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1-{3-[(2-amino-5-ethylpyrimidin-4-yl)amino]piperidin-1-yl}ethan-1-one
N-{[6-chloro-4-(cyclopentylamino)quinazolin-2-yl]methyl}-1,3-thiazole-4-carboxamide
2-amino-2-(3,5-dimethyl-1H-pyrazol-4-yl)-N-{[2-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
1-[(3R,4S)-3-amino-4-(3-methoxyphenyl)pyrrolidin-1-yl]-2-[methyl(pyridin-4-ylmethyl)amino]ethan-1-one
3-chloro-4-fluoro-N-[2-(propane-2-sulfonyl)ethyl]-1-benzothiophene-2-carboxamide
N-[(2-methoxyphenyl)methyl]-1-[(2-methylphenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
4-({4-methyl-5-[1-(1,3-oxazole-4-carbonyl)piperidin-3-yl]-4H-1,2,4-triazol-3-yl}methyl)morpholine
7-methoxy-3-({4-[2-(pyridin-4-yl)ethyl]piperazin-1-yl}methyl)-1,2-dihydroquinolin-2-one
2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-[3-(pyridin-2-yl)propyl]acetamide
3-[({1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}(methyl)amino)methyl]pyrrolidin-3-ol
2-[3-(1H-imidazol-1-yl)propyl]-9-(4-methoxypyrimidin-2-yl)-2,9-diazaspiro[5.5]undecan-3-one
3-[1-(cyclopropylmethyl)-1H-pyrazol-5-yl]-1-[2-methoxy-2-(thiophen-2-yl)ethyl]urea
2,6-dimethoxy-N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)pyridine-3-carboxamide
1-(4-ethoxy-3-methylphenyl)-3-[3-(pyridazin-3-yl)-1,2,4-oxadiazol-5-yl]propan-1-one
(2S,4R)-1-(2,2-diphenylethyl)-4-[(1-methylpiperidin-4-yl)amino]-N-(propan-2-yl)pyrrolidine-2-carboxamide
4-(2-methyl-1H-imidazol-1-yl)-1-[4-(1H-1,2,3,4-tetrazol-1-yl)butanoyl]piperidine-4-carboxylic acid
3-{2-[3-(3-fluoro-4-phenylbenzoyl)piperidin-1-yl]-2-oxoethyl}-1,2,3-oxadiazol-3-ium-5-olate
4-{2-[(4aR,7aS)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-2-oxoethoxy}-3-methylbenzoic acid
4-hydroxy-2-[(4-methanesulfonamidopiperidin-1-yl)methyl]quinoline-6-carboxamide
1-(3-{[3-(3-methoxypiperidine-1-carbonyl)-1H-pyrazol-5-yl]methoxy}phenyl)ethan-1-one
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-N-{[1-(2-methoxyethyl)pyrrolidin-3-yl]methyl}acetamide
N-(2,1,3-benzoxadiazol-5-ylmethyl)-2-(2,4-dioxoimidazolidin-1-yl)acetamide
2-amino-4-cyclopropyl-6-(thiophene-2-carbonyl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
8-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
9-(5-ethyl-1H-pyrrole-2-carbonyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
N-(3-{4-[(3,5-dimethylphenyl)methyl]-3-oxopiperazin-1-yl}-3-oxopropyl)methanesulfonamide
2-(4-{[1-ethyl-3-(2-methyl-1,3-thiazol-4-yl)-1H-1,2,4-triazol-5-yl]methyl}piperazin-1-yl)pyrimidine
[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl](methyl)[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]amine
1-(8-chloroquinolin-5-yl)-3-[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]urea
2-(1-benzothiophen-7-yl)-N-methylbenzamide
3-(dimethyl-1,2-oxazol-4-yl)-N-[2-(4-sulfamoylphenyl)ethyl]propanamide
1-(dimethylamino)-2-(4-{[4-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)propan-2-ol
1-methanesulfonyl-4-[2-(4-methoxynaphthalen-1-yl)-1H-imidazol-1-yl]piperidine
2-[4-(3-benzyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]pyrrolidine-1-carboxamide
(1R,5S,6S)-N-(2,3-dihydro-1H-inden-2-yl)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3-azabicyclo[3.1.0]hexane-6-carboxamide
(1R,5S)-6-{3-[(4-methyl-1,2,3,6-tetrahydropyridin-1-yl)sulfonyl]benzoyl}-6-azabicyclo[3.2.1]octane
methyl[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl][3-(oxolan-2-yl)propyl]amine
1-({1-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]piperidin-3-yl}methyl)-1H-1,2,3-triazole-4-carboxylic acid
N-cyclopropyl-2-(morpholin-4-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]pyrimidine-5-carboxamide
2-(3-ethyl-1,2-oxazole-5-carbonyl)-7-[(3-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decane
(4aS,8aS)-2-{[2-fluoro-5-(trifluoromethyl)phenyl]methyl}-decahydro-2,7-naphthyridin-4a-ol
methyl (2S,4R)-1-[1-(2-phenylethyl)piperidin-4-yl]-4-(1,2,5-thiadiazole-3-amido)pyrrolidine-2-carboxylate
ethyl 4-(2-phenylethyl)-1-[1-(pyridin-3-yl)propan-2-yl]piperidine-4-carboxylate
4-[(2,6-difluorophenyl)methyl]-1-[(3-methoxyphenyl)methyl]piperazin-2-one
5-(7-chloro-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-methyl-1-(2-phenylethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
4-benzyl-3-[1-(4,6-dimethylpyrimidin-2-yl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
2-(4-phenylphenyl)-N-[2-(1H-pyrazol-4-yl)ethyl]acetamide
5-[1-(3-methylbutyl)-1H-imidazol-2-yl]-2-(pyrrolidin-1-yl)pyrimidine
(4aR,8aR)-1-(furan-2-carbonyl)-6-(3-methoxybenzoyl)-decahydro-1,6-naphthyridine
N-(2-chloro-4-fluoro-5-methylphenyl)-4-ethyl-2-methyl-3-oxopiperazine-1-carboxamide