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11-(2-chloropyridine-4-carbonyl)-3,7-dimethyl-3,7,11-triazaspiro[5.6]dodecane
N-({7-[(2E)-3-(2,3-difluorophenyl)prop-2-enoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)thiophene-3-sulfonamide
(3S)-1-[6-(methoxymethyl)-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-N,N-dimethylpyrrolidin-3-amine
3-({[2-(dimethylamino)-6-ethylpyrimidin-4-yl]amino}methyl)-1λ6-thiolane-1,1-dione
[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl][2-(1H-imidazol-1-yl)ethyl]methylamine
5-{4-[2-(methylsulfanyl)ethyl]piperazine-1-carbonyl}-2-(pyridin-3-yl)pyrimidine
(3aS,6aS)-2-cyclopentanecarbonyl-5-[2-(3-fluorophenyl)ethyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-(3-hydroxy-3-methylbutyl)-N-[2-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)propyl]benzamide
4-[(3-phenyl-1,2-oxazol-5-yl)methyl]-1-[3-(1H-pyrazol-1-yl)propyl]piperidin-4-ol
3-(3-hydroxy-3-methylbutyl)-N-methyl-N-[2-(4-methyl-1H-1,3-benzodiazol-2-yl)ethyl]benzamide
(3R,4S)-1-{[4-(3-hydroxyprop-1-yn-1-yl)phenyl]methyl}-3,4-dimethylpiperidin-4-ol
1-tert-butyl-4-[4-(2-fluorophenyl)-1H-imidazol-2-yl]pyrrolidin-2-one
N-[(5-methyl-1H-1,3-benzodiazol-2-yl)methyl]-2-(4-oxo-3,4-dihydroquinazolin-3-yl)acetamide
N-{1-[4-(dimethylamino)phenyl]-3-hydroxypropan-2-yl}-6-methylimidazo[1,2-a]pyridine-2-carboxamide
6-[furan-2-yl(phenyl)methyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
2-{5-[(3-methyl-6-oxo-1,6-dihydropyridazin-1-yl)methyl]-3-[(1-methylpiperidin-4-yl)methyl]-1H-1,2,4-triazol-1-yl}acetic acid
(1S,5R)-3-[(5-propylfuran-2-yl)methyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
4-[(1-{1-[(2-chloro-4-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperidin-3-yl)methyl]morpholine
2-(2-hydroxyethyl)-8-[(5-methoxy-1H-indazol-3-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
3-{[1-(hydroxymethyl)cyclopropyl]methyl}-3-methyl-1-{3-[(trifluoromethyl)sulfanyl]phenyl}urea
1-[5-(methoxymethyl)furan-2-carbonyl]-2-(3-methoxyphenyl)azetidine
5-{3-[(4-methoxyphenyl)methyl]-1,2,4-oxadiazol-5-yl}-N-[2-(1H-pyrazol-1-yl)ethyl]pyridin-2-amine
3-(6-methoxypyridin-3-yl)-6-methyl-4H-chromen-4-one
N-[cyclopropyl(3-methylpyridin-2-yl)methyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
3-[(2-methoxyethyl)(methyl)sulfamoyl]-N-(oxan-3-ylmethyl)benzamide
(1S,5R)-3-[3-(3-methoxyphenoxy)propyl]-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
1-(adamantan-1-yl)-4-(oxolane-3-carbonyl)piperazine
6-propyl-2-(4-{[4-(pyrazin-2-yl)piperazin-1-yl]methyl}phenyl)-3,4-dihydropyrimidin-4-one
N-({5-[(3-chloro-4-fluorophenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)cyclobutanecarboxamide
5-cyclopentyl-3-({4-[2-(methylsulfanyl)propyl]-1H-1,2,3-triazol-1-yl}methyl)-1,2,4-oxadiazole
2-benzyl-9-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-2,9-diazaspiro[5.5]undecan-3-one
(3aR,6aR)-2-[(4-acetyl-1-methyl-1H-pyrrol-2-yl)methyl]-5-(cyclobutylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
8-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)acetyl]-2-ethyl-2,8-diazaspiro[4.5]decan-3-one
8-[(5-chloro-2-fluorophenyl)methyl]-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
2-({2-[1-(ethanesulfonyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
5-[2,2-bis(prop-2-en-1-yl)pyrrolidine-1-carbonyl]-1-[3-(2-oxopyrrolidin-1-yl)propyl]piperidin-2-one
(1S,5R)-6-(2,3-dihydro-1H-indene-5-carbonyl)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
4-benzyl-1-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propyl]-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-1H-indole-7-carboxamide
({4-[(dimethylamino)methyl]thiophen-2-yl}methyl)(methyl)[(trimethyl-1H-pyrazol-4-yl)methyl]amine
1-benzyl-5-[(cyclohexylmethyl)amino]-N,N-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-(1-{6-methylimidazo[1,2-a]pyridine-2-carbonyl}piperidin-3-yl)-1,3-benzoxazole
N-{1-[1-(carbamoylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
1-[(2-methoxyphenyl)methyl]-N-methyl-N-[2-(oxan-4-yl)ethyl]-6-oxopiperidine-3-carboxamide
(1R,3S)-3-methoxy-3-methyl-7-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)-7-azaspiro[3.5]nonan-1-ol
4-[4-(3-{[4-(hydroxymethyl)phenyl]methyl}pyrrolidine-1-carbonyl)phenyl]-2-methylbutan-2-ol
(3S,4S)-4-propyl-1-[2-(2H-1,2,3,4-tetrazol-2-yl)acetyl]pyrrolidine-3-carboxylic acid
1-(carbamoylmethyl)-N-[3-(1H-1,2,3-triazol-1-yl)propyl]piperidine-3-carboxamide
3-(2-methoxybenzoyl)piperidine
{1-[(2,4,5-trimethylphenyl)methyl]pyrrolidin-3-yl}methanamine