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3-[(1R,5S)-6-azabicyclo[3.2.1]octane-6-carbonyl]-N-(1H-imidazol-2-ylmethyl)benzene-1-sulfonamide
2-[({5-[1-(5-ethyl-1,2,4-oxadiazol-3-yl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)(methyl)amino]ethan-1-ol
2-[4-(2H-1,3-benzodioxol-5-yl)-3-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl]-N-[2-(ethylsulfanyl)ethyl]acetamide
2-{[benzyl(1,1-dioxo-1λ6-thiolan-3-yl)amino]methyl}pyridine-3-carboxylic acid
(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)(methyl){[5-methyl-2-(5-methylfuran-2-yl)-1,3-oxazol-4-yl]methyl}amine
2-amino-4-[3,5-dimethyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]-6-(3-hydroxyphenyl)pyridine-3-carbonitrile
1-{[5-(methoxymethyl)furan-2-yl]methyl}-N-[4-(pyridin-3-yloxy)phenyl]piperidine-2-carboxamide
(5S,9aS,9bS)-5-(2,5-difluorophenyl)-2-[(4-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-cyclohexyl-2-{[(3-ethyl-1,2-oxazol-5-yl)methyl](methyl)amino}butanamide
4,6-dimethyl-1-(2-{[1-methyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}ethyl)-1,2-dihydropyrimidin-2-one
4-(1,3-dimethyl-1H-pyrazol-4-yl)-2-[4-(2-phenylethyl)piperazin-1-yl]pyrimidine
N-cyclopentyl-1-(2-methylpropyl)-5-[3-(pyridin-4-yl)propanoyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
3-(4-methyl-1,3-thiazol-5-yl)-1-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}propan-1-one
(3aS,6aS)-1-oxo-2-(prop-2-en-1-yl)-5-{thieno[2,3-d]pyrimidin-4-yl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-3-one
N-[(1-benzylpiperidin-4-yl)methyl]-2-[4-(hydroxymethyl)phenyl]-N-methylacetamide
N-cyclopentyl-2-(1,1-dioxo-1λ6-thiolan-3-yl)-N-propylacetamide
1-{1'-[(2-methoxy-4-methylphenyl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}propan-1-one
5-hydroxy-1,2-dimethyl-N-[(1r,4r)-4-(4H-1,2,4-triazol-4-yl)cyclohexyl]-1H-indole-3-carboxamide
(3S,4R)-4-(2,3-dimethoxyphenyl)-1-(5-methylthiophene-2-carbonyl)pyrrolidine-3-carboxylic acid
N-ethyl-2-(5-fluoro-2-methoxyphenyl)pyridine-4-carboxamide
5-(3-oxo-3-{4-[(pyridin-2-yl)amino]piperidin-1-yl}propyl)imidazolidine-2,4-dione
N-[1-(2,3-dihydro-1H-inden-2-yl)-5-oxopyrrolidin-3-yl]-2-(2,5-dimethylphenyl)acetamide
(3R,4R)-N-cyclohexyl-4-hydroxy-4-(2-methoxyethyl)-3-methylpiperidine-1-carboxamide
2-[4-(1,2-oxazol-3-ylmethyl)-1-(propan-2-yl)piperazin-2-yl]ethan-1-ol
(1S,5R)-3-(4-oxo-4-phenylbutyl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-{1-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}pyridine
6-methoxy-4-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]-1,2,3,4-tetrahydroquinolin-2-one
1-[(3aS,6aS)-1-(piperidine-1-carbonyl)-octahydropyrrolo[3,4-b]pyrrol-5-yl]-2-[(3-amino-1H-1,2,4-triazol-5-yl)sulfanyl]ethan-1-one
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-2-(thiophen-2-yl)pyrimidine-5-carboxamide
9-methoxy-7-(8-methoxy-4-methylquinolin-2-yl)-4-[(1-methyl-1H-pyrrol-2-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-[(4-fluorophenyl)methyl]-N-[(1R)-2-hydroxy-1-phenylethyl]-1H-1,2,3-triazole-4-carboxamide
3-(3-chlorophenyl)-N-[(5-methyl-4H-1,2,4-triazol-3-yl)methyl]-3-phenylpropanamide
2-{2-[1-(5-phenyl-1,2-oxazole-3-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}acetamide
4-phenoxy-1-{[(1s,4s)-4-aminocyclohexyl]methyl}piperidine-4-carboxylic acid
7-methanesulfonyl-N,4-dimethyl-N-[(1-methylpiperidin-3-yl)methyl]quinazolin-2-amine
1-methyl-N-{[1-(4-methylpiperazin-1-yl)cyclohexyl]methyl}-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)(methyl){[3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}amine
1-(2-{2-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}pyrimidin-4-yl)pyrrolidin-3-ol
4-amino-N-[(5-methylthiophen-2-yl)methyl]-N-(prop-2-en-1-yl)pyridine-2-carboxamide
{1-[1-(3,5,7-trimethyl-1H-indole-2-carbonyl)piperidin-3-yl]piperidin-4-yl}methanol
3-(1-ethyl-1H-1,2,3-triazol-4-yl)-1-[2-(2-oxoimidazolidin-1-yl)ethyl]urea
{[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}[(4-methanesulfonylmorpholin-2-yl)methyl]amine
dimethyl({4-[1-(morpholine-4-carbonyl)piperidin-2-yl]phenyl}methyl)amine
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-6-(methoxymethyl)pyridine-2-carboxamide
(3S,5R)-1-(2-phenylacetyl)-5-[(pyridin-3-ylmethyl)carbamoyl]piperidine-3-carboxylic acid
4-[4-(3,6-dimethylpyrazin-2-yl)piperazine-1-carbonyl]-6-methyl-1,2-dihydropyridin-2-one
2-{[2-(5-chloro-2-methoxyphenyl)-5-fluoropyrimidin-4-yl]amino}ethan-1-ol
2-{8-[2-(dimethylamino)ethyl]-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}-N-methylpyridine-4-carboxamide
methyl 1-benzyl-5-{[(2E)-2-methylbut-2-en-1-yl]amino}-3-(pyridine-3-amido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate