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(1R,5R)-6-[(2-ethyl-1,3-thiazol-4-yl)methyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
N-methyl-2-[2-methyl-4-oxo-1-(2-phenylethyl)-4,5,6,7-tetrahydro-1H-indol-3-yl]-N-(propan-2-yl)acetamide
N-[(2-ethoxypyridin-3-yl)methyl]-5-(oxolan-2-yl)thiophene-2-carboxamide
3,5-dimethyl-1-[3-(4H-1,2,4-triazol-4-yl)propyl]-1H-1,2,4-triazole
2-(4-chlorophenyl)-2-hydroxy-1-[4-(pyridin-3-ylmethoxy)piperidin-1-yl]ethan-1-one
N-[2-(dimethylamino)ethyl]-N-methyl-1-(5-propyl-1,2-oxazole-4-carbonyl)piperidin-3-amine
ethyl 4-{3-phenyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}piperidine-1-carboxylate
methyl 2-[(2,3-dimethylphenyl)sulfamoyl]-6-(2-methylpropanoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
2-[4-(4-methyl-1,4-diazepan-1-yl)-6-oxo-1,6-dihydropyridazin-1-yl]-N-[1-(pyridin-2-yl)propyl]acetamide
6-(4-methoxypiperidin-1-yl)-N-[(3-propyl-1,2-oxazol-5-yl)methyl]pyridine-3-carboxamide
3-butanamido-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]benzamide
1-(3-benzylphenyl)-3-[(3-hydroxypiperidin-3-yl)methyl]urea
2-methyl-8-{2-[4-(oxolan-3-yl)-1H-1,2,3-triazol-1-yl]ethoxy}quinoline
3-(1,1-dioxo-1λ6-thiolan-3-yl)-3-(2-hydroxyethyl)-1-(3-methoxy-4-methylphenyl)urea
3-({1-[2-(4-methyl-1,2,5-oxadiazol-3-yl)acetyl]pyrrolidin-3-yl}methyl)benzamide
methyl 1-methyl-2-[2-(trifluoromethyl)morpholin-4-yl]-1H-1,3-benzodiazole-5-carboxylate
3-(1H-1,3-benzodiazol-1-yl)-1-[1-(2-hydroxyethyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl]propan-1-one
(1H-1,3-benzodiazol-2-ylmethyl)[(5-methylthiophen-2-yl)methyl](pyridin-4-ylmethyl)amine
3-[2-(2-ethyl-1H-imidazol-1-yl)ethyl]-1-[2-methoxy-5-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]urea
2-{4-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]-1-[(6-methylpyridin-2-yl)methyl]piperazin-2-yl}ethan-1-ol
4-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
3-acetyl-N-(2-tert-butyl-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-5-yl)-1H-pyrazole-5-carboxamide
N-(2-{4H,5H,6H-cyclopenta[d][1,3]thiazol-2-yl}ethyl)-2-(pyridin-3-yl)pyrimidine-5-carboxamide
6-methyl-3-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
5-methyl-1-(4-methylphenyl)-4-[(6-methylpyridin-2-yl)methyl]piperazin-2-one
1-cyclopropanecarbonyl-N-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}piperidine-4-carboxamide
N,N-diethyl-1-({1-[2-(2-fluorophenyl)acetyl]piperidin-3-yl}methyl)-1H-1,2,3-triazole-4-carboxamide
N-cyclopentyl-4-[2-(4-fluorophenyl)morpholin-4-yl]-4-oxobutanamide
methyl 3-[1-ethyl-3-(4-phenylpiperazine-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]propanoate
2-amino-3-ethyl-N-{2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}-3H-imidazo[4,5-b]pyridine-6-carboxamide
ethyl 4-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-amido]piperidine-1-carboxylate
1-cyclopentyl-4-{2,3-dimethyl-4-oxo-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}pyrrolidin-2-one
N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)cyclopropanesulfonamide
[(1-cyclopentylpiperidin-4-yl)methyl]({[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl})(pyridin-3-ylmethyl)amine
N-[(5-{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)methyl]acetamide
2-(2-aminopyrimidin-5-yl)-N,8-dimethyl-N-(pyridin-2-ylmethyl)quinoline-4-carboxamide
N-[2-(dimethylamino)-2-(furan-2-yl)ethyl]-2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-amine
3-[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]propanamide
N-(cyclopropylmethyl)-6-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperidine-3-carboxamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-cyclopropyl-4-(1H-pyrazol-4-yl)butanamide
N-[2-(ethanesulfonyl)ethyl]-1-(4-methoxyphenyl)-2,2-dimethylcyclopropane-1-carboxamide
N-[1-(1-cyclopropylethyl)-4-methyl-1H-pyrazol-5-yl]-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)acetamide
N-[2-(dimethylamino)ethyl]-3-{1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}propanamide
N-[2-(3-benzyl-1,2,4-oxadiazol-5-yl)ethyl]-3-(4-methyl-1,3-thiazol-5-yl)propanamide
N-[2-(4-methylmorpholin-2-yl)ethyl]-3-phenyl-1,2-oxazole-5-carboxamide
9-(1-cyclopropyl-1H-pyrrole-2-carbonyl)-2-(3-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
(3aS,6aS)-2-(dimethylcarbamoyl)-5-[4-(ethylamino)pyrimidin-2-yl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-[(3R,4S)-1-[3-(1H-1,3-benzodiazol-1-yl)propanoyl]-4-(dimethylamino)piperidin-3-yl]propanoic acid
1-[3-(cyclopentyloxy)phenyl]-3-[1-(pyrazin-2-yl)propan-2-yl]urea
7-(oxan-4-yl)-2-(1,3-thiazol-2-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one