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3-[(3-methoxyphenyl)methyl]-8-[(1-methyl-1H-indol-3-yl)methyl]-1-(3-methylbutyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(2S,4R)-4-amino-N-ethyl-1-(2-{4-oxo-3H,4H-thieno[3,2-d]pyrimidin-3-yl}acetyl)pyrrolidine-2-carboxamide
2-(1H-indol-3-yl)-N-[1-(pyrazin-2-yl)piperidin-3-yl]acetamide
6-methyl-2-[5-(1H-pyrazol-5-yl)furan-2-yl]-1H-1,3-benzodiazole
1-(3-{5-[(4-hydroxypiperidin-1-yl)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2-methoxyethan-1-one
N2,N2-dimethyl-N5-[(4-phenyl-1,3-thiazol-2-yl)methyl]-5,6,7,8-tetrahydroquinazoline-2,5-diamine
4-[(3-propoxypiperidin-1-yl)methyl]benzene-1,2-diol
N-[(5-carbamoyl-1,2,4-oxadiazol-3-yl)methyl]-2-[(3S)-3-hydroxypyrrolidin-1-yl]-1-methyl-1H-1,3-benzodiazole-5-carboxamide
1-[4-(3,5-dimethyl-1H-pyrazol-1-yl)benzoyl]-3-[(4-fluorophenyl)methyl]piperidine
2-[1-(2-methylpropanoyl)piperidin-4-yl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-[1-(4-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}phenyl)ethyl]acetamide
{3-[(2,4-difluorophenyl)methyl]-1-(thiophene-3-carbonyl)piperidin-3-yl}methanol
5-{[(3-hydroxypropyl)[(5-methylthiophen-2-yl)methyl]amino]methyl}-2-methoxybenzoic acid
[1-(dimethyl-1,3-thiazol-4-yl)ethyl](methyl)({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)amine
1-{5-cyclopropyl-1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-1H-pyrazole-4-carbonyl}-N,N-diethylpyrrolidin-3-amine
(1R,5R)-3-[(1-ethyl-1H-pyrazol-4-yl)sulfonyl]-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonane
[(3R,4R)-4-(azepan-1-ylmethyl)-1-(pyridine-4-carbonyl)pyrrolidin-3-yl]methanol
3-(2-ethyl-1H-imidazol-1-yl)-1-(6-hydroxy-1,4-oxazepan-4-yl)propan-1-one
1-(2-methoxyacetyl)-N-methyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]piperidine-4-carboxamide
(2S,4S)-N,N-diethyl-4-[(1-ethylpiperidin-4-yl)amino]-1-(naphthalen-1-ylmethyl)pyrrolidine-2-carboxamide
1-[(2-fluorophenyl)methyl]-N-[2-(methylsulfanyl)ethyl]-6-oxopiperidine-3-carboxamide
1-{2-ethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}-4-[(2-methylphenyl)methyl]piperazine
1-cyclopropyl-N-({2-methylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)-6-oxopiperidine-3-carboxamide
N-(4-methylphenyl)-3-oxo-3-{2-[5-(propan-2-yl)-1,2-oxazol-3-yl]pyrrolidin-1-yl}propanamide
2-[4-(5-methoxypyridin-3-yl)-1H-pyrazol-1-yl]-N-(1-phenyl-1H-pyrazol-5-yl)acetamide
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)pyrrolidine-3-carboxylic acid
6-cyclopentyl-N,1-dimethyl-N-[2-(pyrrolidin-1-yl)ethyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-[(2-fluorophenyl)methyl]-4-{[3-(3-methoxyphenyl)-1,2-oxazol-5-yl]methyl}piperidin-4-ol
2-[(2-{[2-(3,5-dimethoxyphenyl)ethyl]carbamoyl}phenyl)amino]acetic acid
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-2-(1H-1,2,3,4-tetrazol-5-yl)benzamide
1-(azepan-1-yl)-3-[(3S,4R)-4-[4-(2-methoxyphenyl)piperazin-1-yl]-1-(pyridin-2-ylmethyl)piperidin-3-yl]propan-1-one
N-{1-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-6-methylpyrazolo[1,5-a]pyrimidine-3-carboxamide
1-{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-methylpiperidin-3-ol
N3-[(1R,2S,4R)-bicyclo[2.2.1]hept-5-en-2-ylmethyl]-N5-methyl-1-(3-methylbutyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
3-({[(5-chloro-2,3-dimethoxyphenyl)methyl]amino}methyl)-N,N-dimethylpyridin-2-amine
1-{3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
1-(3-chlorophenyl)-5-methyl-4-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperazin-2-one
N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-5-phenyl-1,2-oxazole-4-carboxamide
3-{[methyl({[3-(methylsulfanyl)phenyl]methyl})amino]methyl}pyrrolidin-3-ol
methyl 2-(azocane-1-sulfonyl)-6-(but-3-enoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
2-ethoxy-5-(2-{[2-(pyridin-3-yl)ethyl]amino}pyrimidin-4-yl)benzoic acid
2-[(1R,3R,5S)-3-(4-methoxyphenyl)-8-azabicyclo[3.2.1]octane-8-carbonyl]benzonitrile
N-[3-(4-methyl-1,3-thiazol-5-yl)propyl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
2-[4-(4-cyclopentyl-1H-1,2,3-triazol-1-yl)piperidine-1-carbonyl]pyrazine
2-(3-{[(3-hydroxy-3-phenylpropyl)(methyl)amino]methyl}-2-methyl-1H-indol-1-yl)acetamide
2-(3-hydroxypropyl)-9-{[1,2,4]triazolo[1,5-a]pyrimidin-2-ylmethyl}-2,9-diazaspiro[5.5]undecan-3-one
3-[2-(4-aminopiperidin-1-yl)-2-oxoethyl]-N-(2-methoxyethyl)-4-methyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
2-({cyclopropyl[(4-hydroxyphenyl)methyl]amino}methyl)-8-fluoroquinolin-4-ol
4-[1-(thiophen-2-ylmethyl)piperidin-4-yl]pyridine
2-{4-[(4-phenyl-1,3-thiazol-2-yl)methyl]-1-(thiophen-2-ylmethyl)piperazin-2-yl}ethan-1-ol