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4-(propan-2-yl)-N-{[1-(propan-2-yl)-1H-1,3-benzodiazol-2-yl]methyl}-1,3-thiazole-2-carboxamide
4-[4-cyclopropyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(1H-imidazol-4-ylmethyl)piperidine
2-({6-[4-(4-cyclopentyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]pyrimidin-4-yl}amino)ethan-1-ol
1-(2-methylpropyl)-4-(1-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}pyrrolidin-3-yl)piperidine
4-{[(4-ethyl-1,3-thiazol-2-yl)methyl]amino}-N-(pyridin-4-ylmethyl)pyridine-2-carboxamide
4-{[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1-[(4-methylphenyl)methyl]piperazin-2-one
5-methyl-6-[4-(propan-2-yl)piperazine-1-carbonyl]-N-[1-(thiophen-2-yl)ethyl]thieno[2,3-d]pyrimidin-4-amine
N-(cyclohexylmethyl)-N-ethyl-5-[(4-ethylpiperazin-1-yl)methyl]-1,2-oxazole-3-carboxamide
N-phenyl-1-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-3-amine
2-[(3S)-3-hydroxypyrrolidin-1-yl]-1-methyl-N-{2-[(2S)-pyrrolidin-2-yl]ethyl}-1H-1,3-benzodiazole-5-carboxamide
methyl[3-(methylsulfanyl)propyl][(3-phenyl-1,2-oxazol-5-yl)methyl]amine
5-methyl-1-[2-(5-methyl-4H-1,2,4-triazol-3-yl)ethyl]-5-phenylpiperidin-2-one
2-(morpholin-4-yl)-2-(4-{[(propan-2-yl)carbamoyl]amino}phenyl)acetic acid
N-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-3-{[(3R)-3-hydroxypyrrolidin-1-yl]sulfonyl}benzamide
4-({1-[1-(2-methylpentyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}methyl)morpholine
5-[3-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)propanoyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
5-(3-chloro-4-fluorophenyl)-3-methyl-1H-1,2,4-triazole
(3S,4R)-4-methyl-3-(2-methylpropyl)-1-[5-(morpholine-4-carbonyl)pyridin-2-yl]piperidin-4-ol
methyl[(4-phenyl-1,3-thiazol-2-yl)methyl](pyridin-2-ylmethyl)amine
1-methyl-5-[(3-methylbutyl)amino]-N-(pyridin-4-ylmethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
(4aS,8aR)-6-[4-(1H-imidazol-1-yl)butanoyl]-1-(2-methylpropyl)-decahydro-1,6-naphthyridin-2-one
N-butyl-1-ethyl-N-methyl-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
[3-(3-methoxypropyl)-1-(1-methylcyclopentanecarbonyl)piperidin-3-yl]methanol
N-[(3S)-2-oxoazepan-3-yl]-2-(phenoxymethyl)-1,3-oxazole-4-carboxamide
1-(furan-3-carbonyl)-N-[4-(3-methylphenyl)phenyl]piperidine-4-carboxamide
methyl[(3-methyl-1,2-oxazol-5-yl)methyl]{[2-(3-methylphenyl)pyrimidin-5-yl]methyl}amine
(2R,3S,6R)-5-(3,5-difluoropyridine-2-carbonyl)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
(3R,4R)-1-[3-(hydroxymethyl)quinolin-2-yl]-4-(4-hydroxypiperidin-1-yl)piperidin-3-ol
(cyclopropylmethyl)({5-methyl-2-[4-(methylsulfanyl)phenyl]-1,3-oxazol-4-yl}methyl)propylamine
N-[2-(pyridin-3-yl)-5,6,7,8-tetrahydroquinazolin-5-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-4-carboxamide
N-[5-(methoxymethyl)-1,3,4-thiadiazol-2-yl]-2-[4-(oxolane-2-carbonyl)piperazin-1-yl]acetamide
2-(2,4-difluorophenyl)-5-(oxolan-3-ylmethyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
6-methyl-4-oxo-N-[2-(pyridin-3-yloxy)propyl]-4H-pyran-2-carboxamide
7-chloro-2-{[methyl({[4-(trifluoromethyl)phenyl]methyl})amino]methyl}quinazolin-4-amine
[(1-methyl-1H-pyrazol-4-yl)methyl]({[5-methyl-2-(3-phenoxyphenyl)-1,3-oxazol-4-yl]methyl})(propan-2-yl)amine
1-[(3R,4R)-3-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]-2-(phenylsulfanyl)ethan-1-one
(4aS,7aR)-1-(furan-2-carbonyl)-4-[(2-methylpyrimidin-5-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-chloro-N-(furan-3-ylmethyl)-N,1-dimethyl-1H-indole-2-carboxamide
4-[1-(thiophen-2-yl)ethyl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-2-(propan-2-yl)-1,3-benzoxazole-5-carboxamide
4-[(3,4-difluorophenyl)methyl]-7-(2,3-dimethoxyphenyl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
(3aR,6aR)-2-cyclopentyl-5-(5-propylpyrimidin-4-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
7-[(8-chloroquinolin-2-yl)methyl]-2,7-diazaspiro[4.4]nonane-1,3-dione
5-ethyl-4-(4-{[2-(furan-2-yl)pyrimidin-5-yl]methyl}piperazin-1-yl)-2-methylpyrimidine
3-cyclopentyl-1-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]propan-1-one
1-{2-[4-(pyridin-4-yloxy)piperidin-1-yl]pyrimidin-4-yl}piperidin-3-ol
2-(3-methyl-5-{1-[2-(propan-2-yl)-1H-imidazol-1-yl]ethyl}-1H-1,2,4-triazol-1-yl)ethan-1-ol
N-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-N-methyl-3-(propan-2-yl)-1,2-oxazole-5-carboxamide
(3-{[1-(4-fluoro-2-methylbenzoyl)pyrrolidin-3-yl]methyl}phenyl)methanol