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N-[(3S,4R)-1-(3-cyano-5-fluorobenzoyl)-4-propylpyrrolidin-3-yl]methanesulfonamide
7-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-2-(pyridin-2-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-({[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}amino)propan-1-ol
4-benzyl-3-(piperidin-4-yl)-1-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
1'-[3-(3-hydroxy-1,2-oxazol-5-yl)propanoyl]-1-methyl-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
4-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]-4H-1,2,4-triazole
2-methyl-1-[2-(pyridin-3-yl)acetyl]-1,4-diazepan-5-one
methyl 3-benzamido-5-{[2-(1,3-thiazol-4-yl)acetamido]methyl}benzoate
N-[4-(1H-1,3-benzodiazol-2-yl)phenyl]-1-(2-oxopropanoyl)piperidine-4-carboxamide
3-(4,5-dimethyl-1H-1,3-benzodiazol-2-yl)-1-[4-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]propan-1-one
N-[2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-[(2-methoxyphenyl)methyl]-1-methyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-[3-(5-cyclopropyl-1H-pyrazol-1-yl)propyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
(3R,4R)-4-(2-methoxyethyl)-3-methyl-1-{[3-(trifluoromethyl)phenyl]methyl}piperidin-4-ol
5-[4-(6-hydroxypyrimidin-4-yl)piperidine-1-carbonyl]-1-(2-methylpropyl)piperidin-2-one
5,7-dimethyl-N-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl}pyrido[2,3-d]pyrimidin-4-amine
N,5-dimethyl-N-(1-methylpiperidin-4-yl)-1-{5H-thiochromeno[4,3-d]pyrimidin-2-yl}-1H-pyrazole-4-carboxamide
1-methyl-6-[4-(1H-pyrazol-1-yl)benzoyl]-3-[4-(trifluoromethoxy)phenyl]-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
1-(3,5-dichloro-4-methylbenzoyl)-3-(methoxymethyl)pyrrolidine
2-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N-methylpyridine-3-carboxamide
2-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepane-1-carbonyl}pyridin-3-ol
3-(dimethylsulfamoyl)-5-{[(4-ethylphenyl)methyl]amino}-N-[3-(1H-imidazol-1-yl)propyl]benzamide
N,2-dimethyl-N-[1-(1,2-oxazol-3-yl)ethyl]-4-phenyl-1,3-thiazole-5-carboxamide
(3R,5S)-5-[(4-methylpiperazin-1-yl)methyl]-1-(2-methylpropyl)-N-(oxolan-2-ylmethyl)piperidine-3-carboxamide
N-(2-{7-[3-(5-methylfuran-2-yl)butyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)oxane-4-carboxamide
4-methyl-2-{4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}-6-(trifluoromethyl)pyrimidine
1-[4-(4-acetylphenyl)piperazin-1-yl]-2-methyl-3-(1H-pyrazol-1-yl)propan-1-one
(1S,5R)-6-(oxane-4-carbonyl)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-{[2-(dimethylamino)pyridin-3-yl]methyl}-3-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)propanamide
2-[4-(8-methylquinolin-5-yl)phenoxy]acetamide
5-(furan-3-ylmethyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
N-{2-[4-(4-fluorophenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]ethyl}-2,3,4-trimethoxybenzamide
4-[4-(2-ethoxyethyl)piperazine-1-carbonyl]-1-(pyridin-3-ylmethyl)pyrrolidin-2-one
N-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]pyrazolo[1,5-a]pyridine-7-carboxamide
1-{4-[6-ethyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]-6-hydroxy-1,4-diazepan-1-yl}ethan-1-one
2,6-dioxo-N-(2-{4-[(4-phenylpiperidin-1-yl)methyl]phenoxy}propyl)-1,2,3,6-tetrahydropyrimidine-4-carboxamide
4-[(3-methylphenyl)methyl]-3-(pyrazin-2-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
6-chloro-N,N-dimethyl-2-[1-(pyridin-2-yl)-1H-pyrazol-4-yl]quinoline-4-carboxamide
N-cyclopropyl-1-[2-(ethylamino)-4-methyl-1,3-thiazole-5-carbonyl]piperazine-2-carboxamide
5-[3-(4-chlorophenyl)-1-(2-hydroxyethyl)-1H-1,2,4-triazol-5-yl]-1-(2-methoxyethyl)piperidin-2-one
5-(3-benzyl-1H-1,2,4-triazol-5-yl)-1,2-dihydropyridin-2-one
5-chloro-N-(cyclopropylmethyl)-N-(2-methoxyethyl)-3-methyl-1H-indole-2-carboxamide
methyl 2-(azocane-1-sulfonyl)-6-(cyclohex-3-ene-1-carbonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-(2-methyl-1-{7-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}propyl)furan-3-carboxamide
(3S,4R)-1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-4-phenylpyrrolidine-3-carboxylic acid
N-[2-(dimethylamino)-1-phenylethyl]-N-methyl-2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carboxamide
2-[1-(2H-1,3-benzodioxol-5-yl)-3-methyl-1H-1,2,4-triazol-5-yl]pyrazine
N-cyclopropyl-1-{1-[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}piperidine-3-carboxamide
methyl 4-{5-methyl-4-[(3-oxo-4-phenylpiperazin-1-yl)methyl]-1,3-oxazol-2-yl}benzoate
7-(1,3-benzothiazol-2-yl)-4-[2-(2-hydroxyethoxy)ethyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol