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5-methyl-N-(2,3,4,9-tetrahydro-1H-carbazol-6-ylmethyl)pyrazine-2-carboxamide
N-[(6-chloro-1H-1,3-benzodiazol-2-yl)methyl]-3-(1-phenylethyl)-1,2-oxazole-5-carboxamide
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-ethyl-N-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]benzamide
(3R,4R)-1-{[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]methyl}-4-(morpholin-4-yl)piperidin-3-ol
N-ethyl-N-[2-(5-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-2,2-dimethyloxane-4-carboxamide
ethyl 2-{1-[1-(difluoromethyl)-1H-pyrazole-3-carbonyl]piperidin-2-yl}acetate
N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-N,3-dimethyl-1-propyl-1H-pyrazole-4-carboxamide
5-(3,5-dimethyl-1H-pyrazol-4-yl)-1,3-benzothiazol-2-amine
(1R,5S,6R,7S)-6-[4-(4-ethyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-3-methyl-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
1-[3-(4-methylphenoxymethyl)piperidin-1-yl]-3-(4H-1,2,4-triazol-4-yl)propan-1-one
2-methoxy-5-(1-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-1H-1,2,3-triazol-4-yl)pyridine
3-[(1-acetylpiperidin-4-yl)oxy]-4-methoxy-N-methyl-N-(oxan-2-ylmethyl)benzamide
(2S,4S)-1-[(2,3-dimethoxyphenyl)methyl]-N-(propan-2-yl)-4-({[2-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
2-{4-[2-(benzyloxy)ethyl]phenyl}-N,N-dimethylacetamide
2-[9-oxo-8-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-2-yl]pyridine-3-carbonitrile
3-{3-[3-(4-fluorophenyl)oxolan-3-yl]-1,2,4-oxadiazol-5-yl}-2-methylpyridine
3-[(5-{3-[(4-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}pyridin-2-yl)amino]-2,2-dimethylpropan-1-ol
2-[(4-benzylpiperazin-1-yl)methyl]-N-methyl-N-propyl-1,3-oxazole-4-carboxamide
4-(1-methyl-4-{2-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl}-1H-pyrazolo[3,4-d]pyrimidin-6-yl)pyridine
5-{1-[(8-methoxy-2H-chromen-3-yl)methyl]pyrrolidin-2-yl}-3-methyl-1,2-oxazole
2-{[(1S,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}benzonitrile
2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)-N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}acetamide
methyl (2S,3S)-2-{[1-cyclopentyl-4-oxo-5-(piperidine-1-carbonyl)-1,4-dihydropyridin-3-yl]formamido}-3-methylpentanoate
1-{2-[(2,2-dimethylpyrrolidin-1-yl)methyl]-6-methoxyphenoxy}-3-(morpholin-4-yl)propan-2-ol
5-methanesulfonyl-2-(4-phenylpiperazin-1-yl)-4-(piperidin-3-yl)pyrimidine
3-[(3R,4S)-1-[(dimethyl-1,2-oxazol-4-yl)methyl]-4-(morpholin-4-yl)piperidin-3-yl]propan-1-ol
1-[2-(3-chlorophenyl)ethyl]-2-(methoxymethyl)-6-methyl-4-oxo-N-[(2-oxo-2,3-dihydro-1H-indol-3-yl)methyl]-1,4-dihydropyridine-3-carboxamide
N-[4-(1H-pyrazol-5-yl)phenyl]-1-(1,3-thiazol-2-ylmethyl)piperidine-3-carboxamide
5-[(4-chlorophenyl)methyl]-N-[2-(dimethylamino)ethyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
5-[1-(3,5-dimethyl-1H-pyrrole-2-carbonyl)piperidin-4-yl]-5-propyl-3-[2-(pyridin-2-yl)ethyl]imidazolidine-2,4-dione
1-[(4S)-4-hydroxy-4-(methoxymethyl)-3,3-dimethylpiperidin-1-yl]-2-[(2-methylphenyl)sulfanyl]ethan-1-one
N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-(2-methoxyethyl)quinoline-4-carboxamide
N-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)-3-phenyl-3-(pyridin-2-yl)propanamide
[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]({6-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]imidazo[2,1-b][1,3]thiazol-5-yl}methyl)methylamine
3-(1-cyclopentyl-4-methyl-1H-pyrazol-5-yl)-1-(2-methoxyethyl)-1-(1,3-thiazol-2-ylmethyl)urea
N-{[5-(dimethylcarbamoyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-1,3-thiazole-4-carboxamide
(3aR,6aR)-2-(prop-2-en-1-yl)-5-[4-(trifluoromethyl)pyrimidin-2-yl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
8-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-1-(3-methylbutyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl}-2,8-diazaspiro[4.5]decane-3-carboxamide
1-[4-(4-fluorophenyl)-1,4-diazepan-1-yl]-2-(pyrazin-2-yl)ethan-1-one
(2S,4R)-4-amino-1-[(5-methoxy-1H-indazol-3-yl)methyl]-N-methylpyrrolidine-2-carboxamide
N-methyl-2-[(prop-2-en-1-yl)amino]-N-[3-(1H-pyrazol-1-yl)propyl]benzamide
9-(1-methyl-1H-pyrazole-3-carbonyl)-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-{1-[(4-fluorophenyl)methyl]-4-[(4-phenyl-1,3-thiazol-2-yl)methyl]piperazin-2-yl}ethan-1-ol
2-[4-(4-cyano-4-phenylpiperidine-1-carbonyl)piperidin-1-yl]acetamide
1-(2-methoxy-4-{[(pyridin-3-ylmethyl)amino]methyl}phenoxy)-3-(thiomorpholin-4-yl)propan-2-ol
5-methyl-N-[2-(1-propylpiperidin-4-yl)ethyl]pyrimidin-2-amine
3-(1H-imidazol-1-ylmethyl)-1-{[5-(4-methoxyphenyl)furan-2-yl]methyl}piperidine
2,2,6,6-tetramethyl-4-({3-propyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}methyl)piperidine
7-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-4-[(2E)-2-methylbut-2-en-1-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepine