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2-{[2-(1H-1,2,3-benzotriazol-1-yl)ethyl]amino}pyridine-3-carboxamide
5-ethyl-N-{[1-(4-methylpiperazin-1-yl)cyclohexyl]methyl}pyrimidin-2-amine
1-(4-{4-[(1R,5S)-6-azabicyclo[3.2.1]octane-6-carbonyl]-2-methoxyphenoxy}piperidin-1-yl)ethan-1-one
7-[(3aR,6aS)-octahydropyrrolo[3,4-c]pyrrol-2-yl]-2,3,5-trimethylpyrazolo[1,5-a]pyrimidine
N5-[(5-fluoro-2-methylphenyl)methyl]-N3-methyl-N3-(2-methylpropyl)-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
1-methyl-4-({5-[(4-methyl-1H-pyrazol-1-yl)methyl]-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-3-yl}methyl)piperidine
1-{4-[methyl(2-phenylethyl)amino]-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-2-[1-(propan-2-yl)piperidin-4-yl]acetamide
3,3-dimethyl-1-[6-(morpholine-4-sulfonyl)-1,2,3,4-tetrahydroisoquinolin-2-yl]butan-1-one
N-[3-(2-methoxyacetamido)-2-methylphenyl]-2-(methoxymethyl)piperidine-1-carboxamide
N-[(3-methoxyphenyl)methyl]-N-methyl-1-[3-(1H-pyrazol-5-yl)phenyl]piperidin-4-amine
5-methyl-4-{3-methyl-1-phenyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-1-(prop-2-en-1-yl)-1H-pyrazole
4-(3-hydroxy-4-methylbenzoyl)-1-(3-methoxyphenyl)piperazin-2-one
{[6-(azocane-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}(methyl)[2-(morpholin-4-yl)ethyl]amine
2-{1-ethyl-8-[(1-methyl-1H-indol-3-yl)methyl]-2,4-dioxo-1,3,8-triazaspiro[4.5]decan-3-yl}acetamide
4-ethyl-3-{1-[(5-fluoro-3-methyl-1H-indol-2-yl)methyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
5-(1-cyclopropanecarbonylpiperidine-4-carbonyl)-4H,5H,6H,7H-[1,3]thiazolo[5,4-c]pyridin-2-amine
1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-4-(4-methoxyphenyl)-2-methylpiperazine
N-(2-methoxyethyl)-6-methyl-N-(pyridin-4-ylmethyl)imidazo[1,2-a]pyridine-2-carboxamide
8-[(dimethyl-1,2-oxazol-4-yl)methyl]-2-(dimethylamino)-1,3,8-triazaspiro[4.5]dec-1-en-4-one
1-[(3-ethoxyphenyl)methyl]-3-(1-ethyl-1H-1,2,4-triazol-3-yl)-1-methylurea
2-(2,4-dimethyl-6-oxo-1,6-dihydropyrimidin-5-yl)-N-[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]acetamide
N,1-diethyl-N-(2-methylprop-2-en-1-yl)-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-cyclopropyl-3-{1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}propanamide
N-[3-(2,3-dihydro-1H-indol-1-yl)propyl]-5-phenyl-1,2-oxazole-3-carboxamide
N-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-3-[(thiophen-2-ylmethyl)amino]benzamide
(3aS,6aS)-5-[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-1-oxo-2-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(3S,4S)-3-hydroxy-N-[3-(4-methylphenyl)phenyl]-4-(piperidin-1-yl)pyrrolidine-1-carboxamide
6-methyl-2-({[(5-methyl-1H-pyrazol-3-yl)methyl]amino}methyl)quinolin-4-ol
5-oxo-1-[(2-phenyl-1,3-oxazol-4-yl)methyl]pyrrolidine-3-carboxylic acid
5-[(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-2-methyl-1,4-dihydropyridin-4-one
{[3-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-5-yl]methyl}(methyl)[1-(thiophen-2-yl)ethyl]amine
3-oxo-N-(2-phenylethyl)-2,8-diazaspiro[4.5]decane-8-carboxamide
1-[3-(N-methylmethanesulfonamido)propanoyl]-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
N-[1-({5-methyl-2-[4-(methylsulfanyl)phenyl]-1,3-oxazol-4-yl}methyl)piperidin-4-yl]acetamide
(1S,6R)-9-(4,5,6,7-tetrahydro-1-benzothiophene-2-carbonyl)-3,9-diazabicyclo[4.2.1]nonan-4-one
2-{[1-(3,5-difluorophenyl)ethyl]amino}-N-(3-fluoro-2-methylphenyl)acetamide
1-{3-[4-(naphthalen-1-yl)-1H-pyrazol-5-yl]piperidin-1-yl}butan-1-one
2-{5-cyclopropyl-4-[4-(propan-2-yl)piperazine-1-carbonyl]-1H-pyrazol-1-yl}-4-(2-methoxyphenyl)pyrimidine
1-{2-[(2R,3R,6R)-3-(3-hydroxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-oxoethyl}piperidin-2-one
(3S,4R)-1-(2,1,3-benzoxadiazol-4-ylmethyl)-N,N-dimethyl-4-(4-methylphenyl)pyrrolidin-3-amine
N-cyclohexyl-4-hydroxy-N-[2-(1H-indol-3-yl)ethyl]-2-methylpyrimidine-5-carboxamide
1-[(4-chlorophenyl)methyl]-6-oxo-N-(2-phenoxyethyl)piperidine-3-carboxamide
3-[(oxolan-3-ylmethyl)sulfamoyl]-N-(pyrimidin-4-ylmethyl)benzamide
(1r,4r)-4-({[2-(azepane-1-carbonyl)-7-methylimidazo[1,2-a]pyridin-3-yl]methyl}amino)cyclohexan-1-ol
3-amino-1-{[2-(naphthalen-1-yl)pyrimidin-5-yl]methyl}pyrrolidine-3-carboxylic acid
6-(2,5-dimethylfuran-3-yl)-N-ethyl-N-methyl-7-(3-methylbut-2-en-1-yl)-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
3-(3-hydroxy-1,2-oxazol-5-yl)-1-[4-(morpholin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]propan-1-one
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-4-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}butanamide
8-(2-propoxyacetyl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one