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8-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-1-(2-methoxyethyl)-3-[(3-methoxyphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-ethyl-3-fluoro-2-methoxy-N-[(5-propyl-1,2,4-oxadiazol-3-yl)methyl]benzamide
N-(2-{7-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)furan-3-carboxamide
3-fluoro-2-{4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine
1-(2-methylphenyl)-4-[5-(1H-pyrazol-1-ylmethyl)furan-2-carbonyl]-1,4-diazepane
1-(1-{[4-hydroxy-3-(prop-2-en-1-yl)phenyl]methyl}piperidin-4-yl)pyrrolidin-2-one
(3R)-1-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-3,4,4-trimethylpyrrolidin-3-ol
4-(4-methylpiperazin-1-yl)-N-(2-methylpropyl)-N-(thiophen-3-ylmethyl)pentanamide
N3-[3-(benzylsulfanyl)propyl]-N1,N1-dimethylpiperidine-1,3-dicarboxamide
methyl 4-[2-(5-hydroxy-2-methoxyphenyl)-1H-imidazol-1-yl]benzoate
1-[6-(4-{[4-(1H-imidazol-1-yl)phenyl]methyl}piperazin-1-yl)pyridin-3-yl]ethan-1-one
N-(adamantan-2-yl)-6-{[benzyl(methyl)amino]methyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-2,3-dihydro-1-benzofuran-5-carboxamide
N-[3-(1H-indol-1-yl)propyl]-4-(pyridin-4-yl)pyrimidin-2-amine
N-[1-({2,4-dimethyl-5-[(4-methylpiperazin-1-yl)methyl]phenyl}methyl)piperidin-3-yl]acetamide
N-[(4-hydroxyazepan-4-yl)methyl]-1-methyl-4-phenylpiperidine-4-carboxamide
4-methoxy-6-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidine
1-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}-3-[4-(trifluoromethyl)benzoyl]piperidine
5-{3-[(4-methoxyphenyl)methyl]-1,2,4-oxadiazol-5-yl}-2-(4-methoxypiperidin-1-yl)pyridine
1-(2-{[cyclohexyl(methyl)amino]methyl}phenyl)-3-[(3S,4S)-4-methoxy-1-methylpyrrolidin-3-yl]urea
N-[(4-methoxyphenyl)methyl]-N-(oxolan-2-ylmethyl)-1H-1,2,3-triazole-5-carboxamide
4-(2-methyl-1H-imidazol-1-yl)-1-[3-(methylcarbamoyl)pyridin-2-yl]piperidine-4-carboxylic acid
3-({3-[4-(2,6-difluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)phenol
N-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]acetamide
1-(5-{1-methyl-1H-pyrazolo[1,5-a]imidazole-7-carbonyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carbonyl)pyrrolidine
2-{4-[hydroxy(1-methyl-1H-imidazol-2-yl)methyl]piperidine-1-carbonyl}pyridin-3-ol
1-{1-[(2,3-dimethoxyphenyl)methyl]piperidin-4-yl}-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
1-{4-[(2-methylphenyl)sulfanyl]piperidin-1-yl}-2-(morpholin-4-yl)ethan-1-one
4-[phenyl({1-[(3-phenyl-1H-1,2,4-triazol-5-yl)methyl]-1H-1,2,3,4-tetrazol-5-yl})methyl]morpholine
1,9-dimethyl-4-[(1-propyl-1H-imidazol-2-yl)methyl]-1,4,9-triazaspiro[5.5]undecane
1-[3-(azonan-1-ylmethyl)phenoxy]-3-(morpholin-4-yl)propan-2-ol
1-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-(2-ethyl-1H-imidazol-1-yl)ethan-1-one
3-methyl-3-{[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]methyl}-1-(4-oxo-4H-chromen-6-yl)urea
N-(1-{1-[(2-chlorophenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-methoxybenzamide
3-(aminomethyl)-4-(2H-1,3-benzodioxol-5-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-2-(3-methyl-1,2-oxazol-5-yl)acetamide
5-(2,6-dimethoxyphenyl)-2,3-dimethylpyrazine
3-{[1-(1-ethyl-3,5-dimethyl-1H-pyrazole-4-carbonyl)pyrrolidin-3-yl]methyl}benzoic acid
5-[3-(2-chlorophenoxy)azetidine-1-carbonyl]-2,2-dimethylthiomorpholin-3-one
3-hydroxy-3-{[4-(6-methylpyridin-2-yl)piperazin-1-yl]methyl}-1-(2-phenylethyl)piperidin-2-one
2-{[3-(2,4-dimethoxybenzoyl)piperidin-1-yl]methyl}pyridine
1-[3-(4-phenylbenzoyl)piperidin-1-yl]-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
N-(carbamoylmethyl)-2-{1-[(3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}acetamide
[(dimethyl-1,2-oxazol-4-yl)methyl][(4-methanesulfonylphenyl)methyl]methylamine
(3S)-1-ethyl-4-{[2-(furan-3-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-methylpiperazin-2-one
2-chloro-N-[2-({2-methyl-2,8-diazaspiro[4.5]decan-3-yl}formamido)ethyl]benzamide
2-(4-{[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]amino}-6-methylpyrimidin-2-yl)phenol
[3-(3-methylbut-2-en-1-yl)-1-(pyridazine-3-carbonyl)piperidin-3-yl]methanol
2-[2-({[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl](methyl)amino}methyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl]pyrimidin-4-amine
4-ethyl-1-[(2-phenyl-1,3-thiazol-4-yl)methyl]-3-(piperidin-4-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one