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1-[4-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]-3-[2-(2-oxo-1,3-oxazinan-3-yl)ethyl]urea
5-{4-[1-(4-methylpiperazin-1-yl)ethyl]piperidine-1-carbonyl}pyridin-2-amine
1-ethyl-5-{1-[1-(1-methyl-1H-pyrazol-5-yl)propyl]-4-phenyl-1H-imidazol-5-yl}-1H-1,2,4-triazole
(2S,4S)-4-amino-1-{[3-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl}pyrrolidine-2-carboxylic acid
2-(3-chloro-5-fluorophenyl)-N-(propan-2-yl)pyrimidin-4-amine
N-(2,5-dimethoxyphenyl)-5-[1-(2,2-dimethylpropyl)-4-hydroxypiperidin-4-yl]-1-benzofuran-2-carboxamide
3-(3-hydroxy-3-methylbutyl)-N-[2-(quinolin-8-yloxy)ethyl]benzamide
(4aS,7aR)-1-[(4-acetylphenyl)methyl]-4-(3-methylbut-2-en-1-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[3-(furan-2-yl)phenyl]-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}piperidin-4-amine
(2E)-N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)-3-(pyridin-4-yl)prop-2-enamide
N,5-dimethyl-N-(1,3-thiazol-4-ylmethyl)-4-{[1-(thiophen-2-yl)ethyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
1-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-2-[2-(thiophen-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethan-1-one
6-fluoro-2-({[(1-methanesulfonylpiperidin-3-yl)methyl]amino}methyl)quinolin-4-ol
N-(1-{[2-(naphthalen-1-yl)pyrimidin-5-yl]methyl}piperidin-3-yl)acetamide
2-[(5-propylfuran-2-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
4-(2-{1-[2-(phenylsulfanyl)ethyl]piperidin-2-yl}ethyl)morpholine
5-chloro-2-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine
N-[1-(3-cyanopyridin-2-yl)piperidin-4-yl]-3-cyclohexyl-1H-pyrazole-4-carboxamide
(3S,4S)-1-({5-[(2E)-2-methylbut-2-en-1-yl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-4-(morpholin-4-yl)pyrrolidin-3-ol
5-methanesulfonyl-2-methyl-N-{[1-(4-methylphenyl)pyrrolidin-3-yl]methyl}pyrimidin-4-amine
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}pent-4-enamide
2-(4-chloro-1H-pyrazol-1-yl)-1-[4-(dimethylamino)-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]propan-1-one
3-(1-methyl-1H-imidazole-2-carbonyl)-1-{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}piperidine
2-[(3-methoxyphenyl)methyl]-4-(oxane-4-carbonyl)morpholine
4-[(3,5-dimethoxyphenyl)methyl]-3-{2-[4-(2-methoxyethyl)piperazin-1-yl]-2-oxoethyl}piperazin-2-one
2-{5-[2-(1H-pyrazol-1-yl)benzoyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl}ethan-1-ol
1-[4-({[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl](methyl)amino}methyl)thiophen-2-yl]ethan-1-one
1-methyl-2-{[(1S,5R)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-1H-1,3-benzodiazole
4-(4-hydroxyphenyl)-N-(prop-2-en-1-yl)-N-(propan-2-yl)benzamide
8-{[3-(4-methoxyphenoxy)phenyl]methyl}-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
({5-[1-(cyclopropanesulfonyl)piperidin-4-yl]-4-ethyl-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
N2-[(2,3-dimethyl-1H-indol-5-yl)methyl]pyrimidine-2,4-diamine
4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]-1-[(3-methylphenyl)methyl]piperidine
2-{5-[3-(difluoromethoxy)phenyl]-3-[(1-methylpiperidin-4-yl)methyl]-1H-1,2,4-triazol-1-yl}ethan-1-ol
(furan-2-ylmethyl)({[2-methanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl})methylamine
N-(furan-2-ylmethyl)-N-{[2-(3-methoxyphenyl)-7-(methylsulfanyl)quinolin-3-yl]methyl}-4-methylbenzamide
3-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-3-methyl-1-{2-[2-(pyridin-2-yl)ethyl]phenyl}urea
3-[1-(2-methoxyethyl)-2-methyl-1H-indol-5-yl]-1-[(3-propyl-1,2-oxazol-5-yl)methyl]urea
N-methyl-2-(morpholin-4-yl)-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}benzamide
N-[3-({cyclopropyl[(5-methylthiophen-2-yl)methyl]carbamoyl}amino)phenyl]butanamide
4-[3-(2-ethylpiperidine-1-carbonyl)benzenesulfonyl]-1,4-oxazepane
N-[3-(2-amino-1,3-thiazol-4-yl)propyl]-6-methoxy-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl](methyl){[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}amine
8-(6-methyl-2-phenylpyrimidin-4-yl)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
2-{8-benzyl-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}-2-oxo-N-propylacetamide
1-(4-aminoazepan-1-yl)-2-(4-chloro-3,5-dimethylphenoxy)-2-methylpropan-1-one
N-[(3R,4S)-1-[(5-methylpyrazin-2-yl)methyl]-4-propylpyrrolidin-3-yl]oxane-4-carboxamide
3-{3-[(2-methylphenyl)methoxy]azetidine-1-carbonyl}-5-(propan-2-yl)-1,2-oxazole
1-(6-methylpyridine-3-carbonyl)-N-[3-(1H-pyrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
5-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]-2-(1H-pyrazol-4-yl)pyridine