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8-[2-(9-methyl-9H-carbazol-3-yl)acetyl]-2,8-diazaspiro[4.5]decan-3-one
N-methyl-N-[1-(2-phenylethyl)piperidin-3-yl]-3-(thiophen-3-yl)propanamide
2-(2,1,3-benzothiadiazol-5-ylmethyl)-7-(2-phenylethyl)-2,7-diazaspiro[4.5]decane
3-(4-chloro-3-fluorophenyl)-1-[(3R)-piperidin-3-yl]urea
(3aS,6aS)-2-(dimethylcarbamoyl)-5-[2-(1H-imidazol-2-yl)ethyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-3-(1H-pyrazol-1-yl)propanamide
4-methyl-5-(2-{3-propyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}ethyl)-1,3-thiazole
4-(1-{5-[1-(piperidin-1-yl)ethyl]furan-2-carbonyl}piperidin-4-yl)thiomorpholine
2-fluoro-N-{3-[(3R,4R)-4-hydroxy-4-(2-methoxyethyl)-3-methylpiperidin-1-yl]-3-oxopropyl}benzamide
1-[3-(benzyloxy)piperidin-1-yl]-2-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}ethan-1-one
2-ethyl-6-methyl-4-oxo-N-(pyridin-3-ylmethyl)-1-(thiophen-2-ylmethyl)-1,4-dihydropyridine-3-carboxamide
N-{[6,7-dimethoxy-2-(3-methoxyphenyl)quinolin-3-yl]methyl}-4-fluoro-N-(oxolan-2-ylmethyl)benzamide
7-methoxy-N-methyl-N-(thian-4-yl)-3,4-dihydro-2H-1-benzopyran-3-carboxamide
methyl 2-{[2-(4-fluorophenoxymethyl)-1,3-oxazol-4-yl]formamido}acetate
1-(2-methoxyethyl)-3-(1-oxo-2,3-dihydro-1H-inden-5-yl)-1-(thiophen-3-ylmethyl)urea
N-(3-ethyl-4-methyl-1-phenyl-1H-pyrazol-5-yl)-2,2-dimethyl-4-oxo-3,4-dihydro-2H-pyran-6-carboxamide
4-(1H-imidazol-1-ylmethyl)-1-({2-[(oxolan-2-ylmethyl)amino]pyrimidin-5-yl}methyl)piperidin-4-ol
N,3-dimethyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-3H-[1,2,3]triazolo[4,5-b]pyridine-6-carboxamide
N-[(4-chloro-1-methyl-1H-indazol-3-yl)methyl]-1-(pyrimidin-2-yl)piperidin-4-amine
6-{7-methyl-6-oxo-2,7-diazaspiro[4.5]decane-2-carbonyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-[(2,6-dichloro-3,4-dimethoxyphenyl)methyl]-4-(hydroxymethyl)azepan-4-ol
3-({1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}(methyl)amino)propane-1,2-diol
1-{[methyl({[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl})carbamoyl]methyl}piperidine-4-carboxamide
1-[(3R,4S)-3-(3-hydroxypropyl)-4-(4-methylpiperazin-1-yl)piperidin-1-yl]-2-phenoxyethan-1-one
7-{imidazo[1,2-a]pyridine-3-carbonyl}-2-(pyridin-3-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-{1-[(2-ethoxyphenyl)methyl]-4-[(5-methylthiophen-2-yl)methyl]piperazin-2-yl}ethan-1-ol
5-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]-N-(pyridin-3-ylmethyl)pyridin-2-amine
(2R,3R)-3-amino-1'-[(2-methoxy-4-methylphenyl)methyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
8-methoxy-N-[(2-methyl-1H-1,3-benzodiazol-6-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
7-(3,6-dimethylpyrazin-2-yl)-4-(piperidine-4-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
{[1-(cyclohexylmethyl)-2-cyclopropylmethanesulfonyl-1H-imidazol-5-yl]methyl}(ethyl)(pyridin-4-ylmethyl)amine
N-methyl-4-{[({2-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)amino]methyl}benzamide
5-(4-cyclobutyl-6-methylpyrimidin-2-yl)-4H,5H,6H,7H-[1,3]thiazolo[5,4-c]pyridin-2-amine
(5S)-5-{[({3-[1-(4-methylphenyl)cyclopentyl]-1,2,4-oxadiazol-5-yl}methyl)(pyridin-4-ylmethyl)amino]methyl}pyrrolidin-2-one
N-methyl-5-(phenoxymethyl)-N-[2-(1H-pyrazol-4-yl)ethyl]-1H-pyrazole-3-carboxamide
N-(5-aminopentyl)-2-methyl-1-benzofuran-5-carboxamide
2-(4-{[4-(2-aminoethyl)phenyl]methyl}-6-hydroxy-1,4-diazepan-1-yl)acetamide
2-(2,4-dioxo-1,3-diazinan-1-yl)-N-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-N-methylbenzamide
2-{4-[(1S,4S)-2-azabicyclo[2.2.1]heptan-2-ylmethyl]phenyl}-6-(phenoxymethyl)-3,4-dihydropyrimidin-4-one
3-[2-(morpholin-4-yl)-2-oxoethyl]-4-(3-phenylpropyl)piperazin-2-one
1-[4-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]-3-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]propan-1-one
3-{5-[1-(2,4-difluorophenoxy)ethyl]-1,2,4-oxadiazol-3-yl}pyridazine
2-{2-[1-({4-oxo-4H-pyrido[1,2-a]pyrimidin-2-yl}methyl)piperidin-3-yl]-1H-imidazol-1-yl}acetamide
2-({[1-(3,4-dihydro-2H-1-benzopyran-3-carbonyl)piperidin-4-yl]oxy}methyl)pyridine
4-(4-{[3-(hydroxymethyl)-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}phenyl)-2-methylbutan-2-ol
1-(2-{4-[(5-chloro-2-hydroxyphenyl)methyl]piperazin-1-yl}ethyl)-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
5-(2-{[1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}ethyl)-1,3,4-thiadiazol-2-amine
N-[1-methyl-4-(morpholin-4-yl)-1H-indazol-3-yl]-2-(1H-1,2,4-triazol-1-yl)acetamide
2-{1-[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]-1H-imidazol-2-yl}pyridine
N-cyclopropyl-5-methyl-4-[(prop-2-en-1-yl)amino]thieno[2,3-d]pyrimidine-6-carboxamide