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2-cyclopropyl-8-{2-[methyl(pyridin-2-ylmethyl)amino]acetyl}-2,8-diazaspiro[5.5]undecan-3-one
[3-(1H-imidazol-2-yl)-2,4,6-trimethylphenyl]methyl acetate
2-(3-fluorophenyl)-1-(3-propyl-1H-pyrazole-4-carbonyl)piperidine
5-methoxy-3-methyl-2-[3-(pyridin-3-yl)azetidine-1-carbonyl]-1H-indole
5-cyclobutanecarbonyl-2-(2,4-difluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
3-(4-fluorophenyl)-1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-1-yl]propan-1-one
1-(1-{3-[(2-methyl-1H-imidazol-1-yl)methyl]piperidin-1-yl}propan-2-yl)-1H-1,3-benzodiazole
3-{2-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]-2-oxoethyl}-4-(propan-2-yl)piperazin-2-one
N-{1-[2-(4-methoxyphenyl)ethyl]-5-oxopyrrolidin-3-yl}-2-methyl-1,3-thiazole-4-carboxamide
N-(2-methoxyethyl)-1-{1-[6-methyl-2-(methylamino)pyrimidin-4-yl]piperidin-4-yl}piperidine-3-carboxamide
2-[(3,4-difluorophenyl)methyl]-8-[2-(propan-2-yloxy)acetyl]-2,8-diazaspiro[4.5]decan-3-one
2-{[1-butyl-3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]methyl}-1,4-dimethylpiperazine
4-(2,6-dimethylquinoline-3-carbonyl)-3-(4-fluorophenyl)piperazin-2-one
(2S)-2-[(4,6-dimethylpyrimidin-2-yl)amino]-2-phenylethan-1-ol
2-ethyl-7-methoxy-4-{[4-(pyrimidin-2-yloxy)phenyl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
(2S,4R)-1-[(4-chlorophenyl)methyl]-4-{[(3,4-difluorophenyl)methyl]amino}-N-(propan-2-yl)pyrrolidine-2-carboxamide
N-[1-(3-cyano-6-methylpyridin-2-yl)piperidin-4-yl]methanesulfonamide
1-(6-methyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-4-phenoxypiperidine-4-carboxylic acid
N-(3-{[4-(hydroxymethyl)-4-(2-phenylethyl)piperidin-1-yl]sulfonyl}phenyl)acetamide
4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(1,3-thiazol-2-yl)piperidine
6-oxo-N-{2-[4-(propan-2-yloxy)phenyl]ethyl}-1-[2-(pyridin-2-yl)ethyl]piperidine-3-carboxamide
7-ethyl-3-(1-ethyl-5-methyl-1H-pyrazol-4-yl)-2,4,5,7-tetraazatricyclo[6.4.0.02,6]dodeca-1(12),3,5,8,10-pentaene
4-({methyl[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]carbamoyl}amino)-N-(oxolan-2-ylmethyl)benzamide
N-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-2-{8-methoxy-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}acetamide
[(3R,4R)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-(4-methyl-1H-imidazole-2-carbonyl)pyrrolidin-3-yl]methanol
4-(1-methyl-1H-imidazol-2-yl)-1-{2-[(4-methylphenyl)methyl]benzoyl}piperidine
4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}-N-(thiophen-2-ylmethyl)benzamide
4-(2-benzyl-1,3-thiazole-4-amido)oxane-4-carboxylic acid
3-(5-fluoro-1H-1,3-benzodiazol-2-yl)-N-methyl-N-[1-(pyridin-3-yl)propyl]propanamide
2-{[4-(2-methoxyphenyl)-5-(pyridin-4-yl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
N4-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-N4,N6,N6-trimethylpyrimidine-4,6-diamine
1-acetyl-N-{2-[methyl(phenyl)amino]propyl}piperidine-4-carboxamide
methyl 3-(2,3-dihydro-1,4-benzodioxine-6-sulfonamido)-5-[(2-ethylbutanamido)methyl]benzoate
1-[2-(4-methoxyphenyl)ethyl]-N,N-dimethyl-5-(thiophen-3-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-{4-[(4aS,7aS)-octahydro-1H-pyrrolo[3,4-b]pyridin-6-yl]-6-methylpyrimidin-2-yl}phenol
2-[1-cyclohexyl-5-(3-ethyl-1H-pyrazol-4-yl)-1H-1,2,4-triazol-3-yl]acetamide
N,N-dimethyl-5-{[8-(6-methylpyridin-2-yl)-1,8-diazaspiro[4.5]decan-1-yl]methyl}pyrimidin-2-amine
2-[(1S,5R)-3-(dimethyl-1,3-thiazole-5-carbonyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
3-(1,3-benzothiazol-2-yl)-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}propanamide
(4S,4aS,8aS)-1-(6-aminopyridine-3-carbonyl)-4-phenyl-decahydroquinolin-4-ol
(3S,9aR)-8-[(3,4-difluorophenyl)methyl]-3-[(4-hydroxyphenyl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-(7-chloro-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-2-(pyridin-4-ylsulfanyl)ethan-1-one
(3R,4R)-4-amino-1-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]piperidin-3-ol
3-[(5-fluoro-2-methoxyphenyl)methyl]-9-methyl-3,9-diazaspiro[5.6]dodecane
1-[5-(cyclohex-1-en-1-yl)-1H-1,3-benzodiazol-2-yl]ethan-1-ol
{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}(methyl)(quinolin-5-ylmethyl)amine
6-[(diethylamino)methyl]-N-[(1-methyl-5-oxopyrrolidin-2-yl)methyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
6-ethyl-2-[1-(propan-2-yl)-1H-pyrazol-4-yl]-4-(pyrrolidine-1-carbonyl)quinoline
4-methyl-6-{4-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]piperazin-1-yl}pyrimidin-2-amine
2-({[4-(butan-2-yloxy)-3-chlorophenyl]methyl}[(1-methyl-1H-imidazol-2-yl)methyl]amino)ethan-1-ol