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4-[2-methyl-3-(1H-pyrrol-1-yl)phenyl]-4H-1,2,4-triazole
2-methoxy-3-[4-(pyridin-3-ylmethoxy)piperidin-1-yl]pyrazine
3-[(3R,4S)-1-{[2-(cyclopentylmethyl)-1H-imidazol-4-yl]methyl}-4-(dimethylamino)piperidin-3-yl]propanoic acid
N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}-5-methyl-1,3-oxazole-4-carboxamide
N-cyclopropyl-1-[1-(3-phenoxypropanoyl)piperidin-4-yl]piperidine-4-carboxamide
1-(6-cyanopyridine-3-carbonyl)-4-(4-methyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
N-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-1,3-dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
6-({4-[2-(methoxymethyl)-5-(trifluoromethyl)-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}methyl)quinoline
5-benzyl-3-(oxan-4-yl)-5-(piperidin-4-yl)imidazolidine-2,4-dione
2-[(7-chloro-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)methyl]phenol
5-[4-(2-ethoxyphenyl)piperazine-1-carbonyl]-N-(2-methylpropyl)-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3-carboxamide
4-[3-(2-hydroxyethyl)-4-(2-methylpropyl)piperazin-1-yl]-N-(propan-2-yl)pyridine-2-carboxamide
propyl (1R,5S,6R)-6-{[4-(furan-2-carbonyl)piperazin-1-yl]methyl}-3-azabicyclo[3.1.0]hexane-3-carboxylate
N-(cyclohexylmethyl)-2,7-diazaspiro[4.5]decane-7-carboxamide
3-methyl-7-{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
1-(cyclohexylmethyl)-N,N-dimethyl-5-{[2-(morpholin-4-yl)ethyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
6-(6-cyclopropylpyrimidin-4-yl)-N-methyl-4-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-2-amine
4-[4-(4-methylphenyl)-3-oxopiperazine-1-carbonyl]benzonitrile
1-(4-hydroxypiperidin-1-yl)-4-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butan-1-one
4-benzyl-1-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-3-ethyl-1,4-diazepan-5-one
8-{[3-(furan-2-yl)phenyl]methyl}-1-[2-(4-methoxyphenyl)ethyl]-3-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-{2,3-dimethyl-5-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carbonyl}-1-phenylpiperazin-2-one
2-cyclopentyl-N-[1-(1,3-thiazol-2-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
2-(5-chloro-2-methoxyphenyl)-2-[4-(1-methylpiperidin-4-yl)piperazin-1-yl]acetic acid
4-[(1r,4r)-4-methylcyclohexanecarbonyl]-1,8-dioxa-4,11-diazaspiro[5.6]dodecane
5-(2-{[2-(4-fluorophenoxy)ethyl]amino}ethyl)-1-[(5-phenyl-1,2-oxazol-3-yl)methyl]pyrrolidin-2-one
N-cyclopropyl-2-{2-ethyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}acetamide
N-(2,1,3-benzoxadiazol-4-ylmethyl)-1-(3,4-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
N-{[2-(2-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}-4-(1H-1,2,4-triazol-1-yl)butanamide
4-(5-{[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonyl)morpholine
N4-[1-(3,4-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]pyrimidine-4,6-diamine
3-[5-(5-methyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanoic acid
3-(1H-1,2,3-benzotriazol-1-yl)-N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]propanamide
2-(2-methoxyethyl)-8-[2-(1-methyl-1H-indol-3-yl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
2-fluoro-6-methoxy-4-{[4-(1-methoxypropan-2-yl)piperidin-1-yl]methyl}phenol
1-(3-chlorophenyl)-4-{1-[(2,6-dimethoxyphenyl)methyl]piperidin-3-yl}piperazine
6-methyl-N-[2-(piperidin-1-yl)-2-(pyridin-3-yl)ethyl]imidazo[2,1-b][1,3]thiazole-5-carboxamide
N-{[2-(dimethylamino)pyridin-3-yl]methyl}-4-methyl-1,3-oxazole-5-carboxamide
N-[(5-methyl-1H-imidazol-4-yl)methyl]-3-(3-methylpiperidine-1-carbonyl)benzene-1-sulfonamide
6-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}pyrazine-2-carboxamide
4-(4-benzyl-1H-pyrazol-5-yl)-1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidine
3-{4-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperazin-1-yl}-2,5-dimethylpyrazine
4-(1-methyl-1H-pyrazol-4-yl)-N-[2-(3-phenylpiperidin-1-yl)ethyl]pyrimidin-2-amine
methyl (2S,4R)-1-[(4-hydroxyphenyl)methyl]-4-{2-[4-(trifluoromethyl)phenyl]benzamido}pyrrolidine-2-carboxylate
N-(1-cyclobutanecarbonylazepan-3-yl)-2-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]acetamide
3-(5-{3-methyl-3H-[1,2,3]triazolo[4,5-b]pyridine-6-carbonyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)propanoic acid
1-ethyl-4-[3-(3-hydroxy-3-methylbutyl)benzoyl]piperazin-2-one
4-{[3-(3-methoxyphenyl)-1,2-oxazol-5-yl]methyl}-1-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}piperidin-4-ol
1-{[3-(difluoromethoxy)phenyl]methyl}-4-ethyl-3-(piperidin-4-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
3-(3-chlorobenzoyl)-1-(4-methanesulfonylbenzenesulfonyl)piperidine