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N-(2-oxo-2,3-dihydro-1H-indol-5-yl)-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine-1-carboxamide
N-(3,3-diphenylpropyl)-6-[3-(1H-1,2,4-triazol-1-yl)propanoyl]-6-azaspiro[2.5]octane-1-carboxamide
1-[4-(5-chloropyridin-2-yl)piperazin-1-yl]-2-(thiophen-3-yl)ethan-1-one
1-(carbamoylmethyl)-N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}piperidine-3-carboxamide
4-[(5-methylfuran-2-yl)methyl]-3-{2-oxo-2-[4-(pyridin-2-ylmethyl)-1,4-diazepan-1-yl]ethyl}piperazin-2-one
4-{1-[(6-ethoxypyridin-3-yl)methyl]piperidin-4-yl}thiomorpholine
N-({7-chloro-2-[3-(hydroxymethyl)piperidin-1-yl]quinolin-3-yl}methyl)-N-(2-methoxyethyl)-5,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
N-methyl-N-[(3-methylthiophen-2-yl)methyl]-5-{[2-(propan-2-yl)-1H-imidazol-1-yl]methyl}-1H-pyrazole-3-carboxamide
4-{[(2-methoxyethyl)[(2E)-3-phenylprop-2-en-1-yl]amino]methyl}benzoic acid
1-ethyl-6-{[(2S)-2-(methoxymethyl)pyrrolidin-1-yl]methyl}-1H-indole
2-(2-chloro-4-fluorophenyl)-2-[methyl(pyridin-2-ylmethyl)amino]acetic acid
4-methyl-6-{4-[3-(2-methylpiperidin-1-yl)azetidin-1-yl]piperidin-1-yl}-2-propylpyrimidine
[9-(naphthalen-2-ylmethyl)-3,9-diazaspiro[5.5]undecan-1-yl]methanol
5-{4-[(3-methylpyridin-2-yl)methyl]piperazine-1-carbonyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
N4-{2-[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]ethyl}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-2,4-diamine
7-{[2-(benzylsulfanyl)pyrimidin-5-yl]methyl}-1-oxa-3,7-diazaspiro[4.5]decan-2-one
N-(1-{5-[(cyclohexylmethyl)sulfanyl]-4-methyl-4H-1,2,4-triazol-3-yl}-2-phenylethyl)-4-fluorobenzene-1-sulfonamide
4-[3-(3,4-difluorophenyl)-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl]-1-methylpiperidin-4-ol
N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-5-(pyridin-4-yl)pyrazolo[1,5-a]pyrimidin-7-amine
5-[3-(2,5-dimethoxyphenyl)pyrrolidine-1-carbonyl]-2-methoxy-4-methyl-1,3-thiazole
1-(carbamoylmethyl)-N-[2-(3-fluorophenyl)-2-hydroxyethyl]piperidine-4-carboxamide
3-(pentan-2-yl)-8-{pyrazolo[1,5-a]pyridine-7-carbonyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(1-{[3-(3-fluorophenyl)phenyl]methyl}piperidin-4-yl)(1-methyl-1H-imidazol-2-yl)methanol
N-(4-pentylphenyl)-4-(pyridin-2-ylmethyl)-1,4-diazepane-1-carboxamide
N,7-dimethyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}imidazo[1,2-a]pyridine-2-carboxamide
2-{1-[(4-methanesulfonylphenyl)methyl]azetidin-3-yl}pyridine
(2R,4S)-1-[2-(3-chloro-4-hydroxyphenyl)acetyl]-4-hydroxypiperidine-2-carboxylic acid
1-(furan-2-ylmethyl)-N-{2-[(3-methylpyridin-2-yl)amino]ethyl}piperidine-4-carboxamide
N-methyl-4-[(2-methylpyridin-3-yl)oxy]-N-(oxan-2-ylmethyl)piperidine-4-carboxamide
5-oxo-1-{2-[2-(pyrrolidin-1-yl)acetamido]phenyl}pyrrolidine-3-carboxylic acid
N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-(2-methoxyethyl)piperidine-4-carboxamide
4-[(6-methylpyridin-3-yl)oxy]-1-pentylpiperidine-4-carboxylic acid
1-[(3R,4S)-3-amino-4-phenylpyrrolidin-1-yl]-2-[3-(1H-1,2,3,4-tetrazol-1-yl)phenoxy]ethan-1-one
N-(2-ethyl-4-{1H-pyrazolo[3,4-b]pyridin-1-yl}phenyl)acetamide
8-(2-ethyl-6-methylpyrimidin-4-yl)quinoline
1-[5-(2-ethoxypyridin-3-yl)-1H-1,3-benzodiazol-2-yl]ethan-1-ol
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-5-methoxy-1-methyl-1H-indole-2-carboxamide
3-[(3R,4S)-4-(4-methylpiperazin-1-yl)-1-[4-(2-methylpropyl)benzoyl]piperidin-3-yl]propan-1-ol
14-[3-ethoxy-4-hydroxy-5-(prop-2-en-1-yl)phenyl]-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
4-(6-{4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl)thiomorpholine
3-[(3R,4S)-4-(4-methylpiperazin-1-yl)-1-(quinolin-2-yl)piperidin-3-yl]propanoic acid
4-{4-[(4-ethoxyphenyl)methyl]piperazin-1-yl}-2-[2-(3-fluorophenyl)ethyl]-2,3-dihydro-1H-isoindole-1,3-dione
N-methyl-N-{[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}-1H-pyrazole-4-carboxamide
1-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)sulfonyl]-4-hydroxypiperidine-4-carboxylic acid
N-[(1R)-1-(4-chlorophenyl)ethyl]-4-[4-(methoxymethyl)-1H-1,2,3-triazol-1-yl]piperidine-1-carboxamide
4-({3-azaspiro[5.5]undecan-9-yl}amino)-1-(2-methoxyethyl)pyrrolidin-2-one
N-(1,3-thiazol-2-yl)-3-{[6-(4H-1,2,4-triazol-4-yl)pyridin-3-yl]formamido}propanamide
4-(1-{[2-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carbonyl)morpholine
(3S,4S)-4-[(dimethylamino)methyl]-1-(7-methoxy-4-methylquinazolin-2-yl)piperidin-3-ol
3-phenoxy-N-[1-(1-{spiro[2.4]heptane-1-carbonyl}piperidin-4-yl)-1H-pyrazol-5-yl]propanamide