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4-hydroxy-2-methyl-N-(4-phenylbutyl)pyrimidine-5-carboxamide
1-{6-[4-(3,4-dichlorophenyl)piperazin-1-yl]pyridin-2-yl}ethan-1-ol
1-[3-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-3-(4-methyl-1H-pyrazol-1-yl)propan-1-one
1-(azepan-1-yl)-3-(7-chloro-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)propan-1-one
N-(pyridin-3-ylmethyl)-3-{[1-(thiolan-3-yl)piperidin-4-yl]oxy}benzamide
2-cyclopentyl-1-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
1-[3-(4-phenoxybenzoyl)piperidin-1-yl]-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
methyl 3-{[(3S,4R)-3-acetamido-4-(4-methylphenyl)pyrrolidin-1-yl]methyl}benzoate
4-{[1-(1-methyl-5-phenyl-1H-pyrrole-2-carbonyl)piperidin-4-yl]methyl}morpholine
N-(2-{imidazo[1,2-a]pyridin-3-yl}ethyl)-1-methyl-1H-pyrazolo[1,5-a]imidazole-7-carboxamide
3-{3-[(4-cyclopropyl-1H-1,2,3-triazol-1-yl)methyl]piperidine-1-carbonyl}-2-ethoxypyridine
methyl (2S)-1-[2-(4-{4-[(2-{imidazo[1,2-a]pyridin-2-yl}ethyl)amino]piperidin-1-yl}phenyl)acetyl]pyrrolidine-2-carboxylate
1-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]-2-(pyridin-3-yl)ethan-1-one
N-[(3-methyl-1-benzofuran-2-yl)methyl]-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
2-(2-ethyl-1H-imidazol-1-yl)-1-[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
N-cyclohexyl-4-(5-methyl-1-propyl-1H-pyrazole-4-amido)piperidine-1-carboxamide
3-(oxan-2-ylmethyl)-3H,4H-thieno[2,3-d]pyrimidin-4-one
2-[4-(2-methoxypyridin-3-yl)-2-methylphenoxy]acetamide
3-[1-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-6-methoxy-3,4-dihydroquinazolin-4-one
2-ethyl-8-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-2,8-diazaspiro[4.5]decan-3-one
(1S,5R)-3-(1-benzothiophene-2-sulfonyl)-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[(2R,3R)-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2,3-dimethyl-1H-indole-5-carboxamide
N-(3-methoxypropyl)-N-(1-methylpiperidin-4-yl)-2-(4H-1,2,4-triazol-4-yl)pyridine-4-carboxamide
2-{4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazin-1-yl}-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
2-(dimethylamino)-2-(2-fluorophenyl)-1-[4-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]ethan-1-one
N-(3-aminopropyl)-2-[methyl(2-phenylethyl)amino]-2,3-dihydro-1H-indene-2-carboxamide
N-(1-{5-[(cyclohexylmethyl)sulfanyl]-4-methyl-4H-1,2,4-triazol-3-yl}-2-phenylethyl)-3-(2-oxopyrrolidin-1-yl)benzamide
N-(oxolan-2-ylmethyl)-3-[1-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)piperidin-4-yl]propanamide
N-(2-acetamidophenyl)-2-[4-(3-methylphenoxy)piperidin-1-yl]acetamide
1-({4-[3-(morpholin-4-yl)propoxy]phenyl}methyl)azetidin-3-ol
1-{4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazin-1-yl}-2-(pyrazin-2-yl)ethan-1-one
1-[5-(4-phenylazepane-1-carbonyl)pyridin-2-yl]piperidin-4-amine
1-butyl-4-(4-cyclopropyl-1H-1,2,3-triazol-1-yl)piperidine
(3S,4R)-4-(hydroxymethyl)-1-[8-(trifluoromethyl)quinolin-4-yl]piperidin-3-ol
5-cyano-N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N,2-dimethyl-6-oxo-1,6-dihydropyridine-3-carboxamide
1-[1-(4-fluorophenyl)ethyl]-5-(1H-imidazol-4-yl)-4-phenyl-1H-imidazole
1-{2-[(4-cyclopentylpyrimidin-2-yl)amino]ethyl}piperidin-4-ol
4-(2-methylpyridin-4-yl)-N-(3-phenyl-1,2,4-thiadiazol-5-yl)piperazine-1-carboxamide
4-(isoquinolin-1-yl)-1-[(3-methoxyphenyl)methyl]piperazin-2-one
2-(2-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]methyl}-1H-pyrrol-1-yl)-1,3-thiazole
N-ethyl-6-[3-(2-ethylphenoxy)azetidin-1-yl]-N-methylpyridine-3-carboxamide
(4aS,8aR)-6-(5-chloro-6-oxo-1,6-dihydropyridine-3-carbonyl)-1-propyl-decahydro-1,6-naphthyridin-2-one
3-{[(butan-2-yl)amino]methyl}-6-cyclopentyl-2-methoxy-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
2-{5-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-1-(2-methylphenyl)-1H-1,2,4-triazol-3-yl}acetamide
3-{[({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)amino]methyl}pyrrolidin-3-ol
5-[3-(1,3-benzoxazol-2-yl)piperidine-1-carbonyl]-1-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-amino-1-[4-(2,5-dihydro-1H-pyrrol-1-yl)-2-(furan-2-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]ethan-1-one
4-[1-(2,2-dimethylpent-4-en-1-yl)pyrrolidin-2-yl]-3,5-dimethyl-1,2-oxazole
6-[4-(furan-3-carbonyl)-1,4-diazepane-1-carbonyl]-2-methyl-1,3-benzoxazole
(3aS,6aR)-5-[3-(2-methyl-1H-imidazol-1-yl)propyl]-3-[3-(morpholin-4-yl)propyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one