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10-methoxy-5-[2-methyl-2-(morpholin-4-yl)propyl]-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
2-(1,3-dimethyl-1H-pyrazol-4-yl)-N,1-bis(propan-2-yl)-1H-1,3-benzodiazole-5-sulfonamide
ethyl 4-[(2-{5,6-dimethyl-4-oxo-3H,4H-thieno[2,3-d]pyrimidin-2-yl}ethyl)amino]piperidine-1-carboxylate
1-[1-(3,3-dimethylbutanoyl)piperidin-3-yl]-N-(2-methoxyethyl)-1H-1,2,3-triazole-4-carboxamide
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-1-(pyrrolidin-1-yl)cyclopentane-1-carboxamide
3-{1-[2-(dimethylamino)benzoyl]piperidin-3-yl}benzoic acid
4-[(5-chloro-2,3-dimethoxyphenyl)methyl]morpholine-2-carboxamide
5-cyclopropyl-N-[(3R,4S)-4-cyclopropyl-1-[3-(methylsulfanyl)propyl]pyrrolidin-3-yl]-1,2-oxazole-3-carboxamide
1-{2-[ethyl(methyl)amino]propanoyl}-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
3-({[(5-cyclopropyl-1H-pyrazol-3-yl)methyl](methyl)amino}methyl)-N-(1-methyl-1H-pyrazol-5-yl)benzamide
6-[(dimethylamino)methyl]-2-oxo-N-(quinolin-3-ylmethyl)-1,2-dihydropyridine-3-carboxamide
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-(pyridin-3-ylmethyl)acetamide
N-({1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]pyrrolidin-3-yl}methyl)methanesulfonamide
2-amino-7-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
6-({3-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-1-yl}methyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-[(2R,3R,6R)-5-(4-methyl-1,3-thiazole-5-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
1-cyclopentyl-4-[3-(2-methyl-1H-imidazol-1-yl)propyl]piperazine
N-[3-(5-cyclopropyl-1H-pyrazol-1-yl)propyl]-1H-pyrazole-4-carboxamide
(2S,5R)-1-{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2,5-dimethylpiperazine
4-[2-(butan-2-yloxy)-3-methoxyphenyl]-1-(oxan-4-yl)-1H-1,2,3-triazole
(3R,4R)-1-(1,3-benzothiazole-6-carbonyl)-3-cyclobutyl-4-methylpyrrolidin-3-ol
2,5-dioxo-6-[2-(phenylamino)ethyl]-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
N-[1-(1-{[5-methyl-2-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]oxolane-3-carboxamide
2-{[(5-{1-[(5-ethylpyridin-2-yl)methyl]piperidin-4-yl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl](methyl)amino}ethan-1-ol
2-ethyl-N-(4-fluoro-3-methylphenyl)pyrrolidine-1-carboxamide
6-(3-chlorophenyl)-N-methyl-7-(3-methylbut-2-en-1-yl)-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
1-{2,7-diazaspiro[4.5]decan-2-yl}-3-{[5-(pyridin-4-yl)-1,3,4-oxadiazol-2-yl]sulfanyl}propan-1-one
1-[4-(4,4-difluoropiperidine-1-carbonyl)phenyl]imidazolidine-2,4-dione
1-methyl-4-[3-(propan-2-yl)-1,2-oxazol-5-yl]-3-(pyridin-3-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
2-[4-(1,3-benzothiazol-2-ylmethyl)-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl]ethan-1-ol
5-chloro-N-[2-(morpholin-4-yl)-2-(pyridin-3-yl)ethyl]thiophene-2-carboxamide
{4-[(4-chlorophenyl)methyl]-1-(oxolane-2-carbonyl)piperidin-4-yl}methanol
3-(furan-2-yl)-2-{[4-(3-methylthiophen-2-yl)-1H-1,2,3-triazol-1-yl]methyl}propan-1-ol
5-[2-(ethylamino)ethyl]-1-[(4-phenyl-1,3-thiazol-2-yl)methyl]pyrrolidin-2-one
2-{[3-(carboxymethyl)morpholin-4-yl]methyl}benzoic acid
N-[(2,3-dimethyl-1H-indol-5-yl)methyl]-2-(1-oxo-2,3-dihydro-1H-isoindol-2-yl)butanamide
[(1,3-dimethylpyrrolidin-3-yl)methyl][(4-ethoxyphenyl)methyl]methylamine
3-[2-(6-hydroxy-2-methylpyrimidin-4-yl)ethyl]-1-(5,6,7,8-tetrahydronaphthalen-1-yl)urea
N-(2-hydroxyethyl)-1,4,6-trimethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
1-[2-(1H-imidazol-1-yl)-1-phenylethyl]-4-(3-methylthiophen-2-yl)-1H-1,2,3-triazole
3-cyclohexyl-N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-N-methyl-1H-pyrazole-4-carboxamide
N-(1-{[5-(2-chlorophenyl)furan-2-yl]methyl}piperidin-4-yl)methanesulfonamide
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N-methyl-2-(morpholin-3-yl)acetamide
1-[(5-cyano-1-methyl-1H-pyrrol-3-yl)methyl]-3-(2-methoxyethyl)piperidine-3-carboxylic acid
(4aR,8aS)-6-(2H-1,3-benzodioxole-5-carbonyl)-1-(2,2-diphenylethyl)-decahydro-1,6-naphthyridin-2-one
N-[(1-benzoylpiperidin-3-yl)methyl]-4-methoxybenzene-1-sulfonamide
5-[6-(pyrrolidin-1-yl)pyridazin-3-yl]-1H-indole
3-propoxy-1-{5-propylpyrazolo[1,5-a]pyrimidin-7-yl}piperidine
4-[(1S,5R)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]pyridin-2-amine
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-2,5-dimethylfuran-3-carboxamide