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1-methyl-2-[1-(oxolan-3-ylmethyl)piperidin-4-yl]-1H-1,3-benzodiazole
N-methyl-N-[(1-phenylpyrrolidin-3-yl)methyl]-2-(pyridin-2-ylsulfanyl)acetamide
N3-benzyl-N5-ethyl-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
7-{[(3S,4S)-3,4-dihydroxy-4-methylpiperidin-1-yl]methyl}-2-(methylsulfanyl)-5H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one
N-[(6-methylpyridin-2-yl)methyl]-2-[1-(naphthalen-2-ylmethyl)-3-oxopiperazin-2-yl]acetamide
8-[(3-chloro-4-fluorophenyl)methyl]-2-[2-(dimethylamino)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
2-[(1R,5S)-3,8-diazabicyclo[3.2.1]octan-8-ylmethyl]-5,8-dimethylquinolin-4-ol
(4aS,8aR)-6-(1H-imidazol-2-ylmethyl)-1-(2-methylpropyl)-decahydro-1,6-naphthyridin-2-one
ethyl 2-(4-{[6-(azocane-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}morpholin-3-yl)acetate
2-(2H-1,3-benzodioxol-5-yl)-1-[3-(2-chlorophenoxy)azetidin-1-yl]ethan-1-one
1-methyl-4-{4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine-1-carbonyl}-1,2,3,4-tetrahydroquinolin-2-one
N-(1-hydroxybutan-2-yl)-N-(pyridin-2-ylmethyl)-2-(trifluoromethyl)benzamide
2-(2-ethyl-1H-1,3-benzodiazol-1-yl)-1-(3-hydroxyazetidin-1-yl)butan-1-one
1-[(4-chlorophenyl)methyl]-N-ethyl-N-(4-hydroxybutyl)-6-oxopiperidine-3-carboxamide
N-[(4-methyl-2-propyl-1,3-thiazol-5-yl)methyl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
5-[(1s,4s)-4-aminocyclohexyl]-1H,5H,6H,7H,8H-pyrido[3,2-f]indazol-7-one
6-[({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)amino]pyridine-3-carboxamide
3-(2,5-dioxoimidazolidin-4-yl)-N-[2-(6-oxo-3-phenyl-1,6-dihydropyridazin-1-yl)ethyl]propanamide
3-methoxy-2-({3-[2-(methylsulfanyl)benzoyl]piperidin-1-yl}methyl)phenol
1-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}-4-(pyrrolidin-1-ylmethyl)piperidine
N-[3-(1H-imidazol-1-yl)propyl]-2-methyl-4-phenylpyridine-3-carboxamide
2-{2-[4-phenyl-1-(pyridin-2-ylmethyl)-1H-imidazol-5-yl]-1H-pyrrol-1-yl}pyridine
1-[(4-methoxyphenyl)methyl]-4-(5-methyl-1H-pyrazole-3-carbonyl)-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
2-(4-methyl-6-{4-[(oxan-4-yl)amino]piperidin-1-yl}pyrimidin-2-yl)phenol
3-[(4-butyl-1H-1,2,3-triazol-1-yl)methyl]-1-cyclopentanecarbonylpiperidine
N-{1-[2-(3-chlorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-4-(1H-pyrazol-1-yl)butanamide
3-[5-(2,3-dihydro-1-benzofuran-5-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]-N-(propan-2-yl)propanamide
2-({[2-(dimethylamino)-6-methylpyrimidin-4-yl]amino}methyl)-N,N-dimethyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
1-(2-hydroxyethyl)-N-(1-phenylethyl)-5-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
[(3R,4R)-4-{[ethyl(methyl)amino]methyl}-1-(pyridine-3-carbonyl)pyrrolidin-3-yl]methanol
6-chloro-2-(2-methoxyphenyl)quinoline
1-(3-chlorophenyl)-4-[(4-{[1-(3-methylthiophene-2-carbonyl)piperidin-4-yl]oxy}phenyl)methyl]piperazine
N-(2-fluoroethyl)-2-{[1-(pyridine-3-carbonyl)piperidin-4-yl]oxy}benzamide
N-butyl-2-methyl-N-(pyridin-3-ylmethyl)-2,8-diazaspiro[4.5]decane-3-carboxamide
4-{3-[(4aS,7aS)-octahydro-1H-pyrrolo[3,4-b]pyridine-6-sulfonyl]benzoyl}morpholine
({2,4-dimethyl-5-[(4-methylpiperazin-1-yl)methyl]phenyl}methyl)(methyl)(pyrazin-2-ylmethyl)amine
5-[5-methyl-1-(pyridin-2-yl)-1H-pyrazole-4-carbonyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylic acid
2-[(1-methanesulfonylpiperidin-4-yl)oxy]-N-(1-phenylethyl)benzamide
(5-{1-[1-(pyrimidin-2-yl)piperidin-3-yl]-1H-1,2,3-triazol-4-yl}furan-2-yl)methanol
(3R,4R)-4-(hydroxymethyl)-1-[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl]piperidin-3-ol
2-(2-phenyl-1H-imidazol-1-yl)-N-{[3-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
2-methoxy-5-methyl-N-{1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}benzene-1-sulfonamide
N-(2-methylpropyl)-4-oxo-N-(pyridin-2-ylmethyl)-4,5,6,7-tetrahydro-1-benzofuran-3-carboxamide
N-[(1-benzylpiperidin-4-yl)methyl]-2-(2,5-dioxoimidazolidin-4-yl)-N-methylacetamide
1-ethyl-4,6-dimethyl-3-[(2S)-2-(morpholine-4-carbonyl)pyrrolidine-1-carbonyl]-1,2-dihydropyridin-2-one
N-(1-{1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)pyridine-3-carboxamide
N-[4-(2,2-dimethylpropanamido)-3-methoxyphenyl]-4-(1H-1,2,4-triazol-5-yl)benzamide
4-{3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidin-2-amine
1-(3-{1-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]-1H-imidazol-2-yl}phenyl)ethan-1-one
2-methyl-N-[1-(1-methyl-1,2,3,6-tetrahydropyridin-4-yl)propyl]-3-(trifluoromethyl)benzamide