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2-(3,6-dioxo-1,2,3,6-tetrahydropyridazin-1-yl)-N-methyl-N-{[2-(2-methylpropoxy)phenyl]methyl}acetamide
7-methyl-2-[3-(pyridin-4-yl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one
N-[1-(3-methylbutan-2-yl)-1H-pyrazol-5-yl]-1-(pyrimidin-2-yl)piperidine-4-carboxamide
3-(3-chlorophenyl)-1-(pyridin-3-ylmethyl)-6-(pyridine-2-carbonyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
1-(3-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-sulfonyl}-4-methoxyphenyl)-1H-pyrazole
3-(2-oxo-2-{4-[2-(phenoxymethyl)-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}ethyl)-2,3-dihydro-1H-isoindol-1-one
2-[4-(pyrimidin-5-yl)phenyl]pyrimidin-5-ol
(2S)-1-{[2-(ethanesulfonyl)-1-(3-phenylpropyl)-1H-imidazol-5-yl]methyl}pyrrolidine-2-carboxamide
5-(1-{[4-(1H-imidazol-1-yl)phenyl]methyl}pyrrolidin-2-yl)-3-methyl-1,2-oxazole
1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-1-yl]-2-(2-methyl-1H-imidazol-1-yl)ethan-1-one
N-{[4-amino-6-(dimethylamino)-1,3,5-triazin-2-yl]methyl}-2-oxo-1,2-dihydroquinoline-4-carboxamide
N-({7-methylimidazo[1,2-a]pyridin-2-yl}methyl)-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
3-(2-amino-1,3-thiazol-4-yl)-N-[3-(1H-indol-1-yl)propyl]propanamide
N-cyclopropyl-N-({4-[(4-fluorophenyl)methoxy]-3-methoxyphenyl}methyl)-2-(trifluoromethyl)benzamide
2-{[(6-methylpyridin-2-yl)methyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
5-({[(3-{2-[4-(2,5-dimethoxybenzenesulfonyl)piperazin-1-yl]ethoxy}phenyl)methyl](methyl)amino}methyl)pyrrolidin-2-one
3-[(2H-1,3-benzodioxol-5-ylmethyl)amino]-N-(1-phenylethyl)propanamide
3-chloro-N-methyl-N-[(5-methyl-1H-1,3-benzodiazol-2-yl)methyl]thiophene-2-carboxamide
(furan-2-ylmethyl)({[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl})(pyridin-2-ylmethyl)amine
2-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-3,7-dimethyl-1H-indole
N-cyclohexyl-5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridin-2-amine
1-{2-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-5-methoxybenzoyl}-4-(methoxymethyl)piperidine
3-(2-amino-1,3-thiazol-4-yl)-1-[3-(2H-1,3-benzodioxol-5-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]propan-1-one
2-[2-({1,9-dimethyl-10-oxo-1,4,9-triazaspiro[5.6]dodecan-4-yl}methyl)phenoxy]acetic acid
2-(cyclopentylmethyl)-7-[(3,4-difluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
4-{[5-(oxolan-2-yl)thiophen-2-yl]methyl}thiomorpholine
N-[(5-{[2-(dimethylamino)ethyl]sulfanyl}-4-(3-methoxyphenyl)-4H-1,2,4-triazol-3-yl)methyl]pent-4-enamide
N-[2-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)ethyl]pyridine-4-carboxamide
1-cyclopropyl-3-(2,3-dihydro-1H-inden-4-yl)-1-[(4-hydroxy-3-methoxyphenyl)methyl]urea
4-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}pyrimidin-2-amine
N-ethyl-5-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-N-(oxolan-2-ylmethyl)-1,2-oxazole-3-carboxamide
9-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]-6-oxa-9-azaspiro[4.5]decane
N,1,3-trimethyl-N-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
1-{1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-4-yl}-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
5-cyclopropanecarbonyl-1'-[(5-fluoro-2-methoxyphenyl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
(2R,6R)-6-methyl-1-(3-methylfuran-2-carbonyl)-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine
N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}-2-(2-ethyl-1H-imidazol-1-yl)acetamide
5-(2-benzyl-1,3-thiazol-4-yl)-3-(2-methoxyethyl)-1,2,4-oxadiazole
2-(3-hydroxypropyl)-8-(3-methoxybenzoyl)-2,8-diazaspiro[5.5]undecan-3-one
N-methyl-N-({4-oxo-3H,4H-thieno[3,2-d]pyrimidin-2-yl}methyl)imidazo[2,1-b][1,3]thiazole-6-carboxamide
(4aS,8aR)-6-[(5-methylfuran-2-yl)methyl]-1-[2-(pyridin-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
N,N-diethyl-2-({1-[(4-methoxyphenyl)methyl]-2-oxo-4-[4-(piperidin-1-ylmethyl)benzoyl]-1,4-diazepan-6-yl}oxy)acetamide
(1S,6R)-9-{3-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]propanoyl}-3,9-diazabicyclo[4.2.1]nonan-4-one
6-{methyl[(3-methylphenyl)methyl]amino}-1-(pent-4-en-1-yl)-1H,4H,5H,8H-imidazo[4,5-e][1,3]diazepine-4,8-dione
N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carboxamide
2-{2-[(4-ethyl-3,3-dimethylpiperazin-1-yl)methyl]-6-methoxyphenoxy}propanoic acid
3-[(cyclopropylmethyl)amino]-N-[(3S)-2-oxoazepan-3-yl]-5-[(propan-2-yl)sulfamoyl]benzamide
5-[4-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidine-1-carbonyl]pyridine-2-carbonitrile
3-(1-ethyl-1H-imidazol-2-yl)-1-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]piperidine
4-methyl-N-[(5-methylpyrazin-2-yl)methyl]-2-(propan-2-yl)-1,3-thiazole-5-carboxamide