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(3S,4R)-N,N-dimethyl-1-[2-methyl-5-(2-methyl-1,3-oxazol-5-yl)benzenesulfonyl]-4-(propan-2-yl)pyrrolidin-3-amine
3-{[3-(5-methyl-2H-1,2,3,4-tetrazol-2-yl)adamantan-1-yl]amino}-N-(2-methylphenyl)propanamide
1-[3-chloro-4-(1H-imidazol-1-yl)phenyl]-3-[(3R,4R)-4-(pyrrolidin-1-yl)oxolan-3-yl]urea
1-[3-(hydroxymethyl)-3-(2-methoxyethyl)piperidin-1-yl]-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
(3S,4S)-1-(4-methoxycyclohexanecarbonyl)-4-(naphthalen-2-yl)piperidin-3-ol
N3-{2-[4-(pyrimidin-2-yl)piperazin-1-yl]ethyl}piperidine-1,3-dicarboxamide
3-(2-amino-1,3-thiazol-4-yl)-1-[(3R,4S)-4-hydroxy-3,4-dimethylpiperidin-1-yl]propan-1-one
N,1-dimethyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-3-propyl-1H-pyrazole-5-carboxamide
3-benzyl-4-[(3-methylphenyl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
2-{1'-[(3-methylthiophen-2-yl)methyl]-2-oxo-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-1-yl}acetamide
6-(2,5-dimethoxyphenyl)-N-(1,4-dioxan-2-ylmethyl)-N-methyl-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridine-3-carboxamide
6-(2,5-dimethylfuran-3-yl)-N-(1H-imidazol-2-ylmethyl)-N,7-dimethyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
2-methoxy-N-[(3R,4S)-1-[3-(methylsulfanyl)propyl]-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
3-{[(5-methylthiophen-2-yl)methyl]({[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl})amino}propan-1-ol
2-(4-tert-butylphenoxymethyl)-4-hydroxy-N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]pyrimidine-5-carboxamide
1-(2-chloroprop-2-en-1-yl)-6,7-dimethoxy-3-({[3-(2-oxopyrrolidin-1-yl)propyl]amino}methyl)-1,2-dihydroquinolin-2-one
3-{imidazo[1,2-a]pyridin-2-yl}-1-[3-(2-methoxyphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]propan-1-one
6-[1-(morpholin-4-yl)cyclohexanecarbonyl]-N-[3-(pyridin-4-yl)propyl]-6-azaspiro[2.5]octane-1-carboxamide
(3S,4R)-1-(2,5-difluorobenzoyl)-4-(2-methoxyphenyl)pyrrolidine-3-carboxylic acid
2-[2-(furan-2-yl)pyrimidin-4-yl]pyridine-4-carboxylic acid
4-(6-methylpyridine-2-carbonyl)-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-(3-hydroxy-3-methylbutyl)-N-methyl-N-{[1-(propan-2-yl)piperidin-3-yl]methyl}benzamide
4-({6-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}methyl)-2-methyl-1H-imidazole
1-cyclopropanecarbonyl-4-(3-fluorophenoxy)piperidine-4-carboxylic acid
(2S,4S)-4-amino-N-methyl-1-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}pyrrolidine-2-carboxamide
3-(3-chloro-1H-1,2,4-triazol-5-yl)-N-[1-methyl-4-(pyridin-3-yloxy)-1H-indazol-3-yl]propanamide
8-methoxy-5-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}-2-[3-(trifluoromethyl)phenyl]-2,3,4,5-tetrahydro-1,5-benzothiazepine
1-(4-fluorophenyl)-N-{[2-(trifluoromethyl)phenyl]methyl}cyclopropane-1-carboxamide
2-[2-(6-methoxypyridin-3-yl)phenoxy]propanamide
3-[2-(4-chlorophenyl)morpholine-4-carbonyl]-1-ethyl-6-methyl-1,2-dihydropyridin-2-one
N-(1-{1-[5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]piperidin-4-yl}-1H-pyrazol-5-yl)acetamide
ethyl({[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl})(1,3-thiazol-2-ylmethyl)amine
6-methyl-3-[(1S,5R)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1,2-dihydropyridin-2-one
1-ethyl-N-methyl-N-(2-phenylethyl)-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
9-(5-ethyl-2-methylpyrimidin-4-yl)-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-(1-benzothiophen-3-yl)pyridine-3-carboxamide
1-({5-[1-(2,2-dimethylpropyl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)piperidin-4-ol
N,N-dimethyl-4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-sulfonamide
{3-ethyl-1-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]piperidin-3-yl}methanol
2,3,5-trimethyl-N-[1-(3,4,5-trimethoxyphenyl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
N-[(3S,4R)-1-(2-ethoxypyridine-3-carbonyl)-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
N-butyl-7-{[2-(methoxymethyl)pyrrolidin-1-yl]sulfonyl}-1,2,3,4-tetrahydroisoquinoline-2-carboxamide
2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]-1-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]ethan-1-one
2-(2-methyl-1,3-thiazol-4-yl)-1-{4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}ethan-1-one
N-[(3,4-difluorophenyl)methyl]-N-[(1-methyl-1H-pyrazol-4-yl)methyl]cyclopropanamine
3-(propan-2-yl)-1-[(1-{[2-(propan-2-yl)pyrimidin-4-yl]methyl}piperidin-3-yl)methyl]urea
6-[(3R,4S)-3-amino-4-propylpyrrolidin-1-yl]-N-ethyl-N-methylpyridine-3-carboxamide
4-(4-methyl-1H-pyrazol-1-yl)-1-[4-(methylcarbamoyl)pyridin-2-yl]piperidine-4-carboxylic acid
1-[(3-chlorophenyl)methyl]-4-[2-(oxolan-2-yl)-3H-imidazo[4,5-b]pyridin-3-yl]piperidine
3-(2-ethylphenoxy)-1-(4-methoxybenzoyl)azetidine