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3-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N,N-dimethylpropanamide
2-ethyl-4-methyl-N-(3-methyl-1,2,4-thiadiazol-5-yl)-3-oxopiperazine-1-carboxamide
3-(3-fluorophenyl)-1-{3-[(4-methoxyphenyl)amino]piperidin-1-yl}propan-1-one
3-[2-(2-chloro-6-fluorophenyl)acetyl]-7-methyl-3,7,11-triazaspiro[5.6]dodecan-12-one
3-ethyl-8-(2,3,4,9-tetrahydro-1H-carbazole-1-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-(carbamoylmethyl)-N-[cyclopropyl(1-methyl-1H-imidazol-2-yl)methyl]piperidine-4-carboxamide
N-ethyl-3,5-dimethyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)furan-2-carboxamide
2-(2,4-dimethoxyphenyl)-2-[methyl(pyridin-2-ylmethyl)amino]acetic acid
N-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-N,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
N-[4-(3-{1-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-1H-pyrazol-3-yl}phenyl)phenyl]-N-methylacetamide
1-(2-methoxyphenyl)-3-{1-[1-(1-phenoxypropan-2-yl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
(2S,3R)-2-{[6-(3-fluoro-4-methoxyphenyl)imidazo[2,1-b][1,3]thiazol-3-yl]formamido}-3-hydroxybutanamide
7-fluoro-N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-2-methylquinoline-4-carboxamide
3-[(3S,7S,8aS)-1,4-dioxo-3-(propan-2-yl)-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(3-chloro-2-methylphenyl)urea
3-{[1-(hydroxymethyl)-9-(pyridin-4-ylmethyl)-3,9-diazaspiro[5.5]undecan-3-yl]methyl}benzonitrile
2-{4-[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]piperazin-1-yl}-N-ethylacetamide
(2R,3S,6R)-5-benzoyl-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-ethoxy-4-[1-(furan-2-ylmethyl)-1H-imidazol-2-yl]phenol
1-(cyclopent-3-en-1-yl)-5-(4-methanesulfonylphenyl)-4-phenyl-1H-imidazole
N-(1-methyl-3-phenyl-1H-pyrazol-5-yl)-2-oxo-1-oxa-3,8-diazaspiro[4.6]undecane-8-carboxamide
2-{4-[2-(2-methoxyphenyl)acetamido]-1H-pyrazol-1-yl}-N-[2,2,2-trifluoro-1-(furan-2-yl)ethyl]acetamide
1-(cyclobutylmethyl)-3-({[(2,3-difluoro-4-methylphenyl)methyl]amino}methyl)-3-hydroxypiperidin-2-one
4-[2-(dimethyl-1,3-thiazol-5-yl)acetyl]-1-[(4-methylphenyl)methyl]piperazin-2-one
2-amino-3-ethyl-N-{pyrazolo[1,5-a]pyridin-3-ylmethyl}-3H-imidazo[4,5-b]pyridine-6-carboxamide
7-[(2,3-difluorophenyl)methyl]-2-(2,2-dimethylpropanoyl)-2,7-diazaspiro[4.5]decan-6-one
N-cyclopropyl-2-(methylamino)-N-(thiophen-3-ylmethyl)pyridine-4-carboxamide
2-(2,6-dimethylphenyl)-2-{methyl[2-(morpholin-4-yl)ethyl]amino}acetic acid
N-[2-(4-methoxyphenyl)ethyl]-N-[(1-methylpiperidin-4-yl)methyl]-2-oxoimidazolidine-4-carboxamide
N-(2-hydroxyethyl)-6-methyl-N-[(trimethyl-1H-pyrazol-4-yl)methyl]imidazo[2,1-b][1,3]thiazole-5-carboxamide
methyl[3-(1-methyl-1H-imidazol-2-yl)propyl](2-phenylpropyl)amine
N-benzyl-5-(1,2,3,4-tetrahydroisoquinolin-5-yl)furan-2-carboxamide
2-(2-ethyl-1H-imidazol-1-yl)-1-[2-methyl-4-(4-methylphenyl)piperazin-1-yl]ethan-1-one
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3-(pyridin-3-yl)propanamide
[(6-ethoxypyridin-3-yl)methyl](methyl)(quinolin-3-ylmethyl)amine
3-[2-(5-ethyl-1,2,4-oxadiazol-3-yl)ethyl]-1-{3-[(2-methylpiperidin-1-yl)methyl]phenyl}urea
3-{1-[4-(pyridin-2-yl)butyl]-1H-imidazol-2-yl}phenol
1-{1-[(4-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-4-[(2-methylphenyl)methyl]piperazine
N-(1H-imidazol-2-ylmethyl)-N-methyl-3-azaspiro[5.5]undecan-9-amine
2-[(dimethyl-1,2-oxazol-4-yl)methyl]-8-(3-hydroxypyridine-2-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
N,5-dimethyl-1-propyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-1H-pyrazole-4-carboxamide
4-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-3-one
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-hydroxybenzamide
(2S,4R)-4-amino-N-ethyl-1-{[6-(4-methylphenyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}pyrrolidine-2-carboxamide
N-(1-{7-[4-(4-methoxyphenyl)-4-oxobutanoyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-2-methylpropyl)furan-3-carboxamide
N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-3-hydroxypropanamide
N-methyl-5-[(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)methyl]furan-2-carboxamide
10-(6-hydroxy-1,4-oxazepane-4-carbonyl)-9-methoxy-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-7-one
2-[4-(1-benzofuran-2-ylmethyl)-1-(3-methylbut-2-en-1-yl)piperazin-2-yl]ethan-1-ol
1-[4-(2-fluorophenyl)pyrimidin-2-yl]-5-(propan-2-yl)-N-[2-(pyridin-4-yl)ethyl]-1H-pyrazole-4-carboxamide
2-[(6-methyl-1H-1,3-benzodiazol-2-yl)methoxy]-N-(thiophen-3-ylmethyl)acetamide