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4-{[2-(4-methoxyphenyl)-7-methylquinolin-3-yl]methyl}-3-methylpiperazin-2-one
N-{2-[({5-[(dimethylamino)methyl]furan-2-yl}methyl)sulfanyl]ethyl}-6-(piperidin-4-yl)pyrimidin-4-amine
{[2-(azocane-1-carbonyl)-6-chloroimidazo[1,2-a]pyridin-3-yl]methyl}(methyl)[2-(1H-pyrazol-4-yl)ethyl]amine
7-methoxy-3-({methyl[(2-methyl-1,3-thiazol-4-yl)methyl]amino}methyl)-1,2-dihydroquinolin-2-one
4-(1-{1-[(4-ethylphenyl)methyl]piperidin-4-yl}-1H-1,2,3-triazole-4-carbonyl)morpholine
2-[5-(2-methyl-1H-1,3-benzodiazol-5-yl)-3-(oxolan-3-yl)-1H-1,2,4-triazol-1-yl]acetic acid
1-(5-ethyl-1,3,4-oxadiazol-2-yl)-4-[3-(pyrrolidin-1-yl)propyl]-1,4-diazepane
N-[(3R,4S)-1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-4-propylpyrrolidin-3-yl]cyclopropanesulfonamide
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-3-(furan-2-yl)-N-methylbenzamide
3-[(1-ethyl-1H-imidazol-2-yl)methyl]-3-methyl-1-[4-(propylsulfanyl)phenyl]urea
N-(1-cycloheptylpiperidin-3-yl)-3-(morpholin-4-yl)propanamide
4-[3-(propan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]-5,6,7,8-tetrahydroquinazolin-2-amine
1-(2-ethoxyethyl)-2-oxo-N-(1-phenylcyclopropyl)-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
5-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-methyl-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)-1H-pyrazole-3-carboxamide
2-(4-fluorophenyl)-1-(1H-pyrrole-2-carbonyl)piperidine
6-oxo-4-[5-(1H-pyrazol-3-yl)thiophen-2-yl]-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridine-3-carboxylic acid
3-[5-(3,5-dimethyl-1-benzofuran-2-carbonyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl]pyridine
1-{2-hydroxy-3-[4-methoxy-2-({methyl[(4-methyl-1H-imidazol-2-yl)methyl]amino}methyl)phenoxy]propyl}piperidin-4-ol
1-(4-ethylpiperazin-1-yl)-3-[3-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)phenoxy]propan-2-ol
4-cyclopropanecarbonyl-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-[4-(2-aminopyrimidin-4-yl)piperidine-1-carbonyl]-6-methyl-1,2-dihydropyridin-2-one
1-[(4-fluoro-3-methoxyphenyl)methyl]-3-(pyrrolidin-1-ylmethyl)piperidin-3-ol
N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]-3-(piperidin-4-ylmethyl)benzamide
1-methyl-6-(2-phenylethyl)-N-(pyridin-3-ylmethyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
{[1-(1,4-dioxan-2-ylmethyl)-3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]methyl}(ethyl)methylamine
(2S)-1-acetyl-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]pyrrolidine-2-carboxamide
ethyl 3-[(3-chlorophenyl)methyl]-1-(2,3-dimethoxybenzoyl)piperidine-3-carboxylate
3-methyl-1-{4-[2-methyl-6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-1-yl}butan-1-one
4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}-N-propylpiperidine-1-carboxamide
1-(4-methoxyphenyl)-N-[(1-methylpiperidin-3-yl)methyl]cyclopentane-1-carboxamide
3-acetamido-N-ethyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}thiophene-2-carboxamide
4-[3-(1H-imidazol-1-ylmethyl)piperidin-1-yl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-2-amine
N-[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]-N-methyl-2,1-benzoxazole-3-carboxamide
(3aR,7aS)-2-[4-(piperidin-1-ylmethyl)benzoyl]-2,3,3a,4,7,7a-hexahydro-1H-isoindole
(1S,5R)-6-(cyclopropylmethyl)-3-(2,4-dimethoxybenzoyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
(2R,6S)-2,6-dimethyl-4-(1-{5-[(methylsulfanyl)methyl]pyridin-2-yl}piperidin-4-yl)morpholine
2,5-dimethyl-3-(2,3,4-trimethoxyphenyl)pyrazine
2-(cyclopentylmethyl)-6-methyl-N-[2-(morpholin-4-yl)ethyl]-4-oxo-1-[3-(2-oxopyrrolidin-1-yl)propyl]-1,4-dihydropyridine-3-carboxamide
3-(3-chlorophenyl)-N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-3-(3-hydroxyphenyl)propanamide
3-(4-methoxyphenoxymethyl)-1-(3-methyl-1,2-oxazole-5-carbonyl)piperidine
2-(3-{[methyl(thiophen-2-ylmethyl)amino]methyl}phenyl)-6-(oxolan-2-yl)-3,4-dihydropyrimidin-4-one
(3aR,6aR)-2-acetyl-5-[1-(pyridine-3-carbonyl)piperidin-4-yl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-{4-[(4-fluoropiperidin-1-yl)methyl]phenyl}-6-(4-hydroxyphenyl)-3,4-dihydropyrimidin-4-one
methyl(pyridin-3-ylmethyl){[2-(pyrrolidin-1-ylmethyl)phenyl]methyl}amine
1-methyl-N-[2-(5-methylfuran-2-yl)ethyl]-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-[(2-fluorophenyl)methyl]-4-[(6-methylpyridin-2-yl)methyl]-1,4-diazepane
methyl(1,2-oxazol-3-ylmethyl){[6-(thiophen-2-yl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}amine
N-(1,4-dioxan-2-ylmethyl)-N-methyl-5-[3-(trifluoromethyl)phenoxymethyl]-1H-pyrazole-3-carboxamide
N-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-1-[(2-fluorophenyl)methyl]piperidin-4-amine
2-methyl-4-oxo-N-[(2-phenoxypyridin-3-yl)methyl]-4,5,6,7-tetrahydro-1-benzofuran-3-carboxamide