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1-(2,3-dihydro-1H-indene-5-carbonyl)-4-(2-methylpyridin-4-yl)-1,4-diazepane
1-[3-({4-[(4-chlorophenyl)methyl]-4-(hydroxymethyl)piperidin-1-yl}methyl)phenyl]ethan-1-one
3-(3-chlorobenzoyl)-1-(1,4-dithiepan-6-yl)piperidine
(3S,4R)-1-(2-oxo-1,2,5,6,7,8-hexahydroquinoline-3-carbonyl)-4-(pyridin-4-yl)pyrrolidine-3-carboxylic acid
2-[1-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)azetidin-3-yl]pyridine
(2S)-2-[(4-ethoxypyrimidin-2-yl)amino]-3-phenylpropanamide
3-[(3R,4S)-1-[5-fluoro-4-(methylamino)pyrimidin-2-yl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
1-[2-(dimethylamino)-6-(pyrazin-2-yl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-4-yl]piperidin-4-ol
8-(3-ethoxypropanoyl)-3-(2-phenylethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-[5-chloro-2-(1H-1,2,4-triazol-1-yl)phenyl]-3-methyl-3-[(5-propyl-1,2,4-oxadiazol-3-yl)methyl]urea
N-[(4-{[(2-fluorophenyl)methyl]amino}-8-methylquinazolin-2-yl)methyl]methanesulfonamide
6-(cyclohex-3-en-1-ylmethyl)-1-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carbonyl}-6-azaspiro[2.5]octane
4-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)thiomorpholine
N-(3,4-difluorophenyl)-1-(2,3-dihydro-1-benzofuran-5-ylmethyl)piperidin-3-amine
1-{1-[(3-ethoxy-4-hydroxyphenyl)methyl]piperidin-4-yl}-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
5-methanesulfonyl-2-methyl-N-[2-(1-methyl-1H-pyrazol-5-yl)ethyl]pyrimidin-4-amine
(1-{2-[5-(2-methyl-1H-imidazol-4-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}piperidin-2-yl)methanol
1-({5-[4-(2-phenylethyl)piperidine-1-carbonyl]pyridin-2-yl}amino)propan-2-ol
(3S,7S)-5-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propanoyl]-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-triene-3-carboxylic acid
1-(3-{[4-(4-fluorophenyl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)butan-1-one
N-[2-(4-methylmorpholin-2-yl)ethyl]-2-(2-methylphenyl)benzamide
4-(6-phenylpyridazin-3-yl)-2-(trifluoromethyl)morpholine
N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-3-(1-methylpiperidin-3-yl)propanamide
1-[(3-chloropyridin-4-yl)methyl]-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
2-{[1-cyclohexyl-3-(2-methyl-1,3-thiazol-4-yl)-1H-1,2,4-triazol-5-yl]methyl}morpholine
2-[4-(4-chlorophenyl)-4-hydroxypiperidin-1-yl]-2-(3-hydroxyphenyl)acetic acid
1-(furan-2-yl)-2-[2-(naphthalen-1-ylmethyl)morpholin-4-yl]ethane-1,2-dione
{[2-(furan-2-yl)pyrimidin-5-yl]methyl}(oxolan-2-ylmethyl)(pyridin-4-ylmethyl)amine
7-{[4-(propan-2-yl)phenyl]methyl}-2-(pyridine-2-carbonyl)-2,7-diazaspiro[4.5]decane
N-(3-{[(3-methylphenyl)methyl]sulfanyl}propyl)-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
1-(2-chlorophenyl)-3-{1-[1-(2-oxopropanoyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
1-[4-(3-ethyl-1,2,4-oxadiazol-5-yl)phenyl]-3-{[3-(2-methylpropyl)-1,2-oxazol-5-yl]methyl}urea
2-[1-(2-chlorophenyl)-5-oxo-3-phenyl-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N,N-diethylacetamide
3-[5-(1-ethyl-1H-imidazol-2-yl)-4-phenyl-1H-imidazol-1-yl]butanoic acid
1-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]-4-(pyridin-3-ylmethyl)-1,4-diazepan-5-one
4-amino-5-(2-fluoro-5-methoxyphenyl)-2-(morpholin-4-yl)-5H,6H,7H,8H-pyrido[2,3-d]pyrimidin-7-one
6-ethyl-N-[2-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)propyl]-2-(morpholin-4-yl)pyrimidin-4-amine
7-(3-chlorophenyl)-4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
{[5-(1,5-dimethyl-1H-pyrrol-2-yl)-1,3,4-oxadiazol-2-yl]methyl}(methyl)[1-(1,2-oxazol-3-yl)ethyl]amine
1-(4-{[2-(morpholin-4-yl)quinolin-3-yl]methyl}piperazin-1-yl)ethan-1-one
N-{[1-(1H-imidazol-1-ylmethyl)cyclopropyl]methyl}-5-oxo-1-(propan-2-yl)pyrrolidine-3-carboxamide
(3aS,6aR)-3-[3-(morpholin-4-yl)propyl]-2-oxo-N-phenyl-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazole-5-carboxamide
N-benzyl-3-({[(1,2-dimethyl-1H-imidazol-5-yl)methyl]amino}methyl)-N-methylpyridin-2-amine
2-(3-fluorophenyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1,3-benzoxazole-5-carboxamide
N-(2-{1-[(4-methoxy-3-methylphenyl)methyl]piperidin-3-yl}ethyl)methanesulfonamide
N-methyl-N-(quinoxalin-2-ylmethyl)-2,8-diazaspiro[4.5]decane-3-carboxamide
naphthalen-1-yl (7S,9aR)-7-[(4-methoxyphenyl)methyl]-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxylate
N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-5-(3-methoxyphenyl)-1,2,4-triazin-3-amine
(8R,9aS)-8-hydroxy-2-[2-(3-methylthiophen-2-yl)ethyl]-octahydro-1H-pyrido[1,2-a]piperazine-1,4-dione
3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-1-[(1-methyl-1H-imidazol-4-yl)sulfonyl]piperidine