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N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]acetamide
(1S,5R)-6-benzyl-3-(3-fluoropyridin-4-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-(2-methoxyethyl)-3-[3-(pyridin-3-yl)propyl]-8-(pyridin-4-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-{1-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]piperidin-4-yl}thiomorpholine
N-methyl-3-(1H-pyrazol-1-yl)-N-(thiophen-3-ylmethyl)benzamide
N-methyl-N-{[2-(trifluoromethyl)phenyl]methyl}pyrimidin-4-amine
1-(2-{4-[2-(furan-2-yl)pyrimidin-5-yl]-1H-1,2,3-triazol-1-yl}ethyl)-2,3-dihydro-1H-indole
(2S,4S)-1-(2,3-dihydro-1H-inden-2-yl)-N-(pyridin-3-ylmethyl)-4-{[2-(2,6,6-trimethylcyclohex-1-en-1-yl)ethyl]amino}pyrrolidine-2-carboxamide
5-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidine-1-carbonyl]-2-methyl-1,4-dihydropyridin-4-one
1-(2-ethoxyethyl)-N-methyl-N-[2-(oxan-4-yl)ethyl]-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
2,6-dimethyl-N-{1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}pyrimidine-4-carboxamide
2-[3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazol-5-yl]morpholine
2-[3-(2-fluorophenoxy)azetidine-1-carbonyl]-3,5,7-trimethyl-1H-indole
4-ethyl-3-{1-[(3-fluoro-4-hydroxy-5-methoxyphenyl)methyl]piperidin-4-yl}-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
1-(3-{4-[(2-methylphenyl)methyl]piperazin-1-yl}-3-oxopropyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]quinoxaline-5-carboxamide
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-ethylbenzamide
2-methoxy-1-{2-[(4-methoxyphenyl)methyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-methylpropan-1-one
2-[4-(2,1,3-benzoxadiazol-4-ylmethyl)-1-(cyclohexylmethyl)piperazin-2-yl]ethan-1-ol
2-cyclohexyl-1-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
8-[(1R,2R,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]-2-[(dimethyl-1,2-oxazol-4-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
2-{1-[(3,4-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-(oxan-4-ylmethyl)acetamide
3-[1-(pyrazin-2-yl)propan-2-yl]-3H,4H-thieno[2,3-d]pyrimidin-4-one
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-2-oxo-6-phenyl-1,2-dihydropyridine-3-carboxamide
4-(4-{1-[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]-1H-imidazol-2-yl}-1H-1,2,3-triazol-1-yl)piperidine
7-(6-chloro-2H-chromene-3-carbonyl)-2-oxa-7-azaspiro[4.5]decane
N-[(3R,4S)-1-[4-(hydroxymethyl)-1,3-thiazol-2-yl]-4-propylpyrrolidin-3-yl]-1-(methoxymethyl)cyclopropane-1-carboxamide
(1H-1,3-benzodiazol-2-ylmethyl)(methyl)[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]amine
4-{[3-(morpholin-4-yl)phenyl]methyl}-1,4-oxazepan-6-ol
4-(2,4-difluoro-3-methoxyphenyl)-1-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}-1H-1,2,3-triazole
2-[1-(2-methylpropyl)-4-(quinolin-6-ylmethyl)piperazin-2-yl]ethan-1-ol
4-({2-[1-(2,5-dimethylbenzoyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
2-chloro-N-methyl-N-[2-(morpholin-4-yl)propyl]pyridine-4-carboxamide
1-[(4-fluorophenyl)methyl]-N-[1-(furan-2-yl)ethyl]-N-methyl-1H-1,2,3-triazole-4-carboxamide
N,N-dimethyl-3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-sulfonamide
(4aS,8aR)-1-butyl-6-(4-ethyl-1,2,3-thiadiazole-5-carbonyl)-decahydro-1,6-naphthyridin-2-one
(2,1,3-benzoxadiazol-5-ylmethyl)[4-(1H-pyrazol-1-yl)butan-2-yl]amine
(5-{[benzyl(1,3-thiazol-2-ylmethyl)amino]methyl}furan-2-yl)methanol
2-[1-(2-methoxyphenyl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]-6-(4H-1,2,4-triazol-4-yl)pyridine
2-{1-ethyl-2,5-dioxo-3-[3-(trifluoromethyl)phenyl]pyrrolidin-3-yl}-N-methyl-N-[(5-propyl-1H-pyrazol-3-yl)methyl]acetamide
dimethyl({4-[1-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperidin-2-yl]phenyl}methyl)amine
5-[4-(1H-imidazol-1-ylmethyl)piperidine-1-carbonyl]-1-[3-(morpholin-4-yl)propyl]piperidin-2-one
ethyl[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl][3-(methylsulfanyl)butyl]amine
(2S,4R)-1-[(3-chlorophenyl)methyl]-4-{[(3-methylphenyl)methyl]amino}-N-(propan-2-yl)pyrrolidine-2-carboxamide
4-(4-{[3-(3,4-dimethoxybenzoyl)piperidin-1-yl]methyl}phenyl)but-3-yn-1-ol
6-tert-butyl-1-methyl-N-[3-(4-methylpiperazin-1-yl)propyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-[3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-3-(4-phenyl-1H-pyrazol-5-yl)piperidine
5-[(4-benzylpiperidin-1-yl)methyl]-N-(thiolan-3-yl)-1,2-oxazole-3-carboxamide
N-[1-(4-cyclopentyl-4H-1,2,4-triazol-3-yl)ethyl]-2-(1-propylpiperidin-4-yl)acetamide
2-methyl-8-(6-phenylpyridine-2-carbonyl)-2,8-diazaspiro[4.5]decan-3-one