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N-[1-(furan-2-carbonyl)piperidin-3-yl]-6-(methoxymethyl)pyrimidin-4-amine
4-cyano-4-methyl-N-[2-(2-phenoxyethoxy)phenyl]piperidine-1-carboxamide
1-{[3-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]methyl}-4-(3-methoxypropyl)piperidine
(3R,4R)-3-cyclobutyl-4-methyl-1-(5-phenyl-1,3,4-thiadiazol-2-yl)pyrrolidin-3-ol
methyl 6-(cyclohex-3-en-1-ylmethyl)-2-(piperidine-1-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
2-[methyl(pyridin-2-ylmethyl)amino]-N-{1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl}acetamide
(5-{[4-(4-cyclohexyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]methyl}furan-2-yl)methanol
6-cyano-N-[(3S,5S)-1-cyclopentyl-5-(ethylcarbamoyl)pyrrolidin-3-yl]pyridine-3-carboxamide
N-{[5-methyl-2-(trifluoromethyl)furan-3-yl]methyl}-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
(5S)-5-{4-[(4-cyclohexyl-1H-1,2,3-triazol-1-yl)methyl]piperidine-1-carbonyl}pyrrolidin-2-one
5-methyl-N-(3-methylbutyl)-4-{[3-(morpholin-4-yl)propyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
6-(dimethylamino)-N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}pyridine-3-carboxamide
1-(4-{[(2S)-2-(methoxymethyl)pyrrolidin-1-yl]methyl}-3-methylphenyl)-1H-pyrazole
N,2,3-trimethyl-N-[1-(3-phenylpropyl)piperidin-3-yl]quinoxaline-6-carboxamide
2-(2-hydroxy-3-methylbutanoyl)-N-(thiophen-2-ylmethyl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
3,5-dimethyl-1-({5-methyl-2-[4-(methylsulfanyl)phenyl]-1,3-oxazol-4-yl}methyl)-1H-1,2,4-triazole
1-benzyl-N-(1,3-thiazol-2-ylmethyl)-5-(1,3-thiazole-5-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2,3,5-trimethyl-N-[2-methyl-1-(1-methyl-1H-imidazol-2-yl)propyl]pyrazolo[1,5-a]pyrimidin-7-amine
5-benzyl-1-(3-methoxyphenyl)-4-propanoylpiperazin-2-one
N-[4-(1H-1,3-benzodiazol-2-yl)phenyl]-1-(oxane-2-carbonyl)piperidine-4-carboxamide
3-[2-(dimethylamino)ethyl]-1-ethyl-8-[(4-hydroxyphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-(3-acetamidopropanamido)-N-ethyl-N-phenylbenzamide
{[4-(3-chlorophenyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}(methyl)(2-phenylpropyl)amine
3-(1H-pyrazol-1-yl)-1-[3-(pyridin-3-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]butan-1-one
3-cyclopentyl-N-cyclopropyl-N-[(1-methyl-1,2,3,6-tetrahydropyridin-4-yl)methyl]propanamide
(3S,4R)-1-(5-chloro-2-fluorobenzoyl)-4-methylpiperidine-3,4-diol
N-methyl-3-(methylsulfanyl)-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}propanamide
2-[4-(morpholin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]pyridin-3-ol
1-methyl-N-{[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}azepane-2-carboxamide
5-({ethyl[(1-methyl-1H-imidazol-2-yl)methyl]amino}methyl)-N-(oxolan-2-ylmethyl)pyrimidin-2-amine
4-[3-(4-methoxy-2,6-dimethylphenyl)phenyl]-4H-1,2,4-triazole
(2R)-3-(3,3-diphenylpiperidin-1-yl)propane-1,2-diol
6-[methyl(1,3-thiazol-2-ylmethyl)amino]-N-[2-(1-methylpiperidin-2-yl)ethyl]pyridine-3-carboxamide
N-{2-[4-(4-ethyl-1-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]thiophen-3-yl}acetamide
4-(1-{[3-(1H-pyrazol-1-yl)phenyl]methyl}azetidin-3-yl)pyridine
N-methyl-N-(1-methylpiperidin-4-yl)-3-(1-{[3-(trifluoromethyl)phenyl]methyl}piperidin-3-yl)propanamide
N,4-dimethyl-N-{2-[4-({methyl[(2-methyl-1,3-thiazol-4-yl)methyl]amino}methyl)phenoxy]ethyl}benzamide
N-{1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl}pyridine-4-carboxamide
(1S,6R)-3-{[2-(methylsulfanyl)phenyl]methyl}-3,9-diazabicyclo[4.2.1]nonane
2-{4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]piperidin-1-yl}pyrimidine
4-(1H-imidazol-2-ylmethyl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
4-(1H-imidazol-2-yl)-1-({2-[2-(3-methylpiperidin-1-yl)ethoxy]phenyl}methyl)piperidine
[5-(1H-indol-4-yl)-1H-1,3-benzodiazol-2-yl]methanol
2-[2-(3-methyl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]-N,N-bis(prop-2-en-1-yl)acetamide
1-benzyl-N-methyl-N-[(5-propyl-1H-pyrazol-3-yl)methyl]piperidine-2-carboxamide
(3R,5S)-N-cyclopentyl-5-[3-(trifluoromethyl)phenoxymethyl]piperidine-3-carboxamide
(1H-imidazol-2-ylmethyl)(methyl)[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]amine
2-(2H-1,3-benzodioxol-5-yl)-N-(1-cycloheptylpiperidin-3-yl)acetamide
methyl 2-[4-(6-hydroxy-2-methylpyrimidin-4-yl)piperidine-1-carbonyl]piperidine-1-carboxylate
4-({dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}(ethyl)amino)butan-1-ol