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2-{8-methylimidazo[1,2-a]pyridin-3-yl}-1-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
1-{1-[6-(propan-2-yl)-2-(trifluoromethyl)pyrimidin-4-yl]piperidin-3-yl}pyrrolidin-2-one
1-{[4-(2H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
4-{4-[(4-chlorophenyl)methyl]piperazin-1-yl}-5-ethyl-6-methylpyrimidin-2-amine
4-(7-methoxy-2H-1,3-benzodioxol-5-yl)-1-methyl-3-(pyridin-3-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
8-(1-methyl-2-oxoimidazolidine-4-carbonyl)-2-(3-phenylpropyl)-2,8-diazaspiro[4.5]decan-3-one
N-cyclopropyl-N-[(3-ethoxyphenyl)methyl]-3-(2-methoxyacetamido)benzamide
N-(2-methoxyethyl)-4-[(2-methoxyethyl)amino]-N,5-dimethylthieno[2,3-d]pyrimidine-6-carboxamide
4-hydroxy-2-{[2-(5-methyl-1,2-oxazol-3-yl)piperidin-1-yl]methyl}quinoline-6-carboxamide
(1-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}piperidin-4-yl)methanol
N3-(1-benzothiophen-2-ylmethyl)-1-cyclopentyl-N3,N5-dimethyl-N5-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
3-(2-amino-1,3-thiazol-4-yl)-N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]propanamide
methyl 1-[1-(7-methoxy-4-methylquinazolin-2-yl)piperidine-4-carbonyl]piperidine-2-carboxylate
1-{3-[3-(hydroxymethyl)-3-(prop-2-en-1-yl)piperidin-1-yl]-3-oxopropyl}pyrrolidin-2-one
N-methyl-2-[4-(methylsulfanyl)phenyl]-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
2-(2H-1,3-benzodioxol-5-yl)-1-{2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidin-1-yl}ethan-1-one
3-[(2-{[4-(pyridin-3-yl)piperazin-1-yl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl)methyl]phenol
[(5-fluoro-1H-indol-2-yl)methyl](methyl){[3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}amine
N-[(3S,5S)-1-ethyl-5-(ethylcarbamoyl)pyrrolidin-3-yl]-3-(4-hydroxyphenyl)-1H-pyrazole-5-carboxamide
(1S,5R)-3-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
(3R,4R)-4-(2-methoxyethyl)-3-methyl-1-(3-phenylpropyl)piperidin-4-ol
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-3-[4-(3-methylphenyl)piperazin-1-yl]propanamide
N-[(3S,7S,8aS)-1,4-dioxo-3-(propan-2-yl)-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-bromobenzamide
(3aR,6aR)-2-cyclopentanecarbonyl-5-(2-methylbenzoyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[1-(methoxymethyl)cyclopentyl]-2-(pyrrolidin-3-yl)benzamide
1-(1-methyl-1H-1,2,3-benzotriazole-5-carbonyl)-4-(5-methylpyridin-2-yl)piperidin-4-ol
3-[(3-cyclohexyl-1,2,4-oxadiazol-5-yl)methyl]-1-(2-fluoro-4-methoxyphenyl)urea
ethyl({[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}){[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}amine
(2S,4S)-1-[(dimethylcarbamoyl)methyl]-N-ethyl-4-[2-(4-methylphenyl)acetamido]pyrrolidine-2-carboxamide
N-(oxan-4-yl)-4-(piperidin-3-yl)benzamide
(1R,9aR)-1-[4-(1-methyl-1,2,3,6-tetrahydropyridin-4-yl)phenoxymethyl]-octahydro-1H-quinolizine
2-[2-(4-hydroxyphenyl)pyrimidin-4-yl]pyridine-4-carboxylic acid
N-cyclobutyl-5-(3-fluorophenyl)-1,2,4-triazin-3-amine
N,1-dimethyl-4-phenyl-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]piperidine-4-carboxamide
1-(2-{2-[(9aS)-octahydro-1H-pyrrolo[1,2-a][1,4]diazepin-2-ylmethyl]phenoxy}ethyl)piperidine
1-methanesulfonyl-4-[1-(methoxymethyl)cyclobutanecarbonyl]-1,4-diazepane
8-[3-(dimethylamino)propanoyl]-3-(2-phenylpropyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-1-[3-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)phenyl]urea
methyl 3-[(3S,4R)-4-[4-(2-fluorophenyl)piperazin-1-yl]-1-{[2-(prop-2-en-1-yloxy)phenyl]methyl}piperidin-3-yl]propanoate
2-{1-[(2,3-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(1H-pyrazol-1-yl)ethyl]acetamide
(3R,7S,8aS)-7-{[(3-chlorophenyl)methyl]amino}-3-[(1S)-1-hydroxyethyl]-octahydropyrrolo[1,2-a]piperazine-1,4-dione
(1S,5R)-6-benzyl-3-{2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-2-oxoethyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
2-{1-[(3,4-difluorophenyl)methyl]piperidin-3-yl}-6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline
1-{6-[6-(cyclopentylamino)-1H-pyrrolo[2,3-b]pyridin-4-yl]pyridin-2-yl}ethan-1-ol
5-chloro-6-{6-[(pyridin-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}pyridine-3-carboxylic acid
1-[3-({[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)phenoxy]-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
3,5-dichloro-N-(1,4-dioxan-2-ylmethyl)-N,4-dimethylbenzamide
(1S,5R)-3-benzyl-6-(3-phenyl-1H-pyrazole-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-[(dimethyl-1,3-thiazol-5-yl)methyl]-1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
1-[(2-fluoro-4-methoxyphenyl)methyl]-4-(pyridin-4-ylmethyl)-1,4-diazepane