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3-ethyl-1-(4-methoxypyrimidin-2-yl)piperidine-3-carboxylic acid
2-(2-aminoethyl)-N-{1-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]ethyl}quinazolin-4-amine
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-4,5,6,7-tetrahydro-1,2-benzoxazole-3-carboxamide
1-butyl-5-{7-methylpyrazolo[1,5-a]pyrimidin-6-yl}-1H-1,2,4-triazole
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-1-methyl-1H-1,2,3-benzotriazole-5-carboxamide
N-[1-(2-phenylethyl)piperidin-3-yl]pyridine-2-carboxamide
1-[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl]-4-(4-methoxybenzoyl)piperazine
4-({4-methyl-5-[1-(4-methylbenzoyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)morpholine
2-butyl-5-[3-(pyridine-2-carbonyl)piperidine-1-carbonyl]-1,3-benzoxazole
(3S)-1-{5-[(3R)-3-hydroxypyrrolidine-1-carbonyl]-1-methyl-1H-1,3-benzodiazol-2-yl}pyrrolidin-3-ol
1-ethyl-3-methyl-N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(pyridin-3-ylmethyl)-1H-pyrazole-5-carboxamide
1-{1,3-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}azonane
3-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}-1,2-dihydropyridin-2-one
2-(dimethylamino)-2-(4-fluorophenyl)-N-[(2-methoxy-4,6-dimethylpyridin-3-yl)methyl]acetamide
3-(4-fluorophenyl)-N-(oxolan-2-ylmethyl)-N-{[4-(pyridin-3-ylmethoxy)phenyl]methyl}benzamide
14-[5-(1H-pyrazol-3-yl)furan-2-yl]-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
4-{[(1R,3S,3aS,6aR)-5-ethyl-1-(hydroxymethyl)-3-(2-methylphenyl)-octahydropyrrolo[3,4-c]pyrrol-1-yl]methyl}phenol
N-ethyl-3-(3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidin-1-yl)propanamide
4-{3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl}butan-1-ol
1-cyclohexyl-N3-methyl-4-oxo-N5-[(4-phenyloxan-4-yl)methyl]-1,4-dihydropyridine-3,5-dicarboxamide
(4aR,7aS)-1-(2-methylpropanoyl)-4-[3-(1H-pyrazol-1-yl)propanoyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-{[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1-phenylpiperazin-2-one
1-(2H-1,3-benzodioxol-5-ylmethyl)-2-[5-(oxan-2-yl)furan-2-yl]-1H-imidazole
1-[4-({3-[2,2-bis(prop-2-en-1-yl)piperidine-1-carbonyl]-1,2-oxazol-5-yl}methoxy)phenyl]ethan-1-one
N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1-[3-(2-methylphenyl)phenyl]piperidin-4-amine
2-{1-methyl-4-[(2-methyl-1-benzothiophen-3-yl)methyl]piperazin-2-yl}ethan-1-ol
(2S,4S)-4-amino-1-(2,3-dihydro-1H-indene-5-carbonyl)pyrrolidine-2-carboxylic acid
1-{1-[(2-butyl-1H-imidazol-4-yl)methyl]piperidin-3-yl}-4-(3-chlorophenyl)piperazine
3-(diphenylmethyl)-N-methyl-N-(thiophen-2-ylmethyl)-1,2-oxazole-5-carboxamide
N-[2-(piperidin-1-yl)-2-(pyridin-3-yl)ethyl]-4-(1H-pyrazol-1-yl)benzamide
2-methyl-6-[4-(pyridin-2-ylmethyl)-1,4-diazepane-1-carbonyl]-4H-pyran-4-one
N-[(1-methanesulfonylpiperidin-3-yl)methyl]-2-(4H-1,2,4-triazol-4-yl)pyridine-4-carboxamide
4-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]-N-(4-methylpyridin-3-yl)morpholine-2-carboxamide
(3aS,7aR)-5-methyl-2-[3-(1-oxo-2,3-dihydro-1H-isoindol-2-yl)propanoyl]-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
N-[(3R,5S)-5-[(3aR,7aS)-2,3,3a,4,7,7a-hexahydro-1H-isoindole-2-carbonyl]pyrrolidin-3-yl]-4-methoxybenzamide
2-[2-(3,4-dichlorophenyl)morpholin-4-yl]pyridine-3-carbonitrile
2-(4-cyclopentylpiperazin-1-yl)-2-(4-methoxy-3-methylphenyl)acetic acid
1-(5-phenyl-1,2-oxazole-3-carbonyl)-4-(pyridin-3-ylmethyl)-1,4-diazepane
1-{[1-(3-chlorophenyl)-1H-pyrazol-4-yl]methyl}-4-ethyl-1,4-diazepane
N,N-dimethyl-1-(4,5,6,7-tetrahydro-1-benzothiophene-3-carbonyl)azepan-4-amine
4-[(2,6-dimethylpyridin-3-yl)oxy]-1-(6-methylpyridazin-3-yl)piperidine-4-carboxylic acid
N-[3-(2-ethyl-1H-imidazol-1-yl)propyl]-3,6-dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
2-(3-chlorophenoxy)-1-[4-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]propan-1-one
N-{[7-methoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}-5-methyl-N-[3-(2-oxopyrrolidin-1-yl)propyl]thiophene-2-carboxamide
3-(1H-1,3-benzodiazol-1-yl)-1-{4-[(4-chlorophenyl)methyl]-4-(hydroxymethyl)piperidin-1-yl}propan-1-one
1-[(4-methyl-1H-imidazol-5-yl)methyl]-4-(1,2,4-oxadiazol-3-yl)piperidine
5-{5,6-dimethylthieno[2,3-d]pyrimidin-4-yl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonitrile
N,5-dimethyl-N-[1-(3-phenylpropyl)piperidin-3-yl]thiophene-2-carboxamide
8-(6-aminopyrimidin-4-yl)-2-[(3,5-difluorophenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
N-(2-{[3-(dimethylsulfamoyl)-5-{[(3-ethoxy-4-hydroxyphenyl)methyl]amino}phenyl]formamido}ethyl)acetamide