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(1R,3R)-N1-[6-ethyl-2-(morpholin-4-yl)pyrimidin-4-yl]cyclopentane-1,3-diamine
1-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-1-yl}-2-(3-methyl-1,2-oxazol-5-yl)ethan-1-one
4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-2,1,3-benzoxadiazole
3-(1-butyl-1H-imidazol-2-yl)-1-(1,2-oxazole-3-carbonyl)piperidine
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-5-(2,6-difluorophenoxymethyl)-1,2-oxazole-3-carboxamide
3-(1,2,3,4-tetrahydroisoquinolin-5-yl)-1,2-dihydropyridin-2-one
3-[1-(3-ethynylbenzoyl)piperidin-3-yl]-N-[(2-fluorophenyl)methyl]propanamide
3-(3-fluorophenyl)-4-[(2R)-2-(methoxymethyl)pyrrolidine-1-carbonyl]-1H-pyrazole
1-[3-(2-benzylmorpholin-4-yl)-3-oxopropyl]azepan-2-one
1-{[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(4-methyl-1,2,5-oxadiazol-3-yl)piperazine
1-(2-{1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]piperidin-4-yl}ethyl)pyrrolidin-2-one
benzyl({[3-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]methyl})methylamine
4-({4-[(3,4-difluorophenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}methyl)-2,6-dimethylphenol
5-(4-chloro-1,3-dimethyl-1H-pyrazol-5-yl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
{4-[(4-methoxyphenyl)methyl]-1-[(2E)-2-methylbut-2-en-1-yl]piperidin-4-yl}methanol
2-methyl-4-phenyl-9-(3-phenyl-1,2,4-oxadiazol-5-yl)-2,9-diazaspiro[5.5]undecan-3-one
2-(dimethylamino)-2-(4-fluorophenyl)-N-[(4-fluorophenyl)methyl]-N-(3-hydroxypropyl)acetamide
8-methyl-4-oxo-N-[1-(pyridin-4-yl)propyl]-1,4-dihydroquinoline-3-carboxamide
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-5-methyl-1,2-oxazole-3-carboxamide
3-(2-methoxy-5-phenylphenyl)-1-(morpholin-2-ylmethyl)urea
4-[1-(pyridin-4-ylmethyl)piperidin-3-yl]morpholine
1-(4-{[6-(hydroxymethyl)-1,4-oxazepan-4-yl]methyl}thiophen-2-yl)ethan-1-one
3-[(1S,9aR)-octahydro-1H-quinolizin-1-yl]-N-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]propanamide
N-benzyl-2-chloro-5-acetamido-N-ethylbenzamide
4-(2-methanesulfonylethyl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
[3-(3-methylbut-2-en-1-yl)-1-(pyrrolidine-1-sulfonyl)piperidin-3-yl]methanol
1-(2-phenylethyl)-4-[(quinoxalin-2-yl)amino]pyrrolidin-2-one
2-(1H-1,3-benzodiazol-1-yl)-N-ethyl-N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]propanamide
4-{[(4-acetylmorpholin-2-yl)methyl]amino}-N-(pyridin-3-ylmethyl)pyridine-2-carboxamide
N-(1-benzylpyrrolidin-3-yl)-3-[1-(2-phenoxyacetyl)piperidin-4-yl]propanamide
(1s,4s)-4-(4-methyl-3-phenylpiperazine-1-carbonyl)cyclohexan-1-ol
1-ethyl-N,4,6-trimethyl-2-oxo-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-1,2-dihydropyridine-3-carboxamide
(3S)-1-{[2-(3-methylphenyl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}pyrrolidin-3-ol
4-{1,3-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-1-(3,5-dimethylphenyl)piperazin-2-one
2-benzyl-4-(thiophene-2-carbonyl)morpholine
4,5-dichloro-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}thiophene-2-sulfonamide
N-[(1R,3R)-3-aminocyclopentyl]-2-methyl-1,3-benzothiazole-5-carboxamide
1-(thiophen-2-ylmethyl)-4-[2-(4H-1,2,4-triazol-4-yl)pyridine-4-carbonyl]piperazine
3-(piperidine-1-carbonyl)-1-(prop-2-en-1-yl)-N-(2,2,2-trifluoroethyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-(3-{6-[(2-methoxyethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}thiophen-2-yl)ethan-1-one
ethyl 1-benzyl-4-(2-phenoxyethyl)piperidine-4-carboxylate
(3S,4R)-1-[2-(3-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)acetyl]-4-(pyridin-4-yl)pyrrolidine-3-carboxylic acid
(5S,9aS,9bS)-5-(2H-1,3-benzodioxol-4-yl)-2-phenyl-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
ethyl 2-[methyl(5-{[4-(1H-1,2,4-triazole-3-carbonyl)piperazin-1-yl]methyl}pyrimidin-2-yl)amino]acetate
4-[3-(furan-2-yl)-1H-pyrazol-1-yl]-1-[2-(1H-pyrazol-1-yl)acetyl]piperidine-4-carboxylic acid
N-(3,4-dimethyl-1H-pyrazol-5-yl)-2-phenylacetamide
2-{4-[3-(oxolan-3-yl)-1H-1,2,4-triazol-5-yl]piperidine-1-carbonyl}pyridine
8-[2-(3-methyl-1H-pyrazol-1-yl)ethyl]-2-(propan-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
(3aS,6aS)-2-[2-(benzenesulfonyl)ethyl]-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1,3,7-trimethyl-N-[2-(4-methylmorpholin-2-yl)ethyl]-1H-indole-2-carboxamide