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N-[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]-3-(4H-1,2,4-triazol-4-yl)benzamide
N-[2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)ethyl]-N-methyl-3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carboxamide
5-(4,4-difluoropiperidine-1-carbonyl)-2-(2-methyl-1,3-thiazol-4-yl)pyrimidin-4-ol
4-[(8-methoxyquinolin-2-yl)methyl]-1λ6-thiomorpholine-1,1-dione
4-methoxy-N-(1-{1-[(2E)-2-methylbut-2-en-1-yl]piperidin-4-yl}-1H-pyrazol-5-yl)benzamide
2-(4,7-dimethyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-methyl-N-{[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
5-[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methoxy]-4,6-dimethyl-2-(propan-2-yl)pyrimidine
1-[1-(4-methoxyphenyl)-5-phenyl-1H-pyrazole-3-carbonyl]piperidin-4-ol
1-[2-amino-6-(methylamino)pyrimidin-4-yl]-4-(1H-imidazol-1-yl)piperidine-4-carboxylic acid
2-methoxy-4-{[4-(4,6,7-trimethylquinazolin-2-yl)-1,4-diazepan-1-yl]methyl}phenol
3-(2-ethyl-1H-imidazol-1-yl)-N-{1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl}propanamide
2-[5-(azepan-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-[3-(1H-indol-1-yl)propyl]acetamide
3-[2-(3,5-dimethylpiperidin-1-yl)ethyl]-8-(trifluoromethyl)-3,4-dihydroquinazolin-4-one
N-methyl-N-{2-[(4-methylphenyl)sulfanyl]ethyl}-2-[6-oxo-4-(pyrrolidin-1-yl)-1,6-dihydropyridazin-1-yl]acetamide
4-(1-{1-[4-(2-fluorophenyl)benzoyl]piperidin-4-yl}-1H-1,2,3-triazole-4-carbonyl)morpholine
4-[5-(2-methoxyphenoxymethyl)-1H-pyrazole-3-carbonyl]-1-phenylpiperazin-2-one
N-(isoquinolin-5-ylmethyl)-N,2-dimethyl-1H-1,3-benzodiazole-5-carboxamide
2-{3-cyclopropyl-5-[6-(3-fluorophenyl)pyridin-3-yl]-1H-1,2,4-triazol-1-yl}acetic acid
3-methyl-7-{[2-methyl-4-(1H-pyrazol-1-yl)phenyl]methyl}-1-oxa-3,7-diazaspiro[4.5]decan-2-one
1-(4-{6-hydroxy-4-[(3-methylpyrazin-2-yl)methyl]-1,4-diazepan-1-yl}piperidin-1-yl)ethan-1-one
2-(7-fluoro-2-methyl-1H-indol-3-yl)-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]acetamide
N,1-dimethyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]piperidine-2-carboxamide
2-[2-(2-fluorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-1-[4-(4-methyl-1,2,5-oxadiazol-3-yl)piperazin-1-yl]ethan-1-one
5-(2-fluorophenoxymethyl)-N-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}-1H-pyrazole-3-carboxamide
1-{3-[4-(furan-2-ylmethyl)piperazine-1-carbonyl]piperidin-1-yl}-2-methoxyethan-1-one
5-methyl-N-[3-(1H-1,2,4-triazol-1-yl)propyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
N-cyclobutyl-3-[methyl(oxolan-3-ylmethyl)sulfamoyl]benzamide
N,N-dimethyl-2-{[2-(2-methyl-1,3-thiazol-4-yl)acetamido]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
5-[benzyl(methyl)amino]-2-[(4-methyl-1,3-thiazol-5-yl)methyl]-2,3-dihydropyridazin-3-one
4-[(dimethyl-1,2-oxazol-4-yl)methyl]-1-methyl-2,3,4,5-tetrahydro-1H-1,4-benzodiazepine-2,5-dione
(1R,3S)-1,3-dihydroxy-N-(2-phenoxyphenyl)-7-azaspiro[3.5]nonane-7-carboxamide
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carbonyl]piperidin-3-amine
N-[(1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}piperidin-3-yl)methyl]acetamide
(1-{[2-(trifluoromethyl)phenyl]methyl}-4-{[3-(trifluoromethyl)phenyl]methyl}piperidin-4-yl)methanol
2-[2-(3,4-dichlorophenyl)morpholin-4-yl]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
2-{[(3,5-dimethyladamantan-1-yl)oxy]methyl}-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
5-methyl-1-phenyl-4-[2-(4H-1,2,4-triazol-4-yl)pyridine-4-carbonyl]piperazin-2-one
{1-[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-3-(prop-2-en-1-yl)piperidin-3-yl}methanol
1-[(4-fluorophenyl)methyl]-N-methyl-N-[(5-propyl-1H-pyrazol-3-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
1-(2-methoxyethyl)-3-methyl-8-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-{1-[5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]piperidin-4-yl}acetamide
3-[2-(methylsulfanyl)benzoyl]-1-[(5-methylthiophen-2-yl)methyl]piperidine
1-(dimethyl-1,3-oxazole-5-carbonyl)-N,N-diethylpyrrolidin-3-amine
1-(3-hydroxy-2,2-dimethylpropyl)-4-{[3-(3-methoxyphenyl)-1,2-oxazol-5-yl]methyl}piperidin-4-ol
3-(3-cyclopropyl-1H-pyrazol-5-yl)-4-[(4-methoxyphenyl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
2-[ethyl({[(3R,4R)-4-(hydroxymethyl)-1-[2-(methylamino)pyrimidine-5-carbonyl]pyrrolidin-3-yl]methyl})amino]ethan-1-ol
(2S,4S)-4-amino-1-(2,5-difluorobenzoyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
methyl 3-[(2R,3S,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]propanoate
2-({[(4-chlorophenyl)methyl]amino}methyl)-4-(pyridin-3-yl)phenol
6-{3-[3-(2,5-difluorobenzoyl)piperidin-1-yl]-3-oxopropyl}-2,3,4,5-tetrahydropyridazin-3-one