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6-(3,3-diphenylpiperidine-1-carbonyl)-1,3-dimethyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-[(9aS)-octahydro-1H-pyrrolo[1,2-a][1,4]diazepine-2-carbonyl]-6-ethyl-1,5-dimethyl-1,2-dihydropyridin-2-one
4-{thieno[2,3-d]pyrimidin-4-yl}piperazine-2-carboxylic acid
N-[2-(3-fluorophenyl)ethyl]-2-{4-[4-({2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}amino)piperidin-1-yl]phenyl}acetamide
4-{2-[2-(3-methylthiophen-2-yl)-1H-imidazol-1-yl]ethyl}benzene-1-sulfonamide
1-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-4-(4-fluorophenyl)-1,4-diazepane
1-{3-[4-(4-fluorophenyl)piperazin-1-yl]piperidin-1-yl}-2,2,3-trimethylbut-3-en-1-one
3-[1-(3-methylbut-2-en-1-yl)piperidin-3-yl]-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
[1-({1-[3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]piperidin-4-yl}methyl)-1H-1,2,3-triazol-4-yl]methanol
N-(2-{5-[(cyclohexylmethyl)sulfanyl]-4-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl}ethyl)thiophene-2-carboxamide
N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-2-(dimethylamino)-2-(2-fluorophenyl)-N-methylacetamide
N-[(4-hydroxyazepan-4-yl)methyl]-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
2-(1-benzofuran-2-carbonyl)-7-[(2-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decane
1-(5-chloropyrimidin-2-yl)-4-[(2-methylpyridin-3-yl)oxy]piperidine-4-carboxylic acid
N-cyclohexyl-N-(2-hydroxy-2-phenylethyl)-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-3-(morpholin-4-yl)propanamide
1-(propan-2-yl)-N-[1-(1-propyl-1H-1,2,4-triazol-5-yl)ethyl]piperidine-4-carboxamide
11-(2,3-dimethyl-1H-indole-5-carbonyl)-3,7-dimethyl-3,7,11-triazaspiro[5.6]dodecane
4-(1H-pyrazol-4-yl)-N-[2-(pyridin-3-yl)-5,6,7,8-tetrahydroquinazolin-5-yl]butanamide
N,N,4-trimethyl-3-({methyl[1-methyl-1-(methylcarbamoyl)ethyl]carbamoyl}methyl)-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
5-(4-cyclohexyl-1,4-diazepane-1-carbonyl)-N,N,4-trimethylpyrimidin-2-amine
N-(2-{2-[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]-1H-imidazol-1-yl}ethyl)-N-methylmethanesulfonamide
N-[(4-hydroxy-6-methylpyrimidin-2-yl)methyl]-2-methyl-1,3-thiazole-4-carboxamide
N-(2-ethoxyethyl)-5-(1-{[5-(hydroxymethyl)furan-2-yl]methyl}pyrrolidin-2-yl)thiophene-2-carboxamide
N-methyl-3-{1-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]piperidin-3-yl}-N-[2-(pyridin-2-yl)ethyl]propanamide
dimethyl[1-(3-{1-[2-(pyrrolidin-1-yl)ethyl]-1H-1,2,3-triazol-4-yl}phenyl)ethyl]amine
2-[1-(4-hydroxy-3-methylbenzoyl)pyrrolidin-3-yl]benzoic acid
N-(1-{1-[(2,5-dimethoxyphenyl)methyl]piperidin-4-yl}-2-(2-fluorophenyl)ethyl)-N-methylthiophene-2-carboxamide
1-(furan-2-ylmethyl)-N-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}piperidine-4-carboxamide
4-[1-(4-methylphenyl)-3-(phenoxymethyl)-1H-1,2,4-triazol-5-yl]pyrrolidin-2-one
4-(1,3-dimethyl-1H-pyrazol-4-yl)-N-[2-(methylsulfanyl)ethyl]pyrimidin-2-amine
1-[2-amino-7-(1,3-thiazol-2-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]piperidine-3-carbonitrile
1-(5-methyl-1,3-benzoxazol-2-yl)-3-(piperidin-1-ylmethyl)pyrrolidin-3-ol
2-(cyclopropylmethyl)-8-[2-(2-ethyl-1H-imidazol-1-yl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
1-methanesulfonyl-3-(4-phenoxybenzoyl)piperidine
2-[(4-chlorophenyl)amino]-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}acetamide
N-[1-(pyrazin-2-yl)propan-2-yl]cyclohex-3-ene-1-carboxamide
N-[(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)methyl]-2-(2,5-dioxo-1-propylimidazolidin-4-yl)acetamide
3-(3-methyl-1H-1,2,4-triazol-5-yl)-N-{4-[(trifluoromethyl)sulfanyl]phenyl}piperidine-1-carboxamide
N-[2-(2-ethoxyphenyl)ethyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
N-tert-butyl-1-cyclohexyl-4-oxo-5-[4-(pyridin-4-ylmethyl)piperazine-1-carbonyl]-1,4-dihydropyridine-3-carboxamide
(3S,4S)-1-[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl]-4-(dimethylamino)piperidin-3-ol
N-[2-(diethylamino)ethyl]-N-methyl-5-(propan-2-yl)-1-[4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
3,7-dimethyl-11-{[5-(oxan-2-yl)furan-2-yl]methyl}-3,7,11-triazaspiro[5.6]dodecane
2-(dimethyl-1,2-oxazol-4-yl)-N-(2-methyl-1,3-benzothiazol-5-yl)pyrrolidine-1-carboxamide
3-[(2,4-difluorophenyl)methyl]-1-(2,5-dimethylpyrimidin-4-yl)piperidine-3-carboxylic acid
2-(5-methyl-1H-pyrazol-1-yl)-1-{4-[4-methyl-5-(morpholin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}ethan-1-one
1-methyl-2-oxo-8-{[3-(trifluoromethyl)phenyl]methyl}-1,8-diazaspiro[4.5]decane-4-carboxylic acid
3-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-6-(propan-2-yloxy)pyridazine
N-[3-(3-{[4-(2,3-dimethylphenyl)piperazin-1-yl]methyl}phenoxy)propyl]-4-methylbenzamide