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2-[4-(1H-1,2,4-triazole-3-carbonyl)piperazin-1-yl]-4-(3,3,3-trifluoropropyl)pyrimidine
N-{1-[1-(pent-4-enoyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2H-1,3-benzodioxole-5-carboxamide
1-{4-[4-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]thiophen-2-yl}ethan-1-one
1-[6-(2,6-dimethylphenyl)pyridine-3-carbonyl]-4-(pyrimidin-2-yl)-1,4-diazepane
(4aR,8aS)-N,N-dimethyl-1-[2-(2,4,6-trifluorophenyl)acetyl]-decahydro-1,6-naphthyridine-6-sulfonamide
N-[4-(3-methylphenyl)phenyl]-1-(oxan-4-yl)piperidine-4-carboxamide
4-oxo-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-3,4-dihydroquinazoline-2-carboxamide
4-(3-methylbutyl)-1-(2-methylphenyl)piperazin-2-one
N-(carbamoylmethyl)-2-{1-[(2-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
2-{[(4-fluorophenyl)methyl](methyl)amino}-1-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
5-methyl-2-[1-(pyridine-4-carbonyl)-4-(pyrrolidin-1-ylmethyl)piperidin-4-yl]pyridine
2-(3-methoxypropyl)-8-[4-methyl-6-(methylamino)pyrimidin-2-yl]-2,8-diazaspiro[5.5]undecan-3-one
N-[2-(1-methylpiperidin-3-yl)ethyl]-1-phenyl-1H-1,2,3-triazole-5-carboxamide
2-{[1-(1-methylpiperidin-4-yl)-3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]methyl}morpholine
[1-(3-fluorophenyl)propan-2-yl]({imidazo[1,2-a]pyridin-2-ylmethyl})amine
N-(4-fluorophenyl)-2-[2-(1H-imidazol-4-yl)ethyl]-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
(1S,5R)-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-3,9-diazabicyclo[3.3.2]decan-10-one
N-[2-(dimethylamino)ethyl]-5-methyl-4-{[1-(thiophen-2-yl)propyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
(1R,5R)-6-(cyclobutylmethyl)-3-(5-methyl-1,2-oxazole-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
2-(furan-2-yl)-1-[(2-methyl-1,3-thiazol-4-yl)methyl]azepane
4-(1-methyl-1H-pyrazol-4-yl)-N-[2-(1-methylpyrrolidin-2-yl)ethyl]pyrimidin-2-amine
2-{1-[(2-methylphenyl)methyl]-4-[1-(2-methylphenyl)piperidin-4-yl]piperazin-2-yl}ethan-1-ol
N-[(3R,4S)-4-cyclopropyl-1-(6-methylpyrimidin-4-yl)pyrrolidin-3-yl]-2-(2,4-dioxoimidazolidin-1-yl)acetamide
N-[1-(cyclopropylmethyl)-1H-indazol-3-yl]-2-(4,5-dichloro-2-methyl-1H-imidazol-1-yl)acetamide
[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl](methyl){[5-methyl-2-(naphthalen-2-yl)-1,3-oxazol-4-yl]methyl}amine
9-{[4-chloro-2-(dimethylamino)-1,3-thiazol-5-yl]methyl}-1-oxa-9-azaspiro[5.5]undecan-5-ol
2-[4-(4-methoxy-2-methylphenyl)phenyl]-2-methylpropanamide
1-(cyclopropylmethyl)-5-(3,4-dimethoxybenzoyl)-N-methyl-N-(1,3-thiazol-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
3-{5-[(3-methylphenyl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
N-({2-[cyclohexyl(methyl)amino]pyridin-3-yl}methyl)-2-(3,6-dioxo-1,2,3,6-tetrahydropyridazin-4-yl)acetamide
1-[(1R,3S)-1-hydroxy-3-methoxy-7-azaspiro[3.5]nonane-7-carbonyl]cyclopropane-1-carboxamide
4-(3-cyclopropyl-1H-1,2,4-triazol-5-yl)benzene-1-sulfonamide
(3aR,6aR)-2-(3-chloro-2-fluorobenzoyl)-5-(cyclobutylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
7-[3-(2-ethyl-1H-imidazol-1-yl)propanoyl]-2-(pyridin-3-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-{2-methyl-2,8-diazaspiro[4.5]decan-8-yl}but-3-en-1-one
(4aR,7aS)-1-[2-(dimethylamino)acetyl]-4-methanesulfonyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-(3-methoxypropyl)-1-[2-methyl-2-(morpholin-4-yl)propyl]piperidine-3-carboxylic acid
3-(cyclopropylmethyl)-1-ethyl-5-(2-ethyl-4-methyl-1,3-thiazol-5-yl)-1H-1,2,4-triazole
1-(2,3-dihydro-1H-inden-2-yl)-4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidine
1-[(3aS,6aS)-3a-(hydroxymethyl)-octahydrocyclopenta[c]pyrrol-2-yl]-2-(2,4-dichlorophenoxy)ethan-1-one
4-{3-[4-(furan-2-carbonyl)piperazine-1-carbonyl]-6-(4-methoxyphenyl)pyridin-2-yl}thiomorpholine
(2S,4S)-1-[(2-chlorophenyl)methyl]-N-(2-methoxyethyl)-4-{[(3-methoxyphenyl)methyl]amino}pyrrolidine-2-carboxamide
6-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-2,5-dioxo-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
butyl(furan-2-ylmethyl)(1H-imidazol-2-ylmethyl)amine
(3aS,7aR)-5-methyl-2-[3-(trimethyl-1H-pyrazol-4-yl)propanoyl]-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
1-[(3-methoxyphenyl)methyl]-6-oxo-N-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]piperidine-3-carboxamide
N,3-dimethyl-N-[(3-phenyl-1H-pyrazol-4-yl)methyl]furan-2-carboxamide
ethyl 5-(dimethyl-1,3-thiazole-5-carbonyl)-1-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
2-methoxy-1-[8-(morpholine-4-sulfonyl)-1,2,3,4-tetrahydroisoquinolin-2-yl]ethan-1-one
3-[2-oxo-2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]-4-(2-phenylethyl)piperazin-2-one