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2-(methoxymethyl)-1-methyl-N-[2-(morpholin-4-yl)ethyl]-5-(2-phenylacetamido)-1H-1,3-benzodiazole-7-carboxamide
N-(2-{[2-(dimethylamino)-4-methylpyrimidin-5-yl]formamido}ethyl)pyridine-3-carboxamide
ethyl 1-[(3-acetylphenyl)methyl]-3-benzylpiperidine-3-carboxylate
5,6-dimethyl-N-[2-(4-methylpiperazin-1-yl)propyl]pyrimidin-4-amine
5-[4-(2-methylphenyl)piperazine-1-carbonyl]-1-(2-phenylethyl)piperidin-2-one
3-[(5-ethylpyridin-2-yl)methyl]-3-methyl-1-{3-[(2-methylpiperidin-1-yl)methyl]phenyl}urea
N-methyl-2-[3-oxo-1-(3-phenylpropyl)piperazin-2-yl]-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
N-(4-{[3-(5-chloro-2-methoxybenzoyl)piperidin-1-yl]methyl}phenyl)acetamide
N-[3-(1H-imidazol-1-yl)butyl]-2,8-dimethylquinoline-4-carboxamide
{1-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]-3-ethylpiperidin-3-yl}methanol
N-(2,3-difluorophenyl)-4-[(1-methylpiperidin-3-yl)methyl]piperazine-1-carboxamide
2-(7-fluoro-2-methyl-1H-indol-3-yl)-N-[2-(pyrrolidine-1-sulfonyl)ethyl]acetamide
[4-(3-phenylpropyl)-1-(pyridin-3-ylmethyl)piperidin-4-yl]methanol
(4aS,7aR)-1-(2-hydroxy-4-methylbenzoyl)-4-(3-methylbut-2-en-1-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-methyl-4-({[(1-methyl-1H-pyrazol-4-yl)methyl](2-methylpropyl)amino}methyl)benzene-1-sulfonamide
5-chloro-4-{[3-(2-hydroxyethyl)-4-[(6-methylpyridin-2-yl)methyl]piperazin-1-yl]methyl}-2-methoxyphenol
3-benzyl-5-(2-ethoxyethyl)-1H-1,2,4-triazole
4-(3-tert-butyl-1H-pyrazol-1-yl)-1-(oxolane-3-carbonyl)piperidine-4-carboxylic acid
N-methyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]-3-(2-methylphenyl)-3-phenylpropanamide
4-methyl-1-{2-[(2E)-2-methylbut-2-en-1-yl]-2,7-diazaspiro[4.5]decan-7-yl}pentan-1-one
2-[3-oxo-1-(thiophen-2-ylmethyl)piperazin-2-yl]-N-[2-(2-oxopiperidin-1-yl)ethyl]acetamide
N-[(5-{[4-(2-hydroxyethoxy)phenyl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)methyl]acetamide
(2S)-2-amino-N-[3-(4-methylphenyl)propyl]-4-(methylsulfanyl)butanamide
4-(1-cyclopropyl-5-oxopyrrolidine-3-carbonyl)-1-[(3-fluorophenyl)methyl]piperazin-2-one
[(3R,4R)-4-{[(2-methoxyethyl)(methyl)amino]methyl}-1-(5-phenyl-1,2,4-oxadiazol-3-yl)pyrrolidin-3-yl]methanol
methyl 2-[3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]benzoate
N-cyclopentyl-3-ethyl-5-methyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)-1,2-oxazole-4-carboxamide
N-cyclopentyl-6-[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
3-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-1-{4-[(furan-2-ylmethyl)sulfanyl]phenyl}-3-methylurea
N-[(3R,4S)-1-acetyl-4-phenylpyrrolidin-3-yl]morpholine-4-sulfonamide
(3aR,6aR)-2-cyclopropanecarbonyl-5-(6-methoxypyrimidin-4-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-(4-benzylpiperidin-1-yl)-3-[1-(pyridine-3-carbonyl)piperidin-4-yl]propan-1-one
4-(3-fluorophenoxy)-1-[5-(1H-imidazol-1-ylmethyl)furan-2-carbonyl]piperidine
(1S,6R)-9-[4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzoyl]-3,9-diazabicyclo[4.2.1]nonane
2-(4-hydroxyhepta-1,6-dien-4-yl)-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
3-{1-[2-(2H-1,3-benzodioxol-5-yl)acetyl]piperidin-4-yl}-4-ethyl-4,5-dihydro-1H-1,2,4-triazol-5-one
1-{2-[4-(2-methylpyridin-4-yl)-1,4-diazepan-1-yl]pyrimidin-4-yl}piperidin-3-ol
2-(4-chlorophenyl)-4-[2-(pyridin-3-yl)-1,3-thiazole-4-carbonyl]morpholine
4-(cyclopropylmethyl)-3-(propan-2-yl)-1-[2-(4H-1,2,4-triazol-4-yl)pyridine-4-carbonyl]-1,4-diazepan-5-one
8-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}-1,3-dioxa-8-azaspiro[4.5]decan-2-one
1-[5-(methoxymethyl)furan-2-carbonyl]-4-phenoxypiperidine-4-carboxylic acid
2-(dimethylamino)-N-methyl-N-[4-(morpholin-4-yl)butyl]-2,3-dihydro-1H-indene-2-carboxamide
2-(3,5-dimethyl-1H-pyrazol-1-yl)-1-{4-[2-(2-methoxyphenoxymethyl)-3H-imidazo[4,5-b]pyridin-3-yl]piperidin-1-yl}ethan-1-one
2-[({6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)methyl]-3,5-dimethylpyridin-4-ol
1-{4-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]-4-oxobutyl}pyrrolidin-2-one
N-cyclopentyl-N-{[4-methoxy-3-(thiophen-2-ylmethoxy)phenyl]methyl}propanamide
3-({[(1,3-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}methyl)-1-(2,2-dimethylpropyl)-3-hydroxypiperidin-2-one
(3S,4S)-1-[6-(hydroxymethyl)pyridine-2-carbonyl]-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
ethyl 1-(4-acetylbenzoyl)-3-[(3-chlorophenyl)methyl]piperidine-3-carboxylate
N4-[2-(2-chlorophenoxy)ethyl]-N2,N2-dimethyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-2,4-diamine