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1-(5-chloropyridin-2-yl)-4-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperazine
2-(4-{[4-(1-hydroxypropyl)piperidin-1-yl]methyl}phenoxy)acetamide
1-(cyclohexylmethyl)-N,N-dimethyl-5-[(2-phenylethyl)amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-(dimethylamino)-2-(4-methylphenyl)-1-{4-[2-(pyrrolidin-1-yl)ethyl]piperazin-1-yl}ethan-1-one
2-[1-(2H-1,3-benzodioxol-5-yl)propan-2-yl]-1-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}-1H-imidazole
1-[(2S,4R)-1-[(2-ethoxyphenyl)methyl]-4-[(4-methoxyphenyl)sulfanyl]pyrrolidine-2-carbonyl]-4-methyl-1,4-diazepane
1-{[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}-N,N-dimethylpyrrolidin-3-amine
N-tert-butyl-2-{pyrazolo[1,5-a]pyrimidin-3-yl}benzene-1-sulfonamide
(4aS,8aR)-6-(furan-2-ylmethyl)-1-[2-(5-methylfuran-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
[(3-tert-butyl-1H-pyrazol-5-yl)methyl][(8-chloroquinolin-2-yl)methyl]methylamine
6-cyclopentyl-1-methyl-N-[1-(3-methylpyridin-2-yl)propyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
3-amino-1-[4-(dimethylamino)-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]propan-1-one
N-(2,3-dihydro-1H-inden-2-yl)-7-(propan-2-yl)-N-propyl-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2-(pyridin-3-yl)acetamide
1-{[3-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-4-[2-(methylsulfanyl)ethyl]piperazine
1-methyl-3-(piperidine-1-carbonyl)-N-[2-(thiophen-2-yl)ethyl]-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-(benzylsulfamoyl)-N,1-dimethylpyrrolidin-3-amine
N-[2-(methylsulfanyl)ethyl]-1-propyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-({1-[(3-chlorophenyl)methyl]pyrrolidin-3-yl}methyl)cyclobutanecarboxamide
4-[1-(cyclohexylmethyl)-1H-1,2,3-triazole-4-carbonyl]-1-[(3-fluorophenyl)methyl]piperazin-2-one
{3-benzyl-1-[1-(3-methoxyphenyl)piperidin-4-yl]piperidin-3-yl}methanol
1-[1-(1-methyl-1H-pyrrole-2-carbonyl)piperidin-3-yl]-2-phenylethan-1-one
2-[(2-ethyl-6-methylpyridin-3-yl)oxy]-1-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}ethan-1-one
2-amino-4-(2,5-dimethoxyphenyl)-6-(furan-2-yl)pyridine-3-carbonitrile
N-ethyl-N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-2-(morpholin-4-yl)pyridine-3-carboxamide
4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-{[4-(methylsulfanyl)phenyl]methyl}piperidine
(1-ethyl-5-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl)methanol
4-[4-(1-methyl-1H-1,2,4-triazol-5-yl)pyrimidin-2-yl]thiomorpholine
[1-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)-3-(2-phenoxyethyl)piperidin-3-yl]methanol
2-amino-2-(3,5-dimethyl-1H-pyrazol-4-yl)-1-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}ethan-1-one
N-cycloheptyl-2-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
N-[(4-hydroxyazepan-4-yl)methyl]-3,5-dimethylbenzamide
N-(1H-indazol-6-yl)-4-(thiomorpholin-4-yl)piperidine-1-carboxamide
1-[2-(morpholin-4-yl)ethyl]-5-[4-(1H-pyrazol-1-ylmethyl)piperidine-1-carbonyl]piperidin-2-one
1-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-3-(1-ethyl-1H-1,2,3-triazol-4-yl)-1-methylurea
(3S,4R)-1-[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-4-phenylpyrrolidine-3-carboxylic acid
6-[({[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]methyl}amino)methyl]-1,4-oxazepan-6-ol
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-2-(3-oxo-2,3-dihydro-1,2-benzothiazol-2-yl)acetamide
N-(2,3-dihydro-1H-inden-2-yl)-1-(6-fluoro-4-methylquinazolin-2-yl)azepan-4-amine
2-(dimethylamino)-2-(2-fluorophenyl)-1-[4-(2-methoxyacetyl)-1,4-diazepan-1-yl]ethan-1-one
1-cyclopropyl-N-(4-phenylbutyl)-1H-pyrrole-2-carboxamide
(1S,5R)-6-(3-fluoro-4-methoxybenzoyl)-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
2-methyl-N-{[3-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-5-yl]methyl}imidazo[1,2-a]pyrimidine-3-carboxamide
(1S,5R)-3-(2,4-difluorobenzoyl)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-[2-methyl-3-({[(2R)-oxolan-2-ylmethyl]amino}methyl)-1H-indol-1-yl]acetamide
6-{3-oxo-3-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazin-1-yl]propyl}-2,3-dihydropyridazin-3-one
3-[1-(5-acetylthiophene-3-carbonyl)piperidin-4-yl]-1-(morpholin-4-yl)propan-1-one
(2R,3R,6R)-5-(3-ethyl-1,2-oxazole-5-carbonyl)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-[2-(pyrrolidin-1-ylmethyl)phenoxy]-3-(thiomorpholin-4-yl)propan-2-ol
2-{5-[2-(methylamino)-1,3-thiazol-4-yl]-3-(2-methylpropyl)-1H-1,2,4-triazol-1-yl}acetic acid