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(2S)-2-{[3-(5-methylfuran-2-yl)-1H-pyrazol-5-yl]formamido}-3-phenylpropanamide
5-ethyl-2-{1-[2-methoxy-5-(4H-1,2,4-triazol-4-yl)phenyl]-1H-imidazol-2-yl}pyridine
6-{3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl}quinoline
1-(2,3-dimethylquinoxalin-6-yl)-3-[2-(N-methylmethanesulfonamido)ethyl]urea
(2,1,3-benzoxadiazol-4-ylmethyl)(methyl){2-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}amine
1-{[2-(propylamino)pyrimidin-5-yl]methyl}-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
2-(3-chlorophenyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
2-{3-[1-(carbamoylmethyl)-4-phenyl-1H-imidazol-5-yl]-2-methyl-1H-indol-1-yl}acetic acid
2-[4-(benzyloxy)butyl]-1,3-thiazole
5-methyl-N-[2-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
2-(morpholin-3-yl)-N-[2-(6-oxo-3-phenyl-1,4,5,6-tetrahydropyridazin-1-yl)ethyl]acetamide
N-[(3S,4R)-4-(propan-2-yl)-1-[5-(trifluoromethyl)pyridin-2-yl]pyrrolidin-3-yl]acetamide
2-(2-phenyl-1H-imidazol-1-yl)-N-{[2-(trifluoromethyl)phenyl]methyl}acetamide
3-{1-[3-(4-chloro-1H-pyrazol-1-yl)propanoyl]piperidin-4-yl}-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
3-{3-[3-(2-methylquinolin-4-yl)phenyl]-1H-pyrazol-1-yl}propan-1-ol
N-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-1H-pyrrolo[2,3-b]pyridin-6-amine
3,5-dimethyl-N-[3-(morpholin-4-yl)propyl]-1-benzofuran-2-carboxamide
N-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-5-methanesulfonyl-4-(piperidin-3-yl)pyrimidin-2-amine
2-{2-[1-(3-propyl-1H-pyrazole-5-carbonyl)piperidin-2-yl]ethyl}pyridine
N-cyclobutyl-3-{[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]sulfamoyl}benzamide
N-[1-(2,4-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(methylamino)acetamide
methyl N-{4-[2-(dimethylcarbamoyl)phenyl]phenyl}carbamate
N-[1-(2,3-dihydro-1H-inden-2-yl)-5-oxopyrrolidin-3-yl]-4-acetamidobutanamide
N,N-dimethyl-4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidine-1-sulfonamide
(1R,5S,6S)-N-tert-butyl-3-{[3-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}-3-azabicyclo[3.1.0]hexane-6-carboxamide
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[(4,6-dimethylpyridin-2-yl)methyl]-2-(1H-imidazol-2-yl)-N-methylbenzamide
N,N-bis(2-hydroxyethyl)-2-[1-(naphthalen-2-ylmethyl)-3-oxopiperazin-2-yl]acetamide
2-[1-(4-methoxyphenyl)-5-oxo-3-phenyl-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-methyl-N-propylacetamide
N-[2-methyl-1-(morpholin-4-yl)propan-2-yl]-5-(phenoxymethyl)-1H-pyrazole-3-carboxamide
3-(2-{4-[2-(pyridin-2-yl)pyrimidin-5-yl]-1H-1,2,3-triazol-1-yl}ethyl)-1,3-oxazinan-2-one
N3-ethyl-4-oxo-1-(2-phenylethyl)-N5-(1,2,3,4-tetrahydronaphthalen-1-yl)-1,4-dihydropyridine-3,5-dicarboxamide
2-[benzyl(methyl)amino]-N-{2-[(2R)-pyrrolidin-2-yl]ethyl}-2,3-dihydro-1H-indene-2-carboxamide
3-[(1-{[3-(thiophen-2-yl)-1H-pyrazol-4-yl]methyl}-1H-1,2,3-triazol-4-yl)methyl]-2,3-dihydro-1,3-benzoxazol-2-one
{1-[4-(1H-1,3-benzodiazol-2-yl)phenyl]ethyl}dimethylamine
1-(2-{[2-(5-methylfuran-2-yl)-1H-imidazol-1-yl]methyl}phenyl)-1H-1,2,4-triazole
N-{[4-(1H-imidazol-1-yl)phenyl]methyl}-N-methylthian-4-amine
4-(pyridin-2-yl)-N-(thiophen-2-ylmethyl)pyrimidin-2-amine
N-methyl-N-(2-phenylethyl)-1-[1-(pyridin-2-ylmethyl)piperidin-4-yl]piperidin-3-amine
1-[3-(2,5-difluorobenzoyl)piperidin-1-yl]-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
N-[4-ethoxy-3-(1H-pyrrol-1-yl)phenyl]-1,1-dioxo-1λ6-thiomorpholine-4-carboxamide
{1-[1-(2-aminoethyl)-1H-1,2,3-triazole-4-carbonyl]-3-(cyclopropylmethyl)piperidin-3-yl}methanol
N-[3-(1H-indazol-1-yl)propyl]-2,2-dimethyloxane-4-carboxamide
(3R,5S)-1-[(3,4-dimethoxyphenyl)methyl]-5-(3-fluorophenoxymethyl)-N-[3-(morpholin-4-yl)propyl]piperidine-3-carboxamide
N-[(3-benzyl-1H-1,2,4-triazol-5-yl)methyl]-4-fluoro-3-methylbenzene-1-sulfonamide
{[7-fluoro-2-(3-methoxyphenyl)quinolin-3-yl]methyl}(thiophen-2-ylmethyl)amine
5-ethyl-N-{2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}pyrazolo[1,5-a]pyrimidin-7-amine
1-{[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2-(2-methoxyethyl)piperidine
1-{1-[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl]piperidin-4-yl}piperidin-3-ol
(2H-1,3-benzodioxol-5-ylmethyl)(1H-imidazol-2-ylmethyl)[(4-methylphenyl)methyl]amine