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4-{[1-(2-amino-6-methylpyrimidin-4-yl)piperidin-4-yl]amino}-1-propylpyrrolidin-2-one
1-(5-methyl-1,2-oxazole-3-carbonyl)-4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidine
1-ethyl-5-(3-fluoro-4-methylphenyl)-1H,4H-pyrazolo[3,4-d]imidazole
N-[1-(1-cyclopropylethyl)-3-methyl-1H-pyrazol-5-yl]-4-(2-methoxyacetyl)-1,4-diazepane-1-carboxamide
N,N-dimethyl-2-{[2-(phenylsulfanyl)acetamido]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
(1R,3S)-3-amino-N-(3-hydroxypropyl)-N-(naphthalen-1-ylmethyl)cyclohexane-1-carboxamide
3-(4-hydroxyphenyl)-N-{2-[(2-methylquinolin-8-yl)oxy]ethyl}-1H-pyrazole-5-carboxamide
1-{6-chloroimidazo[1,2-a]pyridine-2-carbonyl}-4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine
N-{[2-(dimethylamino)-1,3-thiazol-4-yl]methyl}-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
(1S,5R)-3-(5-methyl-1H-indazole-3-carbonyl)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-(2-{[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
1-(4-methoxybenzoyl)-4-[2-(phenylsulfanyl)ethyl]piperazine
(2S,4R)-N-(2-methoxyethyl)-4-{[(2-methoxynaphthalen-1-yl)methyl]amino}-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxamide
diethyl({[3-(4-phenylpiperidine-1-carbonyl)pyrazolo[1,5-a]pyrimidin-6-yl]methyl})amine
5-propyl-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)-1,2,4-oxadiazol-3-amine
N-[(3R,5S)-5-(ethylcarbamoyl)-1-[(5-methylfuran-2-yl)methyl]pyrrolidin-3-yl]-1H-1,2,4-triazole-5-carboxamide
8-(9H-fluoren-2-ylmethyl)-1-methyl-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-{[(4aS,7aR)-4-(2-methylpropyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]methyl}benzoic acid
4-(5-methylpyridin-2-yl)-1-(2,3,4,5-tetrahydro-1-benzoxepine-4-carbonyl)piperidin-4-ol
4-(piperidin-3-yl)-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}benzamide
6-(2-chlorophenyl)-2-{3-[(diethylamino)methyl]phenyl}-3,4-dihydropyrimidin-4-one
2-(3-{1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl}piperidin-1-yl)pyridine
(1S,3R)-3-[2-(4-chlorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]cyclohexan-1-amine
N-(5-ethyl-1,3,4-thiadiazol-2-yl)-2-[4-ethyl-5-oxo-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-1-yl]propanamide
1-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
2-cyclopropyl-6-(1-{[5-(oxan-2-yl)furan-2-yl]methyl}piperidin-4-yl)-3,4-dihydropyrimidin-4-one
N,N,6,8-tetramethyl-2-[2-(propan-2-yl)pyrimidin-5-yl]quinoline-4-carboxamide
N-(3-benzyl-1H-1,2,4-triazol-5-yl)-3-(2-methoxyphenoxy)azetidine-1-carboxamide
1-ethyl-2-{[(1S,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}-1H-1,3-benzodiazole
{[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}(methyl)[1-(1,3-thiazol-2-yl)ethyl]amine
2-tert-butyl-4-hydroxy-N-{3-[(pyridin-3-yl)amino]propyl}pyrimidine-5-carboxamide
2-methyl-N-[(2-methylphenyl)methyl]-N-(prop-2-en-1-yl)-3-(1H-pyrazol-1-yl)propanamide
3-methyl-N-({4-[(3-phenylpropyl)amino]quinazolin-2-yl}methyl)-5,6-dihydro-1,4-dioxine-2-carboxamide
2-[1-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)pyrrolidin-2-yl]pyridine
(2S,4S)-N-methyl-4-(4-{4-[(4-methylpiperidin-1-yl)methyl]phenyl}-1H-1,2,3-triazol-1-yl)pyrrolidine-2-carboxamide
N-{2H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-N-methyl-3-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]propanamide
1-{2-[1-(2-hydroxyethyl)-3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]ethyl}-2,3-dihydro-1H-1,3-benzodiazol-2-one
[(1-{[1-(2,3-dihydro-1-benzofuran-2-carbonyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)methyl](methyl)amine
(1-benzofuran-2-ylmethyl)(methyl)[(5-methyl-1H-pyrazol-3-yl)methyl]amine
N-[(3R,4S)-1-methanesulfonyl-4-(propan-2-yl)pyrrolidin-3-yl]-1,5-dimethyl-1H-pyrazole-4-carboxamide
8-[(2S)-2-aminopropanoyl]-3-hexyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-(2-chloroprop-2-en-1-yl)-3-({[1-(furan-2-yl)ethyl]amino}methyl)-6,7-dimethoxy-1,2-dihydroquinolin-2-one
(2R,3R,6R)-5-methyl-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-[(2-fluorophenyl)methyl]-4-(2-methyl-1H-imidazol-1-yl)piperidine-4-carboxylic acid
(1R,2S)-2-(methoxymethyl)-N-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}cyclopentan-1-amine
(2S)-N-[(5-chloro-3-methyl-2-phenyl-1H-indol-7-yl)methyl]-1-methylpyrrolidine-2-carboxamide
4-[4-(aminomethyl)-1H-1,2,3-triazol-1-yl]-N-(cyclohexylmethyl)piperidine-1-carboxamide
N-[(1-methyl-1H-imidazol-2-yl)methyl]quinoline-6-carboxamide
3-(2-{3-[(3,4-dimethylphenyl)amino]piperidin-1-yl}-2-oxoethyl)-1,3-thiazolidine-2,4-dione
1-ethyl-3-[(3-methoxyphenyl)methyl]-8-(thiophen-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione