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N-[(1-benzyl-1H-imidazol-2-yl)methyl]-2-tert-butyl-4-hydroxy-N-methylpyrimidine-5-carboxamide
N-methyl-N-(quinolin-5-ylmethyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
N-cyclopentyl-2-methyl-N-[(5-methylthiophen-2-yl)methyl]-1,3-thiazole-4-carboxamide
3-(4-methyl-4H-1,2,4-triazol-3-yl)-1-(3-phenylpiperazin-1-yl)propan-1-one
({6-chloro-2-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]imidazo[1,2-a]pyridin-3-yl}methyl)[(3-ethyl-1,2-oxazol-5-yl)methyl]amine
(3-{2-[1-(isoquinolin-1-yl)piperidin-3-yl]-1H-imidazol-1-yl}propyl)dimethylamine
(1R,2S,4R)-N-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)bicyclo[2.2.1]hept-5-ene-2-carboxamide
methyl 6-(2-cyclopropylacetyl)-2-[(2,3-dihydro-1H-inden-5-yl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
4-[5-({4-[(2-fluorophenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}methyl)thiophen-2-yl]-2-methylbut-3-yn-2-ol
3-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-2-methyl-4,5,6,7-tetrahydro-1H-indol-4-one
N,N-bis(1,3-oxazol-4-ylmethyl)-2-{2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-3-yl}acetamide
2-methyl-6-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridine
3-(5-fluoro-2-methylphenyl)-5-[3-(1H-1,2,4-triazol-1-yl)propyl]-1,2,4-oxadiazole
4-chloro-N-[2-(2-hydroxyethoxy)ethyl]-1-methyl-1H-indole-2-carboxamide
N-[3-(5-amino-1,3,4-thiadiazol-2-yl)propyl]-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
1-[1-(oxan-4-yl)piperidine-3-carbonyl]-4-(1,3-thiazol-2-yl)piperazine
N-[(5-chloro-3-methyl-2-phenyl-1H-indol-7-yl)methyl]-1-(methoxymethyl)cyclobutane-1-carboxamide
(1S,5R)-6-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
4-(4-{[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-1-yl)quinazoline
(2R,3R,6R)-3-(4-fluorophenyl)-5-(quinolin-2-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
5-[5-chloro-2-(prop-2-en-1-yloxy)phenyl]-1-methyl-1H,4H-pyrazolo[3,4-d]imidazole
7-{[4-(benzyloxy)piperidin-1-yl]methyl}-4-(thiophen-2-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
6-methyl-1-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]-4-(trifluoromethyl)-1,2-dihydropyridin-2-one
N-methyl-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-2-(thiophene-2-sulfonamido)acetamide
4-{2-[4-(dimethylamino)phenyl]acetyl}-1-[(4-methylphenyl)methyl]piperazin-2-one
1-{2-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-1-yl]-2-oxoethyl}piperidin-2-one
1-(4-chlorophenyl)-5-methyl-4-(3-propyl-1H-pyrazole-4-carbonyl)piperazin-2-one
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-2-(1H-1,2,3,4-tetrazol-5-yl)benzamide
N-[(2S)-1-hydroxy-3-methylbutan-2-yl]-6-[4-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
2-[4-(1H-indol-2-ylmethyl)-1-(3-methylbut-2-en-1-yl)piperazin-2-yl]ethan-1-ol
(1R,3S)-3-{3-benzyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl}cyclopentan-1-amine
N-(2-phenylethyl)-1-{2-[(2,3,4-trimethoxyphenyl)formamido]ethyl}-1H-1,2,3-triazole-4-carboxamide
3-{[4-(2-methylphenoxy)piperidin-1-yl]methyl}pyridin-2-amine
4-[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-methyl-1H-1,2,4-triazol-5-yl]morpholine
3-(1-methylcyclopropyl)-1-{4-[3-(4-methylpiperazine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}propan-1-one
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-8-methylimidazo[1,2-a]pyridine-2-carboxamide
2-ethyl-6-methyl-N-[3-(morpholin-4-yl)propyl]-4-oxo-1-[2-(piperidin-1-yl)ethyl]-1,4-dihydropyridine-3-carboxamide
1-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}-8-(pyridin-2-yl)-1,8-diazaspiro[4.5]decane
4-[4-methyl-2-(piperidin-1-yl)pyrimidine-5-carbonyl]-1,4-oxazepan-6-ol
8-(5-chlorothiophene-2-carbonyl)-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
[(4-chloro-1-methyl-1H-pyrazol-3-yl)methyl][3-(1H-imidazol-1-yl)propyl](pyridin-3-ylmethyl)amine
3-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-{[4-(2-methylpropyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}benzamide
(2S,4S)-N-methyl-4-[4-(pyrrolidin-1-ylmethyl)-1H-1,2,3-triazol-1-yl]pyrrolidine-2-carboxamide
N-(4-fluorophenyl)-1-(1-methyl-1H-indole-3-carbonyl)piperazine-2-carboxamide
2-amino-2-methyl-1-(4-{4-methyl-5-[(4-methylpiperazin-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)propan-1-one
3,3-dimethyl-1-{2-oxo-2-[4-oxo-2-(pyridin-2-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethyl}urea
4-(1-{5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperidin-4-yl)morpholine
2-{4-[(1S,4S)-2-azabicyclo[2.2.1]heptan-2-ylmethyl]phenyl}-6-(pyridin-3-yl)-3,4-dihydropyrimidin-4-one
N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-3-(trimethyl-1H-pyrazol-4-yl)propanamide