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N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-5-methyl-2-{[1-(pyridin-4-ylmethyl)piperidin-4-yl]oxy}benzamide
2-(2-{[2-(6-hydroxy-2-methylpyrimidin-4-yl)ethyl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
methyl 4-[5-methyl-4-({2-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}methyl)-1,3-oxazol-2-yl]benzoate
(2R,6R)-4-[2-(5-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)acetyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
2-[1-({1-[1-(2-fluorophenyl)propan-2-yl]piperidin-4-yl}methyl)-1H-1,2,3-triazol-4-yl]propan-2-amine
(3S)-1-{[2-(4-chlorophenyl)-5,8-dimethoxyquinolin-3-yl]methyl}pyrrolidin-3-ol
(1,4-dioxan-2-ylmethyl)[(4-methanesulfonylphenyl)methyl]methylamine
N-{2H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-2-(dimethylamino)-2-(3-fluorophenyl)-N-methylacetamide
2-(2,5-dioxoimidazolidin-1-yl)-N-(2-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-4-yl)acetamide
4-(4-chlorophenoxy)-N-[1-(1H-pyrazol-1-yl)propan-2-yl]piperidine-4-carboxamide
N-[(1-benzylpyrrolidin-3-yl)methyl]-5-methyl-4-(1-methyl-1H-pyrazol-4-yl)pyrimidin-2-amine
N-cyclopropyl-N-({3-[(2-fluorophenyl)methoxy]phenyl}methyl)-5-methylthiophene-2-carboxamide
5-methanesulfonyl-2-methyl-N-(pyridin-4-ylmethyl)pyrimidin-4-amine
(3R,5R)-N-{2-[4-(dimethylamino)phenyl]ethyl}-5-(pyrrolidine-1-carbonyl)piperidine-3-carboxamide
3-(2,3-dihydro-1,4-benzodioxin-6-ylsulfanyl)-1-[(3S,4S)-3,4-dihydroxypiperidin-1-yl]propan-1-one
8-(2,5-difluorobenzoyl)-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
(1R,3S)-7-[3-(dimethylamino)benzoyl]-3-[2-(dimethylamino)ethoxy]-7-azaspiro[3.5]nonan-1-ol
1-{5-[(cycloheptylamino)methyl]-2-methoxyphenoxy}-3-[methyl(propan-2-yl)amino]propan-2-ol
6-methyl-2-{[5-(2-methylprop-1-en-1-yl)-4-phenyl-1H-imidazol-1-yl]methyl}-3,4-dihydropyrimidin-4-one
N-[(7S,8aS)-2-methyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-2,1-benzoxazole-3-carboxamide
4-[(2-chlorophenyl)methyl]-1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-1,4-diazepan-5-one
4-[5-(pyridin-3-yl)furan-2-carbonyl]morpholine
2-(4-{[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}morpholin-3-yl)acetic acid
[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl][(6-chloropyridin-3-yl)methyl]amine
3,5-dimethyl-1-(1-{2-methylthieno[2,3-d]pyrimidin-4-yl}pyrrolidin-3-yl)-1H-pyrazole
N-(2-methyl-2,3-dihydro-1-benzofuran-5-yl)-2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carboxamide
N-[(3S,5S,9S)-2,8-dioxo-1,7-diazatricyclo[7.3.0.03,7]dodecan-5-yl]benzamide
3-{5-[(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocin-5-yl)methyl]thiophen-3-yl}prop-2-yn-1-ol
N-[2-(3-carbamoylpiperidin-1-yl)ethyl]-6-chloro-1-methyl-1H-indole-2-carboxamide
(4aR,8aR)-2-{[2-(ethylamino)pyrimidin-5-yl]methyl}-7-methanesulfonyl-decahydro-2,7-naphthyridin-4a-ol
1-[(3S)-3-ethylmorpholin-4-yl]-2-(4-phenylpiperidin-1-yl)ethan-1-one
3-(4-chlorophenyl)-5-(oxolane-2-carbonyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
[1-(4-methyl-1,2,5-oxadiazole-3-carbonyl)-3-(3-methylbut-2-en-1-yl)piperidin-3-yl]methanol
methyl 1-(cyclopropylmethyl)-3-[(4-methyl-1,3-thiazol-5-yl)methyl]-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxylate
(2S,4R)-N-ethyl-4-[2-(3-fluorophenyl)acetamido]-1-(1H-imidazol-2-ylmethyl)pyrrolidine-2-carboxamide
1-(4-benzyl-6-hydroxy-1,4-diazepan-1-yl)-3-methyl-3-phenylbutan-1-one
1-[2-(pyridin-2-yl)-4-{[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]amino}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
[1-(dimethyl-1,3-thiazol-4-yl)ethyl][(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]methylamine
4-{4-[1-ethyl-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazol-5-yl]benzoyl}morpholine
1-{4-[4-(dimethylamino)-5-methylpyrimidin-2-yl]piperazin-1-yl}-3-methylbutan-1-one
4-{2-methyl-4-oxo-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-1-(pyridin-2-ylmethyl)pyrrolidin-2-one
(3S,9aR)-3-benzyl-8-[(2,4-dimethylphenyl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-[3-(4-chlorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
8-(1-methoxypropan-2-yl)-1-(3-methoxypropyl)-3-(naphthalen-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidine-1-carbonyl)-1,2-dihydropyridin-2-one
2-[(2,2-dimethylpropyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
5-[6-(pyrrolidine-1-carbonyl)pyrazin-2-yl]pyridin-3-amine
(3aS,6aS)-2-[(4-acetyl-1-methyl-1H-pyrrol-2-yl)methyl]-5-[3-(methylsulfanyl)propyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-(ethanesulfonyl)-3-(4-methoxy-2-methylbenzoyl)piperidine
4-[3-(cyclopropylmethyl)-3-(hydroxymethyl)piperidine-1-carbonyl]-N,N-dimethylpiperidine-1-carboxamide