(propan-2-yl)pyrrolidin-3-yl]thiophene-2-carboxamide
N-{[7-chloro-2-(4-hydroxypiperidin-1-yl)quinolin-3-yl]methyl}-2-(dimethyl-1,2-oxazol-4-yl)-N-[2-(4-fluorophenyl)ethyl]acetamide
3-(2-oxo-2-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}ethyl)-3,4-dihydroquinazolin-4-one
2-(2-chlorophenoxy)-1-[3-hydroxy-3-(pyrrolidin-1-ylmethyl)piperidin-1-yl]ethan-1-one
4-hydroxy-N-(oxolan-2-ylmethyl)-2-(pyridin-2-yl)pyrimidine-5-carboxamide