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1-{1-[(3-ethyl-1H-pyrazol-5-yl)methyl]piperidin-4-yl}-3-(pyrrolidine-1-carbonyl)piperidine
2-[methyl(pyridin-4-ylmethyl)amino]-N-[1-(3-phenylpropyl)piperidin-3-yl]acetamide
4-(4-benzylpiperazin-1-yl)-2-[(2-chlorophenyl)methyl]-2,3-dihydro-1H-isoindole-1,3-dione
4-{4-[1-(3,5-dimethoxyphenyl)-1H-imidazol-2-yl]-1H-1,2,3-triazol-1-yl}piperidine
[(1-methyl-1H-pyrazol-4-yl)methyl](2-methylpropyl){[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}amine
(1R,2S,6R,7S)-4-[4-(methoxymethyl)-5-methyl-1,2-oxazole-3-carbonyl]-4-azatricyclo[5.2.2.02,6]undecane
N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-1-methyl-6-oxo-1,6-dihydropyridine-3-carboxamide
8-({3-methylimidazo[1,5-a]pyridin-1-yl}methyl)-3-(2-phenylpropyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-(1-phenylpiperidin-4-yl)-2-(1-propylpiperidin-4-yl)acetamide
2-methyl-N-{2-[2-(pyridin-4-yl)-1,3-thiazol-4-yl]ethyl}-1-benzofuran-5-carboxamide
N-methyl-2-{[4-(3-methyl-1-propyl-1H-pyrazol-4-yl)pyrimidin-2-yl]amino}ethane-1-sulfonamide
N-(1-butyl-4-methyl-1H-pyrazol-5-yl)-2-(quinazolin-4-yloxy)acetamide
N-[(3S,7S,8aS)-3-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3-bromobenzamide
4-[2-(pyridin-3-yl)pyrimidine-5-carbonyl]thiomorpholine
N-methyl-N-[(5-{[methyl({2-[(4-methylphenyl)sulfanyl]ethyl})amino]methyl}furan-2-yl)methyl]methanesulfonamide
9-methoxy-7-(3-methoxyphenyl)-4-[(3-methylthiophen-2-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
(3R,5R)-5-(morpholine-4-carbonyl)-N-{[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}piperidine-3-carboxamide
4-[4-(2-methoxyacetamido)-1H-pyrazol-1-yl]-N-[1-(1-phenyl-1H-pyrazol-4-yl)ethyl]benzamide
2-cyclopropyl-N-[(2-phenyl-1,3-thiazol-5-yl)methyl]-1,3-benzoxazole-6-carboxamide
N-(1-{1-[(2-cyanophenyl)methyl]-1,2,5,6-tetrahydropyridin-3-yl}propyl)-N-methylacetamide
2-(cyclopropylmethyl)-8-[2-(methylamino)pyrimidine-5-carbonyl]-2,8-diazaspiro[5.5]undecan-3-one
3-(dimethyl-1H-1,2,4-triazol-3-yl)-1-(furan-3-ylmethyl)-1-methylurea
({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)(methyl)[3-(1H-pyrazol-1-yl)propyl]amine
2-(4-{5-cyclopropyl-1-[4-(2-methoxyphenyl)pyrimidin-2-yl]-1H-pyrazole-4-carbonyl}piperazin-1-yl)phenol
2-(2H-1,3-benzodioxol-5-ylmethyl)-4-{4-[4-(pyridin-2-yl)piperazine-1-carbonyl]piperidin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
2-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1H,2H-pyrrolo[1,2-d][1,2,4]triazin-1-one
(1S,5R)-6-[5-(methoxymethyl)thiophene-2-carbonyl]-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
2-amino-4-[1-(4-methylpyridin-2-yl)-1H-pyrrol-2-yl]-6-(1H-pyrrol-2-yl)pyridine-3-carbonitrile
2-[2-(methylsulfanyl)propyl]-1H-1,3-benzodiazole-5-carbonitrile
5-(2-chlorophenyl)-N-[(1-cyclopropyl-5-oxopyrrolidin-3-yl)methyl]furan-2-carboxamide
(1R,5R)-3-(2-chloro-4,5-difluorobenzoyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonane
N-(1-{7-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)pyridine-3-carboxamide
N,2,6,8-tetramethyl-N-(thian-4-yl)quinoline-4-carboxamide
(2S,4R)-1-[(2-aminopyridin-3-yl)methyl]-N-ethyl-4-[2-(methylsulfanyl)acetamido]pyrrolidine-2-carboxamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-4-methoxy-N-{[7-(methylsulfanyl)-2-(morpholin-4-yl)quinolin-3-yl]methyl}benzamide
1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-4-{2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperazine
(2R)-1-(dimethyl-1,3-thiazole-4-carbonyl)pyrrolidine-2-carboxamide
3-{5-[(3-cyanophenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-N-cyclopropylpropanamide
5-{[(3-tert-butyl-1H-pyrazol-5-yl)methyl](methyl)carbamoyl}-2,1,3-benzoxadiazol-1-ium-1-olate
1-[2-(1-{3-azaspiro[5.5]undecan-9-yl}piperidin-4-yl)ethyl]pyrrolidin-2-one
[(3-{2-[1-(2H-1,3-benzodioxole-5-carbonyl)piperidin-2-yl]ethoxy}phenyl)methyl](methyl)(quinolin-8-ylmethyl)amine
3-(3,5-dimethyl-1H-pyrazol-1-yl)-1-[(3R,5R)-3-(hydroxymethyl)-5-(pyrrolidin-1-ylmethyl)piperidin-1-yl]propan-1-one
9-[5-(propan-2-yl)-1,3,4-thiadiazol-2-yl]-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
N-methyl-N-[(3-methylpyridin-4-yl)methyl]-4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzamide
9-methyl-3-(2-methyl-5-propylpyrimidin-4-yl)-3,9-diazaspiro[5.6]dodecan-10-one
(4aS,8aR)-6-(5-fluoropyrimidin-2-yl)-1-[2-(1H-imidazol-4-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
methyl[3-(methylsulfanyl)propyl](quinolin-5-ylmethyl)amine
2-butyl-8-(1-methyl-6-oxo-1,6-dihydropyridazine-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
2-({1-cyclohexyl-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}methyl)-1-ethyl-1H-imidazole
4-[(2E)-3-[4-(dimethylamino)phenyl]prop-2-en-1-yl]-1-[(2-methyl-1,3-thiazol-4-yl)methyl]-6-(pyridin-2-ylmethoxy)-1,4-diazepan-2-one