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2-{[(3aS,6aS)-5-{2-ethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}-octahydropyrrolo[3,4-b]pyrrol-1-yl]methyl}-1-methyl-1H-imidazole
2-(dimethyl-1,3-thiazol-5-yl)-1-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}ethan-1-one
2-chloro-N-[1-(cyclohexylmethyl)piperidin-3-yl]-6-fluorobenzamide
2-[5-(3,5-dimethyl-1H-pyrazol-4-yl)-4-phenyl-1H-imidazol-1-yl]-N-(5-fluoro-2-methylphenyl)acetamide
4-(1-{3-[(1-methylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl}ethyl)-1,2-dihydrophthalazin-1-one
[1-methyl-4-({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)piperazin-2-yl]methanol
4-[3-(3-methoxyphenoxy)azetidine-1-carbonyl]-2,7,8-trimethylquinoline
(2S,4R)-N-{imidazo[1,2-a]pyridin-2-ylmethyl}-1-[(4-methoxy-3-methylphenyl)methyl]-4-[(4-methoxyphenyl)sulfanyl]pyrrolidine-2-carboxamide
(1r,4r)-4-({[(8-fluoro-4-hydroxyquinolin-2-yl)methyl]amino}methyl)cyclohexane-1-carboxamide
2-(dimethylamino)-N-ethyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-2-(4-methylphenyl)acetamide
5-fluoro-N2-{[2-(2-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}-N4-methylpyrimidine-2,4-diamine
[(dimethyl-1,2-oxazol-4-yl)methyl][1-(2-methoxyphenyl)propan-2-yl]amine
N-methyl-5-(1-{7-methylpyrazolo[1,5-a]pyrimidine-6-carbonyl}pyrrolidin-2-yl)thiophene-2-carboxamide
3-[3-(4-fluorophenyl)pyrrolidine-1-carbonyl]-1,2-dimethyl-1H-indol-5-ol
N-{[2-(morpholin-4-yl)pyridin-3-yl]methyl}quinoxaline-5-carboxamide
6-[4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepane-1-carbonyl]-1,3-benzothiazole
4-(2-fluoroethyl)-8-thia-4,6-diazatricyclo[7.5.0.02,7]tetradeca-1(9),2(7),5-trien-3-one
N-(2-methoxyethyl)-1-[1-(5-propyl-1,2,4-oxadiazol-3-yl)piperidin-4-yl]piperidine-3-carboxamide
1-[(3S,4R)-3-ethyl-4-hydroxy-4-methylpiperidin-1-yl]-2-[5-(4-fluorophenyl)-2H-1,2,3,4-tetrazol-2-yl]ethan-1-one
N-[3-(1H-indol-1-yl)propyl]-6,6-dimethyl-5-oxothiomorpholine-3-carboxamide
(3R,4S)-4-cyclopropyl-1-[(3-methylpyridin-2-yl)methyl]pyrrolidin-3-amine
N-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-methyl-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2-[2-(1H-imidazol-4-yl)ethyl]-8-[2-(methylsulfanyl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
4-methoxy-N-{2-[2-(4-methyl-1H-imidazol-5-yl)-1H-imidazol-1-yl]ethyl}benzene-1-sulfonamide
2-methyl-4-{1-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propyl]piperidin-3-yl}-6-(pyrrolidin-1-yl)pyrimidine
N-(2-fluoroethyl)-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-1-(7-methoxy-2,3,4,5-tetrahydro-1H-3-benzazepin-3-yl)ethan-1-one
N-(butan-2-yl)-N-[(2-fluorophenyl)methyl]-5-(methoxymethyl)furan-2-carboxamide
1-{2-[1-(2-fluorophenyl)-3-phenyl-1H-1,2,4-triazol-5-yl]ethyl}pyrrolidin-2-one
N-(1-benzylpyrrolidin-3-yl)-6-(morpholin-4-yl)pyrimidin-4-amine
3,3-dimethyl-1-(4-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperazin-1-yl)butan-1-one
1-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-3-(trifluoromethyl)-1,2-dihydropyridin-2-one
N-ethyl-5-{3-oxa-9-azaspiro[5.5]undecane-9-carbonyl}pyrimidin-2-amine
1-(4-fluorophenyl)-N-(oxolan-2-ylmethyl)-N-(thiophen-3-ylmethyl)cyclopropane-1-carboxamide
2-[1-(3-phenyl-1,2-oxazole-4-carbonyl)pyrrolidin-2-yl]-1,3-benzothiazole
2-(1-{[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methyl}-1H-pyrazol-4-yl)ethan-1-ol
4-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N5-(adamantan-1-yl)-N2,N2-dimethyl-5,6,7,8-tetrahydroquinazoline-2,5-diamine
N-ethyl-5-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyrimidin-2-amine
1-[4-hydroxy-4-(hydroxymethyl)azepan-1-yl]-3-(1H-indol-3-yl)propan-1-one
(4aR,8aR)-2-methanesulfonyl-7-(2-methoxypyridine-4-carbonyl)-decahydro-2,7-naphthyridin-4a-ol
1-cyclohexyl-N-(2-{imidazo[1,2-a]pyrimidin-2-yl}ethyl)-1H-1,2,3-triazole-4-carboxamide
5-[(3-hydroxypropyl)amino]-N-methyl-1-(2-phenylethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
8-[(2,4-dimethoxyphenyl)methyl]-2-(3-methoxypropyl)-2,8-diazaspiro[4.5]decan-3-one
1-{3-[4-(trifluoromethyl)phenyl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}but-2-yn-1-one
N,5,7-trimethyl-N-[(5-methylfuran-2-yl)methyl]pyrazolo[1,5-a]pyrimidine-2-carboxamide
N,N,5-trimethyl-2-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidin-4-amine
2-(2-aminoethyl)-N-(isoquinolin-5-ylmethyl)-N-methylquinazolin-4-amine
ethyl 1-[(3-acetylphenyl)methyl]-4-[(3-fluorophenyl)methyl]piperidine-4-carboxylate
2-methyl-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-1H-1,3-benzodiazole-5-carboxamide