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(3S,4R)-1-{2-[(2R,6S)-2,6-dimethylpiperidin-1-yl]acetyl}-4-phenylpyrrolidine-3-carboxylic acid
2-(3-chlorophenoxy)-N-{2-[4-(4-methyl-1,4-diazepane-1-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl}propanamide
N-(furan-2-ylmethyl)-2,5-dimethyl-N-(prop-2-en-1-yl)-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
1-{2-[2-(trifluoromethyl)morpholin-4-yl]pyrimidin-4-yl}piperidin-4-ol
4-{[3-(3-methoxyphenyl)phenyl]methyl}-1,4-oxazepan-6-ol
2-(2,5-dimethoxyphenyl)-1-[7-(2,6-dimethoxyphenyl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethan-1-one
2-(dimethylamino)-2-(2-fluorophenyl)-N-{3-[methyl(phenyl)amino]propyl}acetamide
N-[2-(1H-indol-1-yl)ethyl]-N,5-dimethyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
2-benzyl-N-[2-(1H-imidazol-4-yl)ethyl]-1,3-thiazole-4-carboxamide
{[1-(1-cycloheptylpiperidin-4-yl)-1H-1,2,3-triazol-4-yl]methyl}(methyl)(2-methylpropyl)amine
2-(3-chloro-4-hydroxyphenyl)-N-[3-(1H-imidazol-1-yl)propyl]-N-(pyridin-4-ylmethyl)acetamide
1-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-(2-methoxyethoxy)ethan-1-one
2-ethoxy-4-{1-[(3R,4R)-4-(4-methylpiperazin-1-yl)oxolan-3-yl]-1H-imidazol-2-yl}phenol
2-{[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidin-1-yl]methyl}benzonitrile
1-(diphenylmethyl)-4-[(3-fluoropyridin-2-yl)methyl]piperazine
1-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]-3-phenoxypropan-1-one
[(6,7-dimethyl-1H-1,3-benzodiazol-2-yl)methyl](propan-2-yl)[(trimethyl-1H-pyrazol-4-yl)methyl]amine
2-{4-cyclobutanecarbonyl-1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecan-9-yl}acetic acid
5-[({[2-(azocan-1-yl)pyridin-3-yl]methyl}amino)methyl]-N,N-dimethyl-1,3-thiazol-2-amine
4-chloro-N-[(3S,5S)-1-(2-ethoxyethyl)-5-(ethylcarbamoyl)pyrrolidin-3-yl]-1H-pyrazole-3-carboxamide
8-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}-1,3-dioxa-8-azaspiro[4.5]decan-2-one
3-(3-chlorophenyl)-N-[(1-ethyl-1H-imidazol-2-yl)methyl]-3-phenylpropanamide
3-(dimethyl-1H-1,2,4-triazol-3-yl)-1-[2-(6-fluoro-1H-1,3-benzodiazol-2-yl)ethyl]urea
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-3-(pyridin-3-yl)propanamide
1-[(2-butyl-1H-imidazol-4-yl)methyl]-N-(3,4-difluorophenyl)piperidin-3-amine
2-{1-cyclohexyl-4-[(3,5-difluorophenyl)methyl]piperazin-2-yl}ethan-1-ol
ethyl 2-{4-[6-(2-chlorophenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]morpholin-3-yl}acetate
N-ethyl-2-{4-[2-(4-methylphenoxymethyl)furan-3-carbonyl]piperazin-1-yl}acetamide
(3R,4S)-1-[3-chloro-4-(pyrrolidin-1-yl)benzoyl]-3,4-dimethylpiperidin-4-ol
ethyl 4-[(4-chlorophenyl)methyl]-1-(1-methoxypropan-2-yl)piperidine-4-carboxylate
(4aS,7aR)-1-(5-ethyl-1,2-oxazole-3-carbonyl)-4-(pyrimidin-2-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[2-(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)ethyl]-2-(pyridin-4-yl)pyrimidine-5-carboxamide
8-[(2R)-2-amino-3-methylbutanoyl]-3-{2-[(2-methoxyethyl)(methyl)amino]ethyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N,N-bis(2-hydroxyethyl)-2-{3-oxo-1-[(3-phenoxyphenyl)methyl]piperazin-2-yl}acetamide
1-benzyl-4-{[3-methyl-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl]methyl}piperidine
7-ethoxy-4-[2-(propylsulfanyl)pyrimidin-5-yl]-1,2,3,4-tetrahydroquinolin-2-one
N-methyl-5-{5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carbonyl}-4H,5H,6H,7H-thieno[3,2-c]pyridine-2-carboxamide
3-({2-[2-(dimethylamino)ethyl]piperidin-1-yl}methyl)pyridin-2-amine
4-[2-methyl-4-(pyrrolidin-1-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-1-(prop-2-en-1-yl)pyrrolidin-2-one
(5-{[({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)(2-methylpropyl)amino]methyl}furan-2-yl)methanol
2-(1-methyl-1H-1,3-benzodiazol-2-yl)-N-{2-methyl-[1,2,4]triazolo[1,5-a]pyridin-8-yl}pyrrolidine-1-carboxamide
8-(1H-imidazol-4-ylmethyl)-2-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decan-3-one
N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}-3-oxo-3,4-dihydroquinoxaline-2-carboxamide
9-[(2,4-difluorophenyl)methyl]-2-[2-(pyridin-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
(3R,4S)-4-[ethyl({[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl})amino]oxolan-3-ol
3-methyl-1-[2-(oxolan-2-ylmethoxy)phenyl]-3-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}urea
methyl (2R,4S)-4-hydroxy-1-(3,4,7-trimethyl-1H-indole-2-carbonyl)piperidine-2-carboxylate
2-(3-fluorophenyl)-N-[1-(2-methyl-1,3-thiazol-4-yl)ethyl]-1,3-benzoxazole-5-carboxamide
N-[(1S,2R)-2-(cyclopentylamino)cyclobutyl]-1-(4-fluorophenyl)-3,5-dimethyl-1H-pyrazole-4-carboxamide
N-methyl-2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]-N-[(5-phenyl-1,2-oxazol-3-yl)methyl]acetamide