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3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]-1-(5-fluoro-2-methylbenzoyl)piperidine
N3-{2-[({5-[(dimethylamino)methyl]furan-2-yl}methyl)sulfanyl]ethyl}piperidine-1,3-dicarboxamide
({3-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]phenyl}methyl)(methyl)(quinolin-5-ylmethyl)amine
5-[3-(benzyloxy)propyl]-3-(oxan-4-yl)-1H-1,2,4-triazole
1-[4-(2-{4-[(dimethylamino)methyl]phenyl}piperidine-1-carbonyl)thiophen-2-yl]ethan-1-one
methyl (2S,4R)-1-methyl-4-(4,5,6,7-tetrahydro-2H-indazole-3-amido)pyrrolidine-2-carboxylate
N,N-dimethyl-3-{[4-(pyrimidin-4-yl)piperidin-1-yl]sulfonyl}benzamide
11-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-3,7-dimethyl-3,7,11-triazaspiro[5.6]dodecane
1-butyl-4-[2-(dimethylamino)-2-(4-fluorophenyl)acetyl]piperazin-2-one
N-[5-(2H-1,3-benzodioxol-5-yl)pyridin-2-yl]methanesulfonamide
2-(2-hydroxyethyl)-6-(6-phenylpyridazin-3-yl)-1H,2H,3H,4H,5H,6H,7H-pyrazolo[3,4-c]pyridin-3-one
N-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-N,2-dimethyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-[1-(3,4-dimethylphenyl)propyl]-2-(2-oxopiperidin-1-yl)acetamide
1-(pyridin-3-ylmethyl)-4-(1,3-thiazol-4-ylmethyl)-1,4-diazepane
3-[(5-methylpyrazin-2-yl)methyl]-1-[2-(propan-2-yloxy)phenyl]urea
2-{N-methyl-1-[1-(propan-2-yl)piperidin-4-yl]formamido}-2-(pyridin-3-yl)acetic acid
4-[4-(7-chloro-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl)phenyl]-2-methylbutan-2-ol
[(5-tert-butyl-1H-pyrazol-3-yl)methyl][(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]methylamine
4-(dimethyl-1,3-thiazol-5-yl)-N-(pyridin-3-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
1-(1H-imidazol-4-ylmethyl)-N-[4-(3-methylphenyl)phenyl]piperidine-4-carboxamide
(3E)-5,5-dimethyl-2-[methyl(pyridin-3-ylmethyl)amino]hex-3-enoic acid
2-[4-phenyl-5-(2-phenylethyl)-1H-imidazol-1-yl]acetamide
N-[(3S)-1-benzylpyrrolidin-3-yl]-3-(1-methyl-1H-pyrazol-5-yl)propanamide
3-{2-[4-(4-fluorophenyl)-1,2,3,6-tetrahydropyridin-1-yl]-2-oxoethyl}-4-[(2-fluorophenyl)methyl]piperazin-2-one
(3R,4R)-1-[(5-ethylpyridin-2-yl)methyl]-3-methyl-4-(oxan-4-yl)piperidin-4-ol
2-[6-hydroxy-4-(oxan-4-yl)-1,4-diazepan-1-yl]-N-(5-methyl-1,2-oxazol-3-yl)acetamide
2-(3-{[4-cyclopentyl-3-(2-hydroxyethyl)piperazin-1-yl]methyl}phenoxy)ethan-1-ol
2-(3-methyl-1H-pyrazol-1-yl)-1-{4-[(oxolan-3-yl)amino]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl}ethan-1-one
(2-{2-[1-(4-methoxy-3-methylbenzoyl)piperidin-3-yl]-1H-imidazol-1-yl}ethyl)dimethylamine
N-({3-[2-(2-fluorophenyl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]thiophene-2-sulfonamide
3-[1-(adamantan-1-yl)piperidin-4-yl]-1-(pyrrolidin-1-yl)propan-1-one
2-methyl-5-(2-{3-[2-(2-methylphenyl)ethyl]piperidin-1-yl}-2-oxoethyl)-3,4-dihydropyrimidin-4-one
2-[3-methoxy-4-(pyrrolidin-1-ylmethyl)phenoxy]-3-(trifluoromethyl)pyridine
2-({[2-(cyclohex-1-en-1-yl)ethyl]amino}methyl)-4-(pyrimidin-5-yl)phenol
1-cyclohexyl-N3-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-N5-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
2-methyl-N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)benzamide
3-(azepane-1-carbonyl)-N-[(2-methoxyphenyl)methyl]-1-methyl-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-[(4-benzylpiperazin-1-yl)methyl]-N-(1,4-dioxan-2-ylmethyl)-N-methyl-1,3-oxazole-4-carboxamide
4-(1-ethyl-1H-pyrazole-4-carbonyl)-6-[(3-fluorophenyl)methoxy]-1-(2-methylpropyl)-1,4-diazepan-2-one
N-(3-hydroxypropyl)-3-(piperidin-3-yl)-N-(pyridin-4-ylmethyl)benzamide
[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl](2-methylpropyl)(pyridin-2-ylmethyl)amine
(1R,5R)-3-[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl]-3-azabicyclo[3.3.1]nonane
2-[4-({4-[(4-fluorophenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}methyl)phenoxy]ethan-1-ol
N-{2-methyl-5-[(propan-2-yl)carbamoyl]phenyl}-4-(pyridin-4-yl)piperazine-1-carboxamide
ethyl 1-(3-fluorophenyl)-5-{[3-(4-methyl-4H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}-1H-pyrazole-4-carboxylate
2-{4-[(2-butyl-1H-imidazol-4-yl)methyl]-1-[(3,4-difluorophenyl)methyl]piperazin-2-yl}ethan-1-ol
(1R,7S)-6-(2,3-dihydro-1H-isoindole-2-carbonyl)-3-[(5-methylpyrazin-2-yl)methyl]-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
1-[3-(2-ethyl-2,5-dihydro-1H-pyrrol-1-yl)-3-oxopropyl]-6-methyl-1,2-dihydropyridin-2-one
2-(5-tert-butyl-2H-1,2,3,4-tetrazol-2-yl)-N-[1-(4-methoxyphenyl)-3-methyl-1H-pyrazol-5-yl]acetamide
2-[(4aR,7aS)-6,6-dioxo-4-(quinolin-4-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]acetic acid