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N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]cyclopropanecarboxamide
(2R)-2-amino-1-[3-(2-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-phenylethan-1-one
4-methyl-2-{1-[3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]piperidin-4-yl}-1H-1,3-benzodiazole
2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]-1-{1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}ethan-1-one
2-chloro-5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}pyridine
2-amino-6-{4-[4-(3-hydroxy-3-methylbutyl)benzoyl]piperazin-1-yl}-3,4-dihydropyrimidin-4-one
1-(2-chlorophenyl)-3-(1-{1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)urea
N-[(3S,4R)-1-{5-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carbonyl}-4-propylpyrrolidin-3-yl]acetamide
2-[(4-benzylpiperazin-1-yl)methyl]-4-phenylphenol
3-{2-[2-(3-methyl-1H-1,2,4-triazol-5-yl)pyrrolidin-1-yl]ethyl}-2,3-dihydro-1,3-benzoxazol-2-one
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)quinoxaline-5-carboxamide
N-[(3S,4R)-1-[2-(2,5-dioxoimidazolidin-1-yl)acetyl]-4-(4-methoxyphenyl)pyrrolidin-3-yl]acetamide
5-methyl-4-(1-methyl-1H-pyrazol-5-yl)-N-{[3-(1H-1,2,4-triazol-1-yl)phenyl]methyl}pyrimidin-2-amine
4-(1-benzofuran-2-yl)-2-{5-methyl-4-[4-(piperidin-1-yl)piperidine-1-carbonyl]-1H-pyrazol-1-yl}pyrimidine
3-{2-[3-(pyridine-2-carbonyl)piperidin-1-yl]ethyl}-2,3-dihydro-1,3-benzoxazol-2-one
2-(2,4-difluorophenoxy)-1-[3-(2,3-dimethoxyphenyl)pyrrolidin-1-yl]ethan-1-one
1-benzyl-8-[(3-hydroxyphenyl)methyl]-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-{[9-(2-methoxyethyl)-1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecan-4-yl]methyl}benzonitrile
9-{[2-(dimethylamino)pyrimidin-5-yl]methyl}-2-(2-methoxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
3-(2-fluorophenyl)-N-[5-(pentan-2-yl)-1,3,4-thiadiazol-2-yl]pyrrolidine-1-carboxamide
2-(2,1,3-benzothiadiazol-5-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-[(2-ethyl-3-methyl-1H-indol-5-yl)methyl]-2-(4H-1,2,4-triazol-4-yl)pyridine-4-carboxamide
4-[2-amino-6-(2H-1,3-benzodioxol-5-yl)-3-cyano-5-methylpyridin-4-yl]benzamide
1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-4-(furan-2-ylmethyl)piperazine
4-(3-propoxypiperidin-1-yl)-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaene
1-[5-(1H-imidazol-1-ylmethyl)furan-2-carbonyl]-4-[(3-methylpyridin-2-yl)methyl]piperazine
N-{[4-(4-methoxyphenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}-2-(thiophen-3-yl)acetamide
4-[4-(4-chlorophenyl)-4-hydroxypiperidine-1-carbonyl]-N,N-dimethylpiperidine-1-carboxamide
4-(1-{4-methyl-6H,7H,8H-cyclopenta[g]quinazolin-2-yl}piperidine-4-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-{[1-(1-ethyl-1H-1,3-benzodiazol-2-yl)-3-(oxolan-3-yl)-1H-1,2,4-triazol-5-yl]methyl}-1,3-oxazolidin-2-one
3-{[4-(4-methylphenyl)-5-(pyrimidin-5-yl)pyrimidin-2-yl]amino}-1λ6-thiolane-1,1-dione
1-[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl]-4-[(2-methoxyphenyl)methyl]piperazine
[(3R,4R)-1-({3-[(dimethylamino)methyl]phenyl}methyl)-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
(3R,4R)-4-(2-ethyl-4-methyl-1H-imidazol-5-yl)-1-methyl-N-[(5-methylpyrazin-2-yl)methyl]pyrrolidine-3-carboxamide
1-({[6-ethyl-2-(morpholin-4-yl)pyrimidin-4-yl]amino}methyl)cyclohexan-1-ol
3-{5-[(1-methyl-1H-imidazol-2-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
2-(3-methoxypropyl)-9-(2-phenylpropyl)-2,9-diazaspiro[5.5]undecan-3-one
1,9-dimethyl-4-(4,5,6,7-tetrahydro-1-benzothiophene-2-carbonyl)-1,4,9-triazaspiro[5.6]dodecan-10-one
3-(1-hydroxypropan-2-yl)-6-phenyl-3H,4H-thieno[2,3-d]pyrimidin-4-one
3-(morpholine-4-carbonyl)-N-[3-(1H-1,2,3,4-tetrazol-1-yl)phenyl]piperidine-1-carboxamide
3-({[1-(hydroxymethyl)cyclopropyl]carbamoyl}methyl)-N-(2-methoxyethyl)-4-methyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
2-(butylsulfanyl)-5-{[3-(5-methyl-1,2,4-oxadiazol-3-yl)piperidin-1-yl]methyl}pyrimidine
1-[3-(2-methylphenoxymethyl)piperidin-1-yl]-2-(1H-pyrazol-1-yl)ethan-1-one
3-({[1-(dimethyl-1,3-thiazol-2-yl)propyl]carbamoyl}amino)-4-methoxy-N-methylbenzamide
1-cyclopropanecarbonyl-N-[4-(3-fluorophenyl)phenyl]piperidine-3-carboxamide
N-({2-[4-(2-methoxyphenyl)piperazin-1-yl]pyridin-3-yl}methyl)-2-oxo-1,3-oxazolidine-4-carboxamide
5-{1-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)benzoyl]pyrrolidin-2-yl}thiophene-2-carboxamide
(4aS,7aR)-6,6-dioxo-N-(propan-2-yl)-4-(pyridine-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
4-[4-(2-chlorophenoxy)piperidine-1-carbonyl]-N-methyl-1,3-thiazol-2-amine
(1s,4s)-4-{[2-methyl-4-(2-methylphenyl)piperazin-1-yl]methyl}cyclohexan-1-amine