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2-(2-methoxyethyl)-9-[2-(propan-2-yl)pyrimidine-5-carbonyl]-2,9-diazaspiro[5.5]undecan-3-one
N-[(6-hydroxy-2-methylpyrimidin-4-yl)methyl]-2-(1-propylpiperidin-4-yl)acetamide
N-[(6-methylpyridin-2-yl)methyl]-1H-indole-6-carboxamide
N-{[2-(1H-imidazol-1-yl)phenyl]methyl}-2-(2-oxo-1,2-dihydropyridin-1-yl)acetamide
4-(2,3-dihydro-1H-inden-5-yloxy)-1-(pyridin-2-ylmethyl)piperidine-4-carboxylic acid
4-(3-cyclopropyl-1H-1,2,4-triazol-5-yl)-6-fluoro-1,2,3,4-tetrahydroquinolin-2-one
2-(4-chloro-3-methyl-1H-pyrazol-1-yl)-1-[3-(hydroxymethyl)-3-(2-methoxyethyl)piperidin-1-yl]ethan-1-one
N-[3-(1H-imidazol-1-yl)propyl]-3-{[(4-methoxyphenyl)methyl]amino}-5-(pyrrolidine-1-sulfonyl)benzamide
methyl 1-[(3R,5S)-1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-5-[(2-phenylethyl)carbamoyl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
1-(2-ethoxyphenyl)-3-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]urea
8-(5-methyl-1,3-oxazole-4-carbonyl)-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-(2-chloro-4,5-difluorophenyl)-1-[3-(hydroxymethyl)-3-(prop-2-en-1-yl)piperidin-1-yl]ethan-1-one
3-{[2-(1-{thieno[3,2-d]pyrimidin-4-yl}piperidin-4-yl)-1H-imidazol-1-yl]methyl}pyridine
2-(2-methyl-1H-imidazol-1-yl)-N-[1-phenyl-3-(propan-2-yl)-1H-pyrazol-5-yl]acetamide
[4-({[(2,3-difluoro-6-methoxyphenyl)methyl](methyl)amino}methyl)oxan-4-yl]methanol
8-(2-amino-2-methylpropanoyl)-3-{2-[(2-methoxyethyl)(methyl)amino]ethyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[2-(morpholin-4-yl)butyl]-3-(pyridin-2-yl)-1H-pyrazole-5-carboxamide
2-(furan-2-yl)-7-methyl-N-[1-(1H-pyrazol-1-yl)propan-2-yl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
8-(3,5-difluoropyridine-2-carbonyl)-2-[2-(dimethylamino)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
5,7-dimethyl-2-(1-propyl-1H-pyrazol-4-yl)-4-(pyrrolidine-1-carbonyl)quinoline
1-{[5-(1-cyclopropanecarbonylpiperidin-4-yl)-4-methyl-4H-1,2,4-triazol-3-yl]methyl}azepane
N-cyclopropyl-1-[4-(1H-pyrazol-4-yl)butanoyl]piperazine-2-carboxamide
1-(2,3-dimethylphenyl)-N-{[3-(ethoxymethyl)-4-methoxyphenyl]methyl}-4,5,6,7-tetrahydro-1H-indazol-4-amine
1-(1-cyclohexanecarbonylpyrrolidine-2-carbonyl)imidazolidin-4-one
[(3R,4R)-1-(4,6-dimethoxypyrimidin-2-yl)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}pyrrolidin-3-yl]methanol
methyl[(1-methyl-1H-imidazol-2-yl)methyl][(3-phenyl-1,2-oxazol-5-yl)methyl]amine
N-(3-cyclopentaneamidophenyl)-3-oxopiperazine-1-carboxamide
2-(3-methoxyphenyl)-1-(4-propylbenzoyl)azetidine
4-[(2,2-difluoroethyl)sulfamoyl]-N-[(3-methyl-1,2-oxazol-5-yl)methyl]benzamide
2-benzyl-8-[3-oxo-3-(pyrrolidin-1-yl)propyl]-2,8-diazaspiro[5.5]undecan-3-one
2,8-dimethyl-N-[(1-methylpiperidin-3-yl)methyl]quinoline-3-carboxamide
8-[(5-chloro-2,3-dimethoxyphenyl)methyl]-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-cyclopropyl-1-[1-(3-phenylpropyl)piperidin-4-yl]piperidine-3-carboxamide
N-(1-hydroxybutan-2-yl)-1-propyl-N-(thiophen-3-ylmethyl)-1H-pyrazole-5-carboxamide
1-[(3-fluorophenyl)methyl]-N-[3-(methylsulfanyl)propyl]-6-oxopiperidine-3-carboxamide
N-methyl-N-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
3-(2-{3-[4-(4-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}-2-oxoethyl)-1,3-oxazolidin-2-one
8-methyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxamide
(3aR,6aR)-N-{imidazo[1,2-a]pyridin-3-ylmethyl}-2-(2-methoxyacetyl)-N-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
4-[2-(benzyloxy)ethyl]-1,3λ6,4-oxathiazinane-3,3-dione
ethyl 2-({2-[2-(dimethylamino)ethyl]morpholine-4-carbonyl}amino)acetate
N-[2-(dimethylamino)-2-(3-methylphenyl)ethyl]-3-methoxy-2,2-dimethylpropanamide
2-{3-cyclopentyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-3-(pyrrolidine-1-carbonyl)pyridine
3-(2H-1,3-benzodioxol-5-yl)-5-[2-(1H-pyrazol-4-yl)ethyl]-1,2,4-oxadiazole
1-acetyl-N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}piperidine-3-carboxamide
2-({2-amino-6-[3-(1H-1,3-benzodiazol-2-yl)piperidin-1-yl]pyrimidin-4-yl}amino)ethan-1-ol
N-[(2-methoxyphenyl)methyl]-3-(pyridin-4-yl)-N-(pyridin-4-ylmethyl)propanamide
2-(2,4-difluorophenoxy)-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}propanamide
N-(2-cyclobutyl-1-methyl-5-{4H,5H,6H,7H-thieno[3,2-c]pyridine-5-carbonyl}-1H-1,3-benzodiazol-7-yl)oxolane-2-carboxamide
5-methyl-2-(quinolin-6-yl)pyrimidin-4-amine